PT778277E - Derivados heterociclicos substituidos como antagonistas do crf - Google Patents

Derivados heterociclicos substituidos como antagonistas do crf

Info

Publication number
PT778277E
PT778277E PT96308092T PT96308092T PT778277E PT 778277 E PT778277 E PT 778277E PT 96308092 T PT96308092 T PT 96308092T PT 96308092 T PT96308092 T PT 96308092T PT 778277 E PT778277 E PT 778277E
Authority
PT
Portugal
Prior art keywords
antagonists
crta
heterocyclic derivatives
derivatives substituted
chem
Prior art date
Application number
PT96308092T
Other languages
English (en)
Inventor
Yuhpyng L Chen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT778277E publication Critical patent/PT778277E/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P5/10—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH
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    • A—HUMAN NECESSITIES
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    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Transplantation (AREA)
  • Emergency Medicine (AREA)
  • Anesthesiology (AREA)
  • Oncology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Addiction (AREA)
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PT96308092T 1995-12-08 1996-11-07 Derivados heterociclicos substituidos como antagonistas do crf PT778277E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US839695P 1995-12-08 1995-12-08

Publications (1)

Publication Number Publication Date
PT778277E true PT778277E (pt) 2003-11-28

Family

ID=21731406

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96308092T PT778277E (pt) 1995-12-08 1996-11-07 Derivados heterociclicos substituidos como antagonistas do crf

Country Status (9)

Country Link
EP (1) EP0778277B1 (pt)
JP (2) JP3457490B2 (pt)
AT (1) ATE243697T1 (pt)
CA (1) CA2192289C (pt)
DE (1) DE69628804T2 (pt)
DK (1) DK0778277T3 (pt)
ES (1) ES2200039T3 (pt)
MX (1) MX9606203A (pt)
PT (1) PT778277E (pt)

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DK0778277T3 (da) 2003-10-27
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DE69628804D1 (de) 2003-07-31
MX9606203A (es) 1998-04-30
CA2192289A1 (en) 1997-06-09
JP3457490B2 (ja) 2003-10-20
EP0778277B1 (en) 2003-06-25
JP2000109431A (ja) 2000-04-18
CA2192289C (en) 2001-02-20
ES2200039T3 (es) 2004-03-01
DE69628804T2 (de) 2003-12-18
ATE243697T1 (de) 2003-07-15

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