PT87986A - Processo para a preparacao de derivados de tieno-imidazol substituido e de composicoes farmaceuticas que os contem, apropriadas como agentes inibidores da secrecao do acido do estomago, para a proteccao do estomago, assim como para o tratamento de inflamacoes intestinais - Google Patents
Processo para a preparacao de derivados de tieno-imidazol substituido e de composicoes farmaceuticas que os contem, apropriadas como agentes inibidores da secrecao do acido do estomago, para a proteccao do estomago, assim como para o tratamento de inflamacoes intestinaisInfo
- Publication number
- PT87986A PT87986A PT87986A PT8798688A PT87986A PT 87986 A PT87986 A PT 87986A PT 87986 A PT87986 A PT 87986A PT 8798688 A PT8798688 A PT 8798688A PT 87986 A PT87986 A PT 87986A
- Authority
- PT
- Portugal
- Prior art keywords
- stomach
- tieno
- secrecy
- imidazole
- derivatives
- Prior art date
Links
- 210000002784 stomach Anatomy 0.000 title 2
- 206010061218 Inflammation Diseases 0.000 title 1
- 239000002253 acid Substances 0.000 title 1
- 239000003795 chemical substances by application Substances 0.000 title 1
- RAXXELZNTBOGNW-UHFFFAOYSA-N imidazole Substances C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 title 1
- 230000002401 inhibitory effect Effects 0.000 title 1
- 230000000968 intestinal effect Effects 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19873723327 DE3723327A1 (de) | 1987-07-15 | 1987-07-15 | Substituierte thienoimidazol-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung als magensaeuresekretionshemmer, magenschutzmittel sowie als medikament gegen intestinale entzuendungen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PT87986A true PT87986A (pt) | 1989-06-30 |
Family
ID=6331583
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT87986A PT87986A (pt) | 1987-07-15 | 1988-07-14 | Processo para a preparacao de derivados de tieno-imidazol substituido e de composicoes farmaceuticas que os contem, apropriadas como agentes inibidores da secrecao do acido do estomago, para a proteccao do estomago, assim como para o tratamento de inflamacoes intestinais |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US4956366A (pt) |
| EP (1) | EP0299389A3 (pt) |
| JP (1) | JPS6431785A (pt) |
| KR (1) | KR890002107A (pt) |
| AU (1) | AU618540B2 (pt) |
| DE (1) | DE3723327A1 (pt) |
| DK (1) | DK393788A (pt) |
| FI (1) | FI883342A7 (pt) |
| HU (1) | HU201078B (pt) |
| IL (1) | IL87122A0 (pt) |
| NO (1) | NO167980C (pt) |
| NZ (1) | NZ225387A (pt) |
| PH (1) | PH26118A (pt) |
| PT (1) | PT87986A (pt) |
| ZA (1) | ZA885093B (pt) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1222412B (it) * | 1987-07-31 | 1990-09-05 | Chiesi Farma Spa | Tiometil e sulfinil metil derivati ad azione antisecretiva acida gastrica,loro procedimento di preparazione e composizioni farmaceutiche che li contengono |
| US5271944A (en) * | 1991-04-05 | 1993-12-21 | Biofor, Ltd. | Pharmacologically enhanced formulations |
| US6852739B1 (en) | 1999-02-26 | 2005-02-08 | Nitromed Inc. | Methods using proton pump inhibitors and nitric oxide donors |
| KR100441901B1 (ko) * | 2001-07-02 | 2004-07-27 | 일동제약주식회사 | 세팔로스포린 유도체의 개선된 제조방법 |
| EP1534278A4 (en) * | 2002-08-01 | 2006-09-06 | Nitromed Inc | NITROSED PROTONATE PUMP INHIBITORS, COMPOSITIONS AND USE METHOD |
| CN102675217A (zh) * | 2012-05-24 | 2012-09-19 | 盛世泰科生物医药技术(苏州)有限公司 | 一种5-溴-2-甲基-4(1h)-嘧啶酮的制备方法 |
| US9068530B2 (en) | 2013-03-15 | 2015-06-30 | Mahle International Gmbh | Connecting rod with lubrication passage |
