PT97796A - Processo para a preparacao de piperidinas substituidas - Google Patents

Processo para a preparacao de piperidinas substituidas

Info

Publication number: PT97796A
Authority: PT; Portugal
Prior art keywords: preparation; piperidines; replaced; processes; novel
Prior art date: 1990-05-31

Application number

PT97796A

Other languages

English (en)

Other versions

PT97796B (pt

Inventor

Dennis Michael Godek

Terry Jay Rosen

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-05-31

Filing date

1991-05-29

Publication date

1992-02-28

1991-05-29 Application filed by Pfizer filed Critical Pfizer

1992-02-28 Publication of PT97796A publication Critical patent/PT97796A/pt

1998-10-30 Publication of PT97796B publication Critical patent/PT97796B/pt

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/73—Unsubstituted amino or imino radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Hydrogenated Pyridines (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pyridine Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

PT97796A 1990-05-31 1991-05-29 Processo para a preparacao de piperidinas substituidas PT97796B (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US53126590A	1990-05-31	1990-05-31

Publications (2)

Publication Number	Publication Date
PT97796A true PT97796A (pt)	1992-02-28
PT97796B PT97796B (pt)	1998-10-30

Family

ID=24116944

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT97796A PT97796B (pt)	1990-05-31	1991-05-29	Processo para a preparacao de piperidinas substituidas

Country Status (26)

