PT98697A - Processo para a preparacao de compostos macrociclicos e de composicoes farmaceuticas que os contem - Google Patents
Processo para a preparacao de compostos macrociclicos e de composicoes farmaceuticas que os contemInfo
- Publication number
- PT98697A PT98697A PT98697A PT9869791A PT98697A PT 98697 A PT98697 A PT 98697A PT 98697 A PT98697 A PT 98697A PT 9869791 A PT9869791 A PT 9869791A PT 98697 A PT98697 A PT 98697A
- Authority
- PT
- Portugal
- Prior art keywords
- pharmaceutical compositions
- compositions containing
- macrocyclic compounds
- preparing macrocyclic
- preparing
- Prior art date
Links
- 150000002678 macrocyclic compounds Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Immunology (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Transplantation (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB909018196A GB9018196D0 (en) | 1990-08-18 | 1990-08-18 | Compounds |
| GB919102305A GB9102305D0 (en) | 1991-02-02 | 1991-02-02 | Compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT98697A true PT98697A (pt) | 1992-07-31 |
| PT98697B PT98697B (pt) | 1999-01-29 |
Family
ID=26297532
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT98697A PT98697B (pt) | 1990-08-18 | 1991-08-16 | Processo para a preparacao de compostos macrociclicos e de composicoes farmaceuticas que os contem |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US5384316A (pt) |
| EP (1) | EP0543879A1 (pt) |
| JP (1) | JPH06500102A (pt) |
| CN (1) | CN1060846A (pt) |
| AU (1) | AU8394291A (pt) |
| IE (1) | IE912886A1 (pt) |
| PT (1) | PT98697B (pt) |
| WO (1) | WO1992003441A1 (pt) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5565560A (en) * | 1991-05-13 | 1996-10-15 | Merck & Co., Inc. | O-Aryl,O-alkyl,O-alkenyl and O-alkynylmacrolides having immunosuppressive activity |
| US5262533A (en) * | 1991-05-13 | 1993-11-16 | Merck & Co., Inc. | Amino O-aryl macrolides having immunosuppressive activity |
| US5457111A (en) * | 1991-09-05 | 1995-10-10 | Abbott Laboratories | Macrocyclic immunomodulators |
| US5252732A (en) * | 1991-09-09 | 1993-10-12 | Merck & Co., Inc. | D-heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynylheteroarylmacrolides having immunosuppressive activity |
| US5247076A (en) * | 1991-09-09 | 1993-09-21 | Merck & Co., Inc. | Imidazolidyl macrolides having immunosuppressive activity |
| GB9203265D0 (en) * | 1992-02-15 | 1992-04-01 | Fisons Plc | Pharmaceutically active compound |
| HUT66531A (en) * | 1992-05-07 | 1994-12-28 | Sandoz Ag | Heteroatoms-containing tricyclic compounds, pharmaceutical prepns contg. them and process for producing them |
| US5284840A (en) * | 1992-06-12 | 1994-02-08 | Merck & Co., Inc. | Alkylidene macrolides having immunosuppressive activity |
| US5284877A (en) * | 1992-06-12 | 1994-02-08 | Merck & Co., Inc. | Alkyl and alkenyl macrolides having immunosuppressive activity |
| GB9218797D0 (en) * | 1992-09-04 | 1992-10-21 | Fisons Plc | Pharmacologically active compounds |
| US5693648A (en) * | 1994-09-30 | 1997-12-02 | Merck & Co., Inc. | O-aryl, O-alkyl, O-alkenyl and O-alkynyl-macrolides having immunosuppressive activity |
| WO2006115509A2 (en) | 2004-06-24 | 2006-11-02 | Novartis Vaccines And Diagnostics Inc. | Small molecule immunopotentiators and assays for their detection |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4659389A (en) * | 1984-02-16 | 1987-04-21 | Ashland Oil, Inc. | Method and composition of asphaltic roofing fluxes |
| US4894366A (en) * | 1984-12-03 | 1990-01-16 | Fujisawa Pharmaceutical Company, Ltd. | Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same |
| WO1989005304A1 (en) * | 1987-12-09 | 1989-06-15 | Fisons Plc | Macrocyclic compounds |
| EP0356399A3 (en) * | 1988-08-26 | 1991-03-20 | Sandoz Ag | Substituted 4-azatricyclo (22.3.1.04.9) octacos-18-ene derivatives, their preparation and pharmaceutical compositions containing them |
-
1991
- 1991-08-14 JP JP3514221A patent/JPH06500102A/ja active Pending
- 1991-08-14 US US07/975,544 patent/US5384316A/en not_active Expired - Fee Related
- 1991-08-14 IE IE288691A patent/IE912886A1/en unknown
- 1991-08-14 EP EP91914660A patent/EP0543879A1/en not_active Withdrawn
- 1991-08-14 WO PCT/GB1991/001384 patent/WO1992003441A1/en not_active Ceased
- 1991-08-14 AU AU83942/91A patent/AU8394291A/en not_active Abandoned
- 1991-08-16 PT PT98697A patent/PT98697B/pt not_active IP Right Cessation
- 1991-08-17 CN CN91108918A patent/CN1060846A/zh active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| AU8394291A (en) | 1992-03-17 |
| US5384316A (en) | 1995-01-24 |
| JPH06500102A (ja) | 1994-01-06 |
| EP0543879A1 (en) | 1993-06-02 |
| IE912886A1 (en) | 1992-02-26 |
| WO1992003441A1 (en) | 1992-03-05 |
| CN1060846A (zh) | 1992-05-06 |
| PT98697B (pt) | 1999-01-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BB1A | Laying open of patent application |
Effective date: 19920318 |
|
| FG3A | Patent granted, date of granting |
Effective date: 19981027 |
|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 20000430 |