PT98697A - Processo para a preparacao de compostos macrociclicos e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de compostos macrociclicos e de composicoes farmaceuticas que os contem

Info

Publication number
PT98697A
PT98697A PT98697A PT9869791A PT98697A PT 98697 A PT98697 A PT 98697A PT 98697 A PT98697 A PT 98697A PT 9869791 A PT9869791 A PT 9869791A PT 98697 A PT98697 A PT 98697A
Authority
PT
Portugal
Prior art keywords
pharmaceutical compositions
compositions containing
macrocyclic compounds
preparing macrocyclic
preparing
Prior art date
Application number
PT98697A
Other languages
English (en)
Other versions
PT98697B (pt
Inventor
Mark Furber
David Keith Donald
Original Assignee
Fisons Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB909018196A external-priority patent/GB9018196D0/en
Priority claimed from GB919102305A external-priority patent/GB9102305D0/en
Application filed by Fisons Plc filed Critical Fisons Plc
Publication of PT98697A publication Critical patent/PT98697A/pt
Publication of PT98697B publication Critical patent/PT98697B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Immunology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Transplantation (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PT98697A 1990-08-18 1991-08-16 Processo para a preparacao de compostos macrociclicos e de composicoes farmaceuticas que os contem PT98697B (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB909018196A GB9018196D0 (en) 1990-08-18 1990-08-18 Compounds
GB919102305A GB9102305D0 (en) 1991-02-02 1991-02-02 Compounds

Publications (2)

Publication Number Publication Date
PT98697A true PT98697A (pt) 1992-07-31
PT98697B PT98697B (pt) 1999-01-29

Family

ID=26297532

Family Applications (1)

Application Number Title Priority Date Filing Date
PT98697A PT98697B (pt) 1990-08-18 1991-08-16 Processo para a preparacao de compostos macrociclicos e de composicoes farmaceuticas que os contem

Country Status (8)

Country Link
US (1) US5384316A (pt)
EP (1) EP0543879A1 (pt)
JP (1) JPH06500102A (pt)
CN (1) CN1060846A (pt)
AU (1) AU8394291A (pt)
IE (1) IE912886A1 (pt)
PT (1) PT98697B (pt)
WO (1) WO1992003441A1 (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5565560A (en) * 1991-05-13 1996-10-15 Merck & Co., Inc. O-Aryl,O-alkyl,O-alkenyl and O-alkynylmacrolides having immunosuppressive activity
US5262533A (en) * 1991-05-13 1993-11-16 Merck & Co., Inc. Amino O-aryl macrolides having immunosuppressive activity
US5457111A (en) * 1991-09-05 1995-10-10 Abbott Laboratories Macrocyclic immunomodulators
US5252732A (en) * 1991-09-09 1993-10-12 Merck & Co., Inc. D-heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynylheteroarylmacrolides having immunosuppressive activity
US5247076A (en) * 1991-09-09 1993-09-21 Merck & Co., Inc. Imidazolidyl macrolides having immunosuppressive activity
GB9203265D0 (en) * 1992-02-15 1992-04-01 Fisons Plc Pharmaceutically active compound
HUT66531A (en) * 1992-05-07 1994-12-28 Sandoz Ag Heteroatoms-containing tricyclic compounds, pharmaceutical prepns contg. them and process for producing them
US5284840A (en) * 1992-06-12 1994-02-08 Merck & Co., Inc. Alkylidene macrolides having immunosuppressive activity
US5284877A (en) * 1992-06-12 1994-02-08 Merck & Co., Inc. Alkyl and alkenyl macrolides having immunosuppressive activity
GB9218797D0 (en) * 1992-09-04 1992-10-21 Fisons Plc Pharmacologically active compounds
US5693648A (en) * 1994-09-30 1997-12-02 Merck & Co., Inc. O-aryl, O-alkyl, O-alkenyl and O-alkynyl-macrolides having immunosuppressive activity
WO2006115509A2 (en) 2004-06-24 2006-11-02 Novartis Vaccines And Diagnostics Inc. Small molecule immunopotentiators and assays for their detection

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4659389A (en) * 1984-02-16 1987-04-21 Ashland Oil, Inc. Method and composition of asphaltic roofing fluxes
US4894366A (en) * 1984-12-03 1990-01-16 Fujisawa Pharmaceutical Company, Ltd. Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
WO1989005304A1 (en) * 1987-12-09 1989-06-15 Fisons Plc Macrocyclic compounds
EP0356399A3 (en) * 1988-08-26 1991-03-20 Sandoz Ag Substituted 4-azatricyclo (22.3.1.04.9) octacos-18-ene derivatives, their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
AU8394291A (en) 1992-03-17
US5384316A (en) 1995-01-24
JPH06500102A (ja) 1994-01-06
EP0543879A1 (en) 1993-06-02
IE912886A1 (en) 1992-02-26
WO1992003441A1 (en) 1992-03-05
CN1060846A (zh) 1992-05-06
PT98697B (pt) 1999-01-29

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Legal Events

Date Code Title Description
BB1A Laying open of patent application

Effective date: 19920318

FG3A Patent granted, date of granting

Effective date: 19981027

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20000430