Country	Link
EP (1)	EP0532515B1 (pt)
JP (2)	JPH0794439B2 (pt)
KR (1)	KR0160142B1 (pt)
CN (2)	CN1037768C (pt)
AT (1)	ATE144498T1 (pt)
AU (1)	AU648558B2 (pt)
BR (1)	BR9106518A (pt)
CA (1)	CA2080249C (pt)
CZ (1)	CZ284663B6 (pt)
DE (1)	DE69122866T2 (pt)
DK (1)	DK0532515T3 (pt)
ES (1)	ES2093099T3 (pt)
FI (1)	FI101376B (pt)
GR (1)	GR3022079T3 (pt)
HU (1)	HU226529B1 (pt)
IE (1)	IE911841A1 (pt)
IL (3)	IL113011A (pt)
MY (1)	MY107819A (pt)
NO (1)	NO180083C (pt)
NZ (2)	NZ238340A (pt)
PL (2)	PL169187B1 (pt)
PT (1)	PT97796B (pt)
RU (1)	RU2077531C1 (pt)
WO (1)	WO1991018878A1 (pt)
YU (1)	YU48030B (pt)
ZA (1)	ZA914133B (pt)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
UA41251C2 (uk) *	1990-01-04	2001-09-17	Пфайзер, Інк.	Гідровані азотвмісні гетероциклічні сполуки, похідні піперидину, фармацевтична композиція та спосіб пригнічення активності речовини р в організмі
US5332817A (en) *	1990-01-04	1994-07-26	Pfizer Inc.	3-aminopiperidine derivatives and related nitrogen containing heterocycles
US5364943A (en) *	1991-11-27	1994-11-15	Pfizer Inc.	Preparation of substituted piperidines
SK284565B6 (sk) *	1991-03-26	2005-06-02	Pfizer Inc.	Spôsob prípravy substituovaných piperidínov
MY110227A (en) *	1991-08-12	1998-03-31	Ciba Geigy Ag	1-acylpiperindine compounds.
DK0613458T3 (da) *	1991-11-12	1998-02-09	Pfizer	Acykliske ethylendiaminderivater som substans P receptorantagonister
CA2150123C (en) *	1992-12-10	2004-12-07	Harry R. Howard	Aminomethylene substituted non-aromatic heterocycles
DK0700384T3 (da)	1993-05-28	1997-12-08	Pfizer	fremgangsmåde til fremstilling og opløsning af 2-phenyl-3-aminopiperidin
TW397825B (en) *	1994-10-14	2000-07-11	Novartis Ag	Aroyl-piperidine derivatives
FR2728169A1 (fr)	1994-12-19	1996-06-21	Oreal	Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
FR2728166A1 (fr)	1994-12-19	1996-06-21	Oreal	Composition topique contenant un antagoniste de substance p
FR2728165A1 (fr)	1994-12-19	1996-06-21	Oreal	Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2741262B1 (fr)	1995-11-20	1999-03-05	Oreal	Utilisation d'un antagoniste de tnf-alpha pour le traitement des rougeurs cutanees d'origine neurogene
CA2291734A1 (en) *	1997-06-27	1999-01-07	Merck Sharp & Dohme Limited	Substituted 3-(benzylamino)piperidine derivatives and their use as therapeutic agents
EP1098881A1 (en) *	1998-07-21	2001-05-16	Syngenta Participations AG	3-substituted pyridine compounds and related synthesis
TR200102490T2 (tr) *	1999-02-24	2001-12-21	F.Hoffmann-La Roche Ag	Fenil ve piridinil türevleri
KR100437587B1 (ko) *	1999-02-24	2004-06-30	에프. 호프만-라 로슈 아게	3-페닐피리딘 유도체 및 그의 뉴로키닌-1 수용체길항제로서의 용도
RS49964B (sr) *	1999-05-17	2008-09-29	Pfizer Products Inc.,	Postupak za dobijanje 2-fenil-3-aminopiridina,njegovih supstituisanih fenil derivata, i njegovih soli
TWI259180B (en) *	2000-08-08	2006-08-01	Hoffmann La Roche	4-Phenyl-pyridine derivatives
JP2011016751A (ja) *	2009-07-08	2011-01-27	Sumitomo Chemical Co Ltd	光学活性３−アミノピペリジン−１−カルボキシレート化合物の製造方法およびその製造方法に用いられる中間体
CN111808017B (zh) *	2020-08-05	2023-11-28	国家纳米科学中心	一种含氮杂环化合物及其制备方法和应用
CN116162055B (zh) *	2023-03-10	2023-09-12	山东汇智药物研究有限公司	一种用n-氧化吡啶衍生物制备哌啶衍生物的方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS52125170A (en) *	1976-04-12	1977-10-20	Yoshitomi Pharmaceut Ind Ltd	Pyridine derivatives
CA1160229A (en) *	1979-03-13	1984-01-10	Pieter T. Haken	Pyridyliminomethylbenzene derivatives
CA1231710A (en) *	1979-07-19	1988-01-19	Haken Pieter Ten	Heterocyclic compounds having fungicidal, herbicidal and plant-growth regulating properties
GB2056974B (en) *	1979-07-19	1984-02-29	Shell Int Research	Heterocyclic acylamino compounds having fungicidal herbicidal and plant-growth regulating properties
EP0100158A3 (en) *	1982-07-28	1985-03-27	The Upjohn Company	(3-pyridinyl)heteroalkarylalkanols, alkanoic acids and esters
US4552960A (en) *	1983-06-20	1985-11-12	Eli Lilly And Company	Fungicidal amines
FR2662696A2 (fr) *	1989-12-13	1991-12-06	Rhone Poulenc Sante	Antagonistes de la serotonine, leur preparation et medicaments les contenant.
UA41251C2 (uk) *	1990-01-04	2001-09-17	Пфайзер, Інк.	Гідровані азотвмісні гетероциклічні сполуки, похідні піперидину, фармацевтична композиція та спосіб пригнічення активності речовини р в організмі