| KR102431436B1 (ko) | 2014-08-29 | 2022-08-10 | 테스 파마 에스.알.엘. | α-아미노-β-카복시뮤콘산 세미알데히드 데카복실라제의 억제제 |
| JP2025532389A (ja) | 2022-10-04 | 2025-09-29 | ザビリュク,アルセニー | 大動脈弁の石灰化の抑制 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4055647A (en) * | 1973-06-14 | 1977-10-25 | Ciba-Geigy Corporation | Condensed pyrrole mercapto compounds having hypotensive and decongestant properties |
| SE416649B (sv) * | 1974-05-16 | 1981-01-26 | Haessle Ab | Forfarande for framstellning av foreningar som paverkar magsyrasekretionen |
| SE7804231L (sv) * | 1978-04-14 | 1979-10-15 | Haessle Ab | Magsyrasekretionsmedel |
| US4472409A (en) * | 1981-11-05 | 1984-09-18 | Byk Gulden Lomberg Chemische Fabrik Gesellschaft Mit Beschrankter Haftung | 2-Pyridylmethyl thio(sulfinyl)benzimidazoles with gastric acid secretion inhibiting effects |
| EP0178438A1 (en) * | 1984-09-19 | 1986-04-23 | Beecham Group Plc | Novel compounds |
| DK8600939A (pt) * | 1985-03-05 | 1986-09-06 | ||
| FI861772L (fi) * | 1985-05-07 | 1986-11-08 | Chemie Linz Ag | Nya tieno(2,3-d)imidazolderivat och foerfarande for deras framstaellning. |
| DE3777855D1 (de) * | 1986-02-20 | 1992-05-07 | Hoechst Ag | Substituierte thienoimidazol-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung als magensaeuresekretionshemmer. |
| DE3639926A1 (de) * | 1986-11-22 | 1988-06-01 | Hoechst Ag | Substituierte thienoimidazoltoluidin-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung als magensaeuresekretionshemmer |
-
1987
- 1987-07-15 DE DE19873723327 patent/DE3723327A1/de not_active Withdrawn
-
1988
- 1988-07-09 EP EP88110991A patent/EP0299389A3/de not_active Withdrawn
- 1988-07-13 PH PH37218A patent/PH26118A/en unknown
- 1988-07-13 NZ NZ225387A patent/NZ225387A/xx unknown
- 1988-07-13 FI FI883342A patent/FI883342A7/fi not_active Application Discontinuation
- 1988-07-13 US US07/218,386 patent/US4956366A/en not_active Expired - Fee Related
- 1988-07-14 ZA ZA885093A patent/ZA885093B/xx unknown
- 1988-07-14 AU AU19032/88A patent/AU618540B2/en not_active Ceased
- 1988-07-14 DK DK393788A patent/DK393788A/da not_active Application Discontinuation
- 1988-07-14 JP JP63173859A patent/JPS6431785A/ja active Pending
- 1988-07-14 PT PT87986A patent/PT87986A/pt unknown
- 1988-07-14 NO NO883145A patent/NO167980C/no unknown
- 1988-07-15 IL IL87122A patent/IL87122A0/xx unknown
- 1988-07-15 KR KR1019880008823A patent/KR890002107A/ko not_active Ceased
- 1988-07-15 HU HU883709A patent/HU201078B/hu not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| IL87122A0 (en) | 1988-12-30 |
| NO167980B (no) | 1991-09-23 |
| NO167980C (no) | 1992-01-02 |
| HU201078B (en) | 1990-09-28 |
| EP0299389A2 (de) | 1989-01-18 |
| FI883342A7 (fi) | 1989-01-16 |
| PH26118A (en) | 1992-02-24 |
| US4956366A (en) | 1990-09-11 |
| AU618540B2 (en) | 1992-01-02 |
| DE3723327A1 (de) | 1989-02-02 |
| FI883342A0 (fi) | 1988-07-13 |
| NZ225387A (en) | 1990-07-26 |
| AU1903288A (en) | 1989-01-19 |
| JPS6431785A (en) | 1989-02-02 |
| DK393788A (da) | 1989-01-16 |
| NO883145L (no) | 1989-01-16 |
| DK393788D0 (da) | 1988-07-14 |
| NO883145D0 (no) | 1988-07-14 |
| KR890002107A (ko) | 1989-04-08 |
| ZA885093B (en) | 1989-03-29 |
| EP0299389A3 (de) | 1990-05-30 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| PT88186A (pt) | Processo para a preparacao de derivados 4'-fosfato de glucosidos da epipodofilotoxina e de composicoes farmaceuticas que os contem | |
