RO81223B - Process for preparing some derivatives of 1-cyclohexyle-4-aryl-pyperidincarboxylic acid - Google Patents

Process for preparing some derivatives of 1-cyclohexyle-4-aryl-pyperidincarboxylic acid

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Publication number
RO81223B
RO81223B RO103173A RO10317381A RO81223B RO 81223 B RO81223 B RO 81223B RO 103173 A RO103173 A RO 103173A RO 10317381 A RO10317381 A RO 10317381A RO 81223 B RO81223 B RO 81223B
Authority
RO
Romania
Prior art keywords
aryl
general formula
derivatives
pyperidincarboxylic
cyclohexyle
Prior art date
Application number
RO103173A
Other languages
Romanian (ro)
Other versions
RO81223A (en
Inventor
Raymond Stokbroekx
Marcel Luyckx
Joannes Willema
Original Assignee
Jannsen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jannsen Pharmaceutica N.V. filed Critical Jannsen Pharmaceutica N.V.
Publication of RO81223A publication Critical patent/RO81223A/en
Publication of RO81223B publication Critical patent/RO81223B/en

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  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Inventia se refera la un procedeu pentru prepararea unor derivati al acidului 1-ciclohexil-4-aril-piperidincarboxilic, cu formula generala I: (vezi formula) în care r reprezinta o grupa hidroxi alchiloxi inferior aril alchiloxi inferior, R1 reprezinta hidrogen sau alchil inferior, Ar1 si Ar2, reprezinta aril tienil sau piridinil, prin reactia unui compus cu formula generala II: 8vezi formula) cu un compus cu formula generala III: (vezi formula) prin hidrogenarea catalitica în prezenta unui catalizator de paladiu sau platina pe suport de carbune.The invention relates to a process for the preparation of 1-cyclohexyl-4-aryl-piperidinecarboxylic acid derivatives of the general formula I wherein R represents a lower alkoxy lower alkyl lower alkyloxy group, R 1 represents hydrogen or lower alkyl , Ar 1 and Ar 2 represent aryl thienyl or pyridinyl by reacting a compound of the general formula II with a compound of the general formula III by catalytic hydrogenation in the presence of a palladium or platinum catalyst on a charcoal support .

RO103173A 1980-01-24 1981-01-21 Process for preparing some derivatives of 1-cyclohexyle-4-aryl-pyperidincarboxylic acid RO81223B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11492480A 1980-01-24 1980-01-24
US19163580A 1980-09-29 1980-09-29

Publications (2)

Publication Number Publication Date
RO81223A RO81223A (en) 1983-02-15
RO81223B true RO81223B (en) 1983-02-28

Family

ID=26812675

Family Applications (1)

Application Number Title Priority Date Filing Date
RO103173A RO81223B (en) 1980-01-24 1981-01-21 Process for preparing some derivatives of 1-cyclohexyle-4-aryl-pyperidincarboxylic acid

Country Status (1)

Country Link
RO (1) RO81223B (en)

Also Published As

Publication number Publication date
RO81223A (en) 1983-02-15

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