1991
- 1991-04-12 CA CA002080249A patent/CA2080249C/en not_active Expired - Fee Related
- 1991-04-12 EP EP91908255A patent/EP0532515B1/en not_active Expired - Lifetime
- 1991-04-12 RU RU9192016444A patent/RU2077531C1/ru not_active IP Right Cessation
- 1991-04-12 PL PL91309053A patent/PL169187B1/pl unknown
- 1991-04-12 DK DK91908255.2T patent/DK0532515T3/da active
- 1991-04-12 AU AU77703/91A patent/AU648558B2/en not_active Ceased
- 1991-04-12 BR BR919106518A patent/BR9106518A/pt not_active Application Discontinuation
- 1991-04-12 AT AT91908255T patent/ATE144498T1/de not_active IP Right Cessation
- 1991-04-12 HU HU9203761A patent/HU226529B1/hu not_active IP Right Cessation
- 1991-04-12 PL PL91297179A patent/PL168236B1/pl unknown
- 1991-04-12 DE DE69122866T patent/DE69122866T2/de not_active Expired - Fee Related
- 1991-04-12 JP JP3508366A patent/JPH0794439B2/ja not_active Expired - Fee Related
- 1991-04-12 KR KR1019920703014A patent/KR0160142B1/ko not_active Expired - Fee Related
- 1991-04-12 ES ES91908255T patent/ES2093099T3/es not_active Expired - Lifetime
- 1991-04-12 WO PCT/US1991/002541 patent/WO1991018878A1/en not_active Ceased
- 1991-05-24 IL IL11301191A patent/IL113011A/xx not_active IP Right Cessation
- 1991-05-24 IL IL9825691A patent/IL98256A/en not_active IP Right Cessation
- 1991-05-29 MY MYPI91000939A patent/MY107819A/en unknown
- 1991-05-29 PT PT97796A patent/PT97796B/pt not_active IP Right Cessation
- 1991-05-30 NZ NZ238340A patent/NZ238340A/xx unknown
- 1991-05-30 NZ NZ250217A patent/NZ250217A/en unknown
- 1991-05-30 CN CN91103654A patent/CN1037768C/zh not_active Expired - Fee Related
- 1991-05-30 ZA ZA914133A patent/ZA914133B/xx unknown
- 1991-05-30 IE IE184191A patent/IE911841A1/en not_active IP Right Cessation
- 1991-05-30 YU YU96291A patent/YU48030B/sh unknown
- 1991-05-30 CZ CS911623A patent/CZ284663B6/cs not_active IP Right Cessation
1992
- 1992-11-27 FI FI925415A patent/FI101376B/fi active
- 1992-11-27 NO NO924598A patent/NO180083C/no not_active IP Right Cessation
1994
- 1994-12-26 JP JP6322305A patent/JP2549609B2/ja not_active Expired - Fee Related
1995
- 1995-03-16 IL IL11301195A patent/IL113011A0/xx unknown
1996
- 1996-12-18 GR GR960403524T patent/GR3022079T3/el unknown
1997
- 1997-08-26 CN CNB971178879A patent/CN1154636C/zh not_active Expired - Fee Related

Also Published As

Publication number	Publication date
GR3022079T3 (en)	1997-03-31
IL113011A (en)	1999-09-22
CS162391A3 (en)	1992-02-19
HU226529B1 (en)	2009-03-30
DE69122866D1 (de)	1996-11-28
PL168236B1 (pl)	1996-01-31
JPH05502238A (ja)	1993-04-22
KR0160142B1 (ko)	1998-12-01
FI925415L (fi)	1992-11-27
PL169187B1 (pl)	1996-06-28
CN1154636C (zh)	2004-06-23
IL98256A0 (en)	1992-06-21
CN1037768C (zh)	1998-03-18
KR930700443A (ko)	1993-03-15
DE69122866T2 (de)	1997-02-20
CZ284663B6 (cs)	1999-01-13
CA2080249C (en)	1996-11-19
ATE144498T1 (de)	1996-11-15
PT97796B (pt)	1998-10-30
HU9203761D0 (en)	1993-03-29
WO1991018878A1 (en)	1991-12-12
JPH0794439B2 (ja)	1995-10-11
JPH07206819A (ja)	1995-08-08
FI101376B1 (fi)	1998-06-15
FI925415A0 (fi)	1992-11-27
BR9106518A (pt)	1993-05-25
AU7770391A (en)	1991-12-31
YU96291A (sh)	1994-06-10
NO180083C (no)	1997-02-12
CN1056876A (zh)	1991-12-11
FI101376B (fi)	1998-06-15
EP0532515A1 (en)	1993-03-24
CA2080249A1 (en)	1991-12-01
JP2549609B2 (ja)	1996-10-30
NO924598D0 (no)	1992-11-27
HUT68166A (en)	1995-05-29
RU2077531C1 (ru)	1997-04-20
IE911841A1 (en)	1991-12-04
CN1183408A (zh)	1998-06-03
NZ238340A (en)	1994-06-27
NO924598L (no)	1992-11-27
AU648558B2 (en)	1994-04-28
IL98256A (en)	1995-11-27
IL113011A0 (en)	1995-06-29
EP0532515B1 (en)	1996-10-23
YU48030B (sh)	1996-10-09
DK0532515T3 (da)	1997-04-21
ZA914133B (en)	1993-01-27
ES2093099T3 (es)	1996-12-16
NO180083B (no)	1996-11-04
NZ250217A (en)	1995-05-26
MY107819A (en)	1996-06-29