| PT92497A (pt) | Processo para a preparacao de derivados de ureia de dipeptideos inibidores de enzimas, e de composicoes farmaceuticas que os contem | |
| PT82591B (pt) | Processo para a preparacao de derivados do acido ascorbico e de composicoes farmaceuticas que os contem | |
| PT80921B (pt) | Processo para a preparacao de derivados de 3-acilaminometil-imidazo {1,2-a} piridinas e de composicoes farmaceuticas que os contem | |
| PT84171B (pt) | Processo para a preparacao de derivados das n alfa-aril-sulfonilamiminoacil-p- -amidinofenil-alaninamidas, bem como dos seus derivados de sintese e das composicoes farmaceuticas que os contem | |
| PT99671A (pt) | Processo para a preparacao de heparosanos-n,o-sulfatados e de composicoes farmaceuticas que os contem | |
| PT91287A (pt) | Processo de preparacao de derivados do acido indazol-3-carboxilico e de composicoes farmaceuticas que os contem | |
| PT84704B (pt) | Processo para a preparacao de derivados do acido tiolactam-n-acetico e de composicoes farmaceuticas que os contem | |
| PT83909B (pt) | Processo para a preparacao de 5-amino e 5-hidroxi-6,8-difluoroquinolonas e de composicoes farmaceuticas antibacterianas que as contem | |
| PT84681B (pt) | Processo para a preparacao de carboxamidas heterociclicas e de composicoes farmaceuticas que as contem | |
| PT97114A (pt) | Processo para a preparacao de derivados de hidantoina e de composicoes farmaceuticas que os contem | |
| MX9205916A (es) | Derivados de acido ciclohexanoacetico, proceso para su preparacion y composicion farmaceutica que los comprende | |
| PT87986A (pt) | Processo para a preparacao de derivados de tieno-imidazol substituido e de composicoes farmaceuticas que os contem, apropriadas como agentes inibidores da secrecao do acido do estomago, para a proteccao do estomago, assim como para o tratamento de inflamacoes intestinais | |
| PT81893B (pt) | Processo para a preparacao de derivados de labdano e de composicoes farmaceuticas que os contem | |
| PT82307B (pt) | Processo para a preparacao de derivados da 4'-demetil-4-epipodofilotoxina e de composicoes farmaceuticas que os contem | |
| PT84187B (pt) | Processo para a preparacao de novos derivados da isoquinolina e de composicoes farmaceuticas que os contem | |
| PT83260B (pt) | Processo para a preparacao de compostos derivados da espergualina e de composicoes farmaceuticas que os contem | |
| PT93067A (pt) | Processo para a preparacao de derivados de 2-hidroxiacidos alifaticos e de eteres de 1-benzil-3-hidroximetilindazol, e de composicoes farmaceuticas que os contem | |
| PT83558B (pt) | Processo para a preparacao de derivados da carboxamida e de composicoes farmaceuticas que os contem | |
| PT89311A (pt) | Processo para a preparacao de novos aminoalcoxi-p-benzonitrilos substituidos utilizaveis como agentes antiarritmicos e de composicoes farmaceuticas que os contem | |
| PT88335A (pt) | Processo para a preparacao de derivados do acido 1,4-dihidro-4-oxo-3-quinolinocarboxilico e de composicoes farmaceuticas que os contem | |
| PT83604B (pt) | Processo para a preparacao de derivados da flavona e de composicoes farmaceuticas que os contem | |
| PT89145A (pt) | Processo para a preparacao de derivados da manumicina e de composicoes farmaceuticas que os contem | |
| PT82901B (pt) | Processo para a preparacao de derivados do acido antranilico dotados de accao terapeutica e de composicoes farmaceuticas que os contem | |
| PT81431B (pt) | Processo para a preparacao de derivados de piridina triciclicos e de composicoes farmaceuticas que os contem |