PT85547A - Processo de preparacao de composicao farmaceuticas a base de derivados de 2-mercapto-imidazol e de preparacao destes derivados - Google Patents

Processo de preparacao de composicao farmaceuticas a base de derivados de 2-mercapto-imidazol e de preparacao destes derivados

Info

Publication number: PT85547A
Authority: PT; Portugal
Prior art keywords: derivatives; mercapto; preparation; pharmaceutical compositions; compositions based
Prior art date: 1986-08-18

Application number

PT85547A

Other languages

English (en)

Other versions

PT85547B (pt

Inventor

Lawrence Ivan Kruse

Joseph Alan Finkelstein

James Simpson Frazee

Thomas Brent Leonard

Carl Kaiser

Original Assignee

Smithkline Beecham Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-08-18

Filing date

1987-08-17

Publication date

1988-08-17

1987-08-17 Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp

1988-08-17 Publication of PT85547A publication Critical patent/PT85547A/pt

1995-03-01 Publication of PT85547B publication Critical patent/PT85547B/pt

Links

OXFSTTJBVAAALW-UHFFFAOYSA-N 1,3-dihydroimidazole-2-thione Chemical class SC1=NC=CN1 OXFSTTJBVAAALW-UHFFFAOYSA-N 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1
241000124008 Mammalia Species 0.000 abstract 1
230000000694 effects Effects 0.000 abstract 1
239000003112 inhibitor Substances 0.000 abstract 1
230000003389 potentiating effect Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/84—Sulfur atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Enzymes And Modification Thereof (AREA)
Plural Heterocyclic Compounds (AREA)

PT85547A 1986-08-18 1987-08-17 Processo de preparacao de composicao farmaceuticas a base de derivados de 2-mercapto-imidazol e de preparacao destes derivados PT85547B (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US89816586A	1986-08-18	1986-08-18

Publications (2)

Publication Number	Publication Date
PT85547A true PT85547A (pt)	1988-08-17
PT85547B PT85547B (pt)	1995-03-01

Family

ID=25409053

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT85547A PT85547B (pt)	1986-08-18	1987-08-17	Processo de preparacao de composicao farmaceuticas a base de derivados de 2-mercapto-imidazol e de preparacao destes derivados

Country Status (15)

Country	Link
EP (2)	EP0288488A4 (pt)
CN (1)	CN87105734A (pt)
AT (1)	ATE72430T1 (pt)
AU (1)	AU7910287A (pt)
DE (1)	DE3776613D1 (pt)
DK (1)	DK210488D0 (pt)
ES (1)	ES2038185T3 (pt)
GR (1)	GR3004345T3 (pt)
HU (2)	HU911945D0 (pt)
NZ (1)	NZ221427A (pt)
PH (1)	PH23530A (pt)
PT (1)	PT85547B (pt)
WO (1)	WO1988001267A1 (pt)
ZA (1)	ZA876073B (pt)
ZW (1)	ZW15387A1 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4835154A (en) *	1987-06-01	1989-05-30	Smithkline Beckman Corporation	1-aralykyl-5-piperazinylmethyl-2-mercaptoimidazoles and 2-alkylthioimidazoles and their use as dopamine-βhydroxylase inhibitors
US4882348A (en) *	1987-12-29	1989-11-21	Smithkline Beckman Corporation	2-(aminoalkylthio)imidazoles as dopamine-β-hydroxylase inhibitors
FR2928544A1 (fr) *	2008-03-17	2009-09-18	Oreal	Utilisation d'inhibiteurs de la dopamine-beta hydroxylase pour la pigmentation capillaire.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS5671074A (en) *	1979-11-12	1981-06-13	Takeda Chem Ind Ltd	1,2-disubstituted-4-halogenoimidazole-5-acetic acid derivative
PT78388B (en) *	1983-04-12	1986-09-15	Smithkline Beckman Corp	Dopamine-beta-hydroxylase inhibitors
US4532331A (en) *	1983-04-12	1985-07-30	Smithkline Beckman Corporation	1-Benzyl-2-aminomethyl imidazole derivatives

1987
- 1987-08-12 NZ NZ221427A patent/NZ221427A/en unknown
- 1987-08-14 ZW ZW153/87A patent/ZW15387A1/xx unknown
- 1987-08-14 PH PH35675A patent/PH23530A/en unknown
- 1987-08-17 AU AU79102/87A patent/AU7910287A/en not_active Abandoned
- 1987-08-17 EP EP19870905838 patent/EP0288488A4/en active Pending
- 1987-08-17 EP EP87307259A patent/EP0260814B1/en not_active Expired - Lifetime
- 1987-08-17 HU HU911945A patent/HU911945D0/hu unknown
- 1987-08-17 DE DE8787307259T patent/DE3776613D1/de not_active Expired - Fee Related
- 1987-08-17 HU HU874557A patent/HU204037B/hu unknown
- 1987-08-17 AT AT87307259T patent/ATE72430T1/de not_active IP Right Cessation
- 1987-08-17 ES ES198787307259T patent/ES2038185T3/es not_active Expired - Lifetime
- 1987-08-17 ZA ZA876073A patent/ZA876073B/xx unknown
- 1987-08-17 PT PT85547A patent/PT85547B/pt not_active IP Right Cessation
- 1987-08-17 WO PCT/US1987/002011 patent/WO1988001267A1/en not_active Ceased
- 1987-08-18 CN CN198787105734A patent/CN87105734A/zh active Pending
1988
- 1988-04-18 DK DK210488A patent/DK210488D0/da not_active Application Discontinuation
1992
- 1992-04-15 GR GR920400699T patent/GR3004345T3/el unknown

Also Published As

Publication number	Publication date
HUT50461A (en)	1990-02-28
ZW15387A1 (en)	1987-11-18
GR3004345T3 (pt)	1993-03-31
ES2038185T3 (es)	1993-07-16
EP0260814A1 (en)	1988-03-23
DK210488A (da)	1988-04-18
EP0288488A4 (en)	1990-09-12
PT85547B (pt)	1995-03-01
ZA876073B (en)	1988-08-31
HU204037B (en)	1991-11-28
EP0260814B1 (en)	1992-02-05
DK210488D0 (da)	1988-04-18
DE3776613D1 (de)	1992-03-19
CN87105734A (zh)	1988-02-24
AU7910287A (en)	1988-03-08
EP0288488A1 (en)	1988-11-02
HU911945D0 (en)	1991-12-30
WO1988001267A1 (en)	1988-02-25
PH23530A (en)	1989-08-25
ATE72430T1 (de)	1992-02-15
NZ221427A (en)	1990-12-21

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Legal Events

Date

Code

Title

Description

1995-03-01

FG3A

Patent granted, date of granting

Effective date: 19940811

1996-06-28

MM3A

Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19960229