Legal Events

Date	Code	Title	Description
1992-02-28	BB1A	Laying open of patent application	Effective date: 19911104
1998-10-30	FG3A	Patent granted, date of granting	Effective date: 19980721
2002-06-28	NF3A	Restitutio in integrum	Free format text: 20020315 RESTITUTIO IN INTEGRUM
2010-01-27	MM4A	Annulment/lapse due to non-payment of fees, searched and examined patent	Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 20100121

Publication	Publication Date	Title
PT97796A (pt)	1992-02-28	Processo para a preparacao de piperidinas substituidas
FI964520L (fi)	1996-11-11	Atsabisykloyhdisteet
PT96857A (pt)	1991-10-31	Processo para a preparacao de oxetanonas
HUT68963A (en)	1995-08-28	Novel 4-arylpiperazines and 4-arylpiperidines, pharmaceutical compositions comprising them and the proces for producing thereof
BR9206823A (pt)	1995-04-25	Preparação de piperidinas substituídas
PT92307A (pt)	1990-05-31	Processo para a preparacao de derivados de 3,5-dimetil-4-metoxipiridina e de produtos intermediarios
PT93702A (pt)	1990-11-20	Processo para a preparacao de 2,7-diazabiciclo{3.3.0}octanos e de produtos intermediarios
BR9200627A (pt)	1992-10-27	Processo para a preparacao de um composto e composto obtido
BR9400016A (pt)	1995-05-02	Processo para preparação de compostos, e compostos
PT97738A (pt)	1992-03-31	PROCESSO PARA A PREPARACAO DE DAIS DE URóNIO
PT98268A (pt)	1992-05-29	Processo para a preparacao de indano-pirrolidino-carbamatos
PT98976A (pt)	1992-07-31	Processo para a preparacao de heteroarilmetilbenzenos
GR3018765T3 (en)	1996-04-30	Process for the preparation of N-(2-hydroxyethyl)-2-hydroxymethyl-3,4,5-trihydroxy-piperidine and of intermediates.
PT882045E (pt)	2004-10-29	Processo para a preparacao de granisetron
DK0431305T3 (da)	1995-04-03	Fremgangsmåde til fremstilling af molluskicide 2,4,5-tribrompyrrol-3-carbonitriler
BR9404139A (pt)	1995-06-13	Processo aperfeiçoado para a preparação de compostos de fórmula (I) ou fórmula (II)
DE59002172D1 (de)	1993-09-09	Neue 1,3-oxazine.
BR9610392A (pt)	1999-07-06	Processo para a preparação de derivados de rodanina substituídos com benzila
BR9201895A (pt)	1993-01-05	Processo para preparar 2-(aminometil)-4-tiazolmetanol e compostos
BR8706887A (pt)	1988-07-26	Processo para a preparacao de compostos