SE311644B - - Google Patents

Info

Publication number: SE311644B
Authority: SE; Sweden
Prior art keywords: group; acid; nitro; prepared; alkyl
Prior art date: 1963-06-05

Application number

SE6822/64A

Other languages

English (en)

Inventor

P Schmidt

A Rossi

K Eichenberger

M Wilhelm

Original Assignee

Ciba Geigy

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1963-06-05

Filing date

1964-06-04

Publication date

1969-06-23

1963-06-05 Priority claimed from CH702763A external-priority patent/CH439319A/de

1964-06-04 Application filed by Ciba Geigy filed Critical Ciba Geigy

1969-06-23 Publication of SE311644B publication Critical patent/SE311644B/xx

Links

238000006243 chemical reaction Methods 0.000 abstract 4
WFDIJRYMOXRFFG-UHFFFAOYSA-N Acetic anhydride Chemical compound CC(=O)OC(C)=O WFDIJRYMOXRFFG-UHFFFAOYSA-N 0.000 abstract 3
239000002253 acid Substances 0.000 abstract 3
125000000217 alkyl group Chemical group 0.000 abstract 3
125000002947 alkylene group Chemical group 0.000 abstract 3
150000001412 amines Chemical class 0.000 abstract 2
125000003277 amino group Chemical group 0.000 abstract 2
150000008064 anhydrides Chemical class 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 2
125000006701 (C1-C7) alkyl group Chemical group 0.000 abstract 1
HROLNPSYNSBBFH-UHFFFAOYSA-N 2-amino-5-(dimethylsulfamoyl)benzoic acid Chemical compound CN(C)S(=O)(=O)C1=CC=C(N)C(C(O)=O)=C1 HROLNPSYNSBBFH-UHFFFAOYSA-N 0.000 abstract 1
GSINPMWETVUGBB-UHFFFAOYSA-N 5-chlorosulfonyl-2-nitrobenzoic acid Chemical compound OC(=O)C1=CC(S(Cl)(=O)=O)=CC=C1[N+]([O-])=O GSINPMWETVUGBB-UHFFFAOYSA-N 0.000 abstract 1
239000005711 Benzoic acid Substances 0.000 abstract 1
VEXZGXHMUGYJMC-UHFFFAOYSA-M Chloride anion Chemical compound [Cl-] VEXZGXHMUGYJMC-UHFFFAOYSA-M 0.000 abstract 1
125000002252 acyl group Chemical group 0.000 abstract 1
230000010933 acylation Effects 0.000 abstract 1
238000005917 acylation reaction Methods 0.000 abstract 1
125000001931 aliphatic group Chemical group 0.000 abstract 1
125000003545 alkoxy group Chemical group 0.000 abstract 1
230000003266 anti-allergic effect Effects 0.000 abstract 1
230000003110 anti-inflammatory effect Effects 0.000 abstract 1
WPYMKLBDIGXBTP-UHFFFAOYSA-N benzoic acid Chemical compound OC(=O)C1=CC=CC=C1 WPYMKLBDIGXBTP-UHFFFAOYSA-N 0.000 abstract 1
230000015572 biosynthetic process Effects 0.000 abstract 1
230000036772 blood pressure Effects 0.000 abstract 1
HPNMFZURTQLUMO-UHFFFAOYSA-N diethylamine Chemical compound CCNCC HPNMFZURTQLUMO-UHFFFAOYSA-N 0.000 abstract 1
230000000694 effects Effects 0.000 abstract 1
RIFGWPKJUGCATF-UHFFFAOYSA-N ethyl chloroformate Chemical compound CCOC(Cl)=O RIFGWPKJUGCATF-UHFFFAOYSA-N 0.000 abstract 1
125000005843 halogen group Chemical group 0.000 abstract 1
238000010438 heat treatment Methods 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
230000007062 hydrolysis Effects 0.000 abstract 1
238000006460 hydrolysis reaction Methods 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
125000002768 hydroxyalkyl group Chemical group 0.000 abstract 1
BUBRXMAMXBDOCS-UHFFFAOYSA-N n,n-dimethyl-2,4-dioxo-1h-3,1-benzoxazine-6-sulfonamide Chemical compound N1C(=O)OC(=O)C2=CC(S(=O)(=O)N(C)C)=CC=C21 BUBRXMAMXBDOCS-UHFFFAOYSA-N 0.000 abstract 1
238000007911 parenteral administration Methods 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
238000002360 preparation method Methods 0.000 abstract 1
238000010992 reflux Methods 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
239000007858 starting material Substances 0.000 abstract 1
238000011200 topical administration Methods 0.000 abstract 1
230000000699 topical effect Effects 0.000 abstract 1
125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C273/00—Preparation of urea or its derivatives, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C273/18—Preparation of urea or its derivatives, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups of substituted ureas
- C07C273/1854—Preparation of urea or its derivatives, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups of substituted ureas by reactions not involving the formation of the N-C(O)-N- moiety

