SA519401954B1 - تركيبة صيدلانية للوقاية من أو معالجة سرطان تشتمل على صورة متعددة الشكل البلوري من تترا أرسينيك هيكسوكسويد - Google Patents

تركيبة صيدلانية للوقاية من أو معالجة سرطان تشتمل على صورة متعددة الشكل البلوري من تترا أرسينيك هيكسوكسويد

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Publication number
SA519401954B1
SA519401954B1 SA519401954A SA519401954A SA519401954B1 SA 519401954 B1 SA519401954 B1 SA 519401954B1 SA 519401954 A SA519401954 A SA 519401954A SA 519401954 A SA519401954 A SA 519401954A SA 519401954 B1 SA519401954 B1 SA 519401954B1
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SA
Saudi Arabia
Prior art keywords
prevention
treatment
cancer
pharmaceutical composition
hexoxide
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SA519401954A
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English (en)
Inventor
الثالث جو باى
زينجلين ليان
Original Assignee
شيماس كو . ليمتد
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Application filed by شيماس كو . ليمتد filed Critical شيماس كو . ليمتد
Publication of SA519401954B1 publication Critical patent/SA519401954B1/ar

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/28Compounds containing heavy metals
    • A61K31/285Arsenic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00Medicinal preparations containing inorganic active ingredients
    • A61K33/24Heavy metals; Compounds thereof
    • A61K33/36Arsenic; Compounds thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C01INORGANIC CHEMISTRY
    • C01GCOMPOUNDS CONTAINING METALS NOT COVERED BY SUBCLASSES C01D OR C01F
    • C01G28/00Compounds of arsenic
    • C01G28/005Oxides; Hydroxides; Oxyacids
    • CCHEMISTRY; METALLURGY
    • C01INORGANIC CHEMISTRY
    • C01PINDEXING SCHEME RELATING TO STRUCTURAL AND PHYSICAL ASPECTS OF SOLID INORGANIC COMPOUNDS
    • C01P2002/00Crystal-structural characteristics
    • C01P2002/60Compounds characterised by their crystallite size
    • CCHEMISTRY; METALLURGY
    • C01INORGANIC CHEMISTRY
    • C01PINDEXING SCHEME RELATING TO STRUCTURAL AND PHYSICAL ASPECTS OF SOLID INORGANIC COMPOUNDS
    • C01P2002/00Crystal-structural characteristics
    • C01P2002/70Crystal-structural characteristics defined by measured X-ray, neutron or electron diffraction data
    • C01P2002/72Crystal-structural characteristics defined by measured X-ray, neutron or electron diffraction data by d-values or two theta-values, e.g. as X-ray diagram
    • CCHEMISTRY; METALLURGY
    • C01INORGANIC CHEMISTRY
    • C01PINDEXING SCHEME RELATING TO STRUCTURAL AND PHYSICAL ASPECTS OF SOLID INORGANIC COMPOUNDS
    • C01P2006/00Physical properties of inorganic compounds
    • C01P2006/80Compositional purity

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Inorganic Compounds Of Heavy Metals (AREA)
  • Medicines Containing Plant Substances (AREA)

Abstract

يتعلق الاختراع الحالي بتركيبة صيدلانية للوقاية من أو معالجة السرطان cancer وطريقة لإنتاجها، وتشتمل التركيبة على هيكسوكسيد تتراسينيك tetraarsenic hexoxide وحيث يكون به محتوى الصورة متعددة الأشكال المتبلرة أ (As4O6-a ) هو 99٪ أو أكثر. وتعرض تركيبة الاختراع الحالي تأثير تثبيط تكاثر خلية السرطان cancer cell وبالتالي يمكن أن تكون مفيدة في شكل عقار مضاد للسرطان anticancer drug. شكل10
SA519401954A 2016-12-09 2019-06-09 تركيبة صيدلانية للوقاية من أو معالجة سرطان تشتمل على صورة متعددة الشكل البلوري من تترا أرسينيك هيكسوكسويد SA519401954B1 (ar)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR1020160167222A KR101844050B1 (ko) 2016-12-09 2016-12-09 육산화사비소의 결정다형을 포함하는 암 예방 또는 치료용 약학 조성물
PCT/KR2017/014082 WO2018105972A1 (ko) 2016-12-09 2017-12-04 육산화사비소의 결정다형을 포함하는 암 예방 또는 치료용 약학 조성물

Publications (1)

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SA519401954B1 true SA519401954B1 (ar) 2024-01-29

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SA519401954A SA519401954B1 (ar) 2016-12-09 2019-06-09 تركيبة صيدلانية للوقاية من أو معالجة سرطان تشتمل على صورة متعددة الشكل البلوري من تترا أرسينيك هيكسوكسويد

Country Status (16)

Country Link
US (1) US11191779B2 (ar)
EP (1) EP3552611A4 (ar)
JP (1) JP6824409B2 (ar)
KR (1) KR101844050B1 (ar)
CN (2) CN108606979A (ar)
AU (1) AU2017371040B2 (ar)
BR (1) BR112019010999A2 (ar)
CA (1) CA3044514C (ar)
CL (1) CL2019001565A1 (ar)
IL (1) IL267132B (ar)
MX (1) MX392459B (ar)
MY (1) MY197417A (ar)
PH (1) PH12019501292A1 (ar)
SA (1) SA519401954B1 (ar)
WO (1) WO2018105972A1 (ar)
ZA (1) ZA201903059B (ar)

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MA41551A (fr) 2015-02-20 2017-12-26 Incyte Corp Hétérocycles bicycliques utilisés en tant qu'inhibiteurs de fgfr4
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US11939331B2 (en) 2021-06-09 2024-03-26 Incyte Corporation Tricyclic heterocycles as FGFR inhibitors
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WO2025165158A1 (ko) * 2024-01-29 2025-08-07 배일주 육산화사비소(As4O6)를 포함하는 방광암 예방 또는 치료용 약학 조성물
KR20250118232A (ko) 2024-01-29 2025-08-05 배일주 육산화사비소(As4O6)를 포함하는 방광암 예방 또는 치료용 약학 조성물

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Also Published As

Publication number Publication date
US20200000846A1 (en) 2020-01-02
JP6824409B2 (ja) 2021-02-03
MX2019006622A (es) 2019-08-01
IL267132A (en) 2019-10-31
MY197417A (en) 2023-06-16
CN108606979A (zh) 2018-10-02
WO2018105972A1 (ko) 2018-06-14
PH12019501292A1 (en) 2019-12-02
CA3044514C (en) 2021-06-15
CL2019001565A1 (es) 2020-02-21
EP3552611A1 (en) 2019-10-16
ZA201903059B (en) 2020-09-30
CA3044514A1 (en) 2018-06-14
JP2020504088A (ja) 2020-02-06
MX392459B (es) 2025-03-24
CN116672363A (zh) 2023-09-01
AU2017371040A1 (en) 2019-06-20
US11191779B2 (en) 2021-12-07
BR112019010999A2 (pt) 2019-10-15
EP3552611A4 (en) 2020-06-24
AU2017371040B2 (en) 2020-05-07
IL267132B (en) 2022-05-01
KR101844050B1 (ko) 2018-05-14

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