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Epidemiology (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

SE6822/64A 1963-06-05 1964-06-04 SE311644B (de)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
CH702763A CH439319A (de)	1963-06-05	1963-06-05	Verfahren zur Herstellung von N,N-aliphatisch disubstituierten 5-Dialkylsulfamyl-anthranil-säureamiden
CH419664		1964-04-02
CH590064		1964-05-06

Publications (1)

Publication Number	Publication Date
SE311644B true SE311644B (de)	1969-06-23

Family

ID=27174751

Family Applications (3)

Application Number	Title	Priority Date
SE6822/64A SE311644B (de)	1963-06-05	1964-06-04
SE8159/66A SE311517B (de)	1963-06-05	1964-06-04
SE8158/66A SE311646B (de)	1963-06-05	1966-06-15

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
SE8159/66A SE311517B (de)	1963-06-05	1964-06-04
SE8158/66A SE311646B (de)	1963-06-05	1966-06-15

Country Status (11)

Country	Link
US (1)	US3318882A (de)
AT (3)	AT254221B (de)
BE (1)	BE648829A (de)
BR (1)	BR6459789D0 (de)
DE (1)	DE1445629B1 (de)
ES (1)	ES300569A1 (de)
FR (3)	FR1403935A (de)
GB (1)	GB1033268A (de)
MY (1)	MY6900400A (de)
NL (1)	NL140236B (de)
SE (3)	SE311644B (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL104059C (de) *	1955-05-03
US3624202A (en) *	1969-01-22	1971-11-30	Roland Jaques	Process for stilling pain
US3678052A (en) *	1970-06-11	1972-07-18	Squibb & Sons Inc	Benzamide derivatives
CH590259A5 (de) *	1973-07-10	1977-07-29	Ciba Geigy Ag
DE2611705A1 (de) *	1976-03-18	1977-09-22	Josef Dipl Chem Dr Rer N Klosa	N-5-(nitrofurfuryliden-)-1-amino- hydantoin enthaltende kristalloesungsmittel
CH627446A5 (fr) *	1978-01-17	1982-01-15	Debiopharm Sa	Nouveaux derives de la benzamide.
CY1344A (en) *	1978-08-10	1987-01-16	Ciba Geigy Ag	Substituted anthranilic acid amides,process for their preparation,and pharmaceutical compositions containing them

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB882090A (en) *	1958-03-04	1961-11-08	Geigy Ag J R	New sulphamoyl benzamides and processes for the production thereof
US3072656A (en) *	1960-01-22	1963-01-08	Ciba Geigy Corp	2-cycloaliphatic-6-sulfamyl-7-halo(or trihalomethyl)-1, 2, 3, 4-tetrahydro-4-quinazolones

1964
- 1964-05-29 FR FR976292A patent/FR1403935A/fr not_active Expired
- 1964-06-01 GB GB22608/64A patent/GB1033268A/en not_active Expired
- 1964-06-02 US US372086A patent/US3318882A/en not_active Expired - Lifetime
- 1964-06-03 DE DE19641445629D patent/DE1445629B1/de active Pending
- 1964-06-03 ES ES300569A patent/ES300569A1/es not_active Expired
- 1964-06-04 AT AT900565A patent/AT254221B/de active
- 1964-06-04 BE BE648829A patent/BE648829A/xx unknown
- 1964-06-04 AT AT482264A patent/AT254176B/de active
- 1964-06-04 SE SE6822/64A patent/SE311644B/xx unknown
- 1964-06-04 NL NL646406335A patent/NL140236B/xx unknown
- 1964-06-04 AT AT900665A patent/AT261593B/de active
- 1964-06-04 SE SE8159/66A patent/SE311517B/xx unknown
- 1964-06-05 BR BR159789/64A patent/BR6459789D0/pt unknown
- 1964-08-21 FR FR985808A patent/FR3529M/fr not_active Expired
- 1964-08-21 FR FR985807A patent/FR3528M/fr not_active Expired
1966
- 1966-06-15 SE SE8158/66A patent/SE311646B/xx unknown
1969
- 1969-12-31 MY MY1969400A patent/MY6900400A/xx unknown

Also Published As

Publication number	Publication date
DE1445629B1 (de)	1971-08-12
ES300569A1 (es)	1964-11-16
MY6900400A (en)	1969-12-31
SE311517B (de)	1969-06-16
AT254221B (de)	1967-05-10
AT261593B (de)	1968-05-10
FR3529M (fr)	1965-09-06
SE311646B (de)	1969-06-23
BR6459789D0 (pt)	1973-07-17
NL140236B (nl)	1973-11-15
AT254176B (de)	1967-05-10
US3318882A (en)	1967-05-09
FR1403935A (fr)	1965-06-25
BE648829A (de)	1964-12-04
NL6406335A (de)	1964-12-07
FR3528M (fr)	1965-09-06
GB1033268A (en)	1966-06-22

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