SE8006119L - Tripeptidderivat och forfarande for framstellning derav - Google Patents
Tripeptidderivat och forfarande for framstellning deravInfo
- Publication number
- SE8006119L SE8006119L SE8006119A SE8006119A SE8006119L SE 8006119 L SE8006119 L SE 8006119L SE 8006119 A SE8006119 A SE 8006119A SE 8006119 A SE8006119 A SE 8006119A SE 8006119 L SE8006119 L SE 8006119L
- Authority
- SE
- Sweden
- Prior art keywords
- amino
- alkylamino
- lower alkyl
- derivatives
- formula
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- 125000000217 alkyl group Chemical group 0.000 claims abstract 10
- 125000003282 alkyl amino group Chemical group 0.000 claims abstract 8
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims abstract 4
- 125000000539 amino acid group Chemical group 0.000 claims abstract 2
- 240000008042 Zea mays Species 0.000 claims 1
- 235000005824 Zea mays ssp. parviglumis Nutrition 0.000 claims 1
- 235000002017 Zea mays subsp mays Nutrition 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 235000005822 corn Nutrition 0.000 claims 1
- 108090000765 processed proteins & peptides Proteins 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- QNAYBMKLOCPYGJ-UWTATZPHSA-N D-alanine Chemical compound C[C@@H](N)C(O)=O QNAYBMKLOCPYGJ-UWTATZPHSA-N 0.000 abstract 1
- DHMQDGOQFOQNFH-UHFFFAOYSA-N Glycine Chemical compound NCC(O)=O DHMQDGOQFOQNFH-UHFFFAOYSA-N 0.000 abstract 1
- 210000003169 central nervous system Anatomy 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
- C07K5/0823—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Pro-amino acid; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Neurology (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- General Chemical & Material Sciences (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Claims (1)
1. PATENTKRAV Aminoskyddade derivat av en fdrening, corn her formeln H - L - Pro - N - CH - C - Y - R3 (I) 11 R12 ,1 R van i R1 Sr vate, lagre alkyl eller NR4R5, van i R4 och R5 vardera Sr lagre alkyl, R2 Sr vats eller lagre alkyl, R3 Sr amino, lagre alkylamino, di(lagre alkyl)-amino eller amino-(lagre alkyl)-amino och Y Sr aminosyraresten Gly eller 0-Ala, med det fOrbehillet att nar R1 an NR4R5, Mr R3 lagre alkylamino, di(lagre alkyl)-amino eller amino-(lagre alkyl)-amino, corn Sr anvAndbara fOr framstallning av peptidderivat enligt formeln I.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/599,450 US4018912A (en) | 1975-07-28 | 1975-07-28 | Tripeptide derivatives with central nervous system activity and preparation thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SE8006119L true SE8006119L (sv) | 1980-09-02 |
Family
ID=24399667
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7608484A SE431330B (sv) | 1975-07-28 | 1976-07-27 | Forfarande for framstellning av tripeptidderivat, vilka har cns-aktivitet |
| SE8006119A SE8006119L (sv) | 1975-07-28 | 1980-09-02 | Tripeptidderivat och forfarande for framstellning derav |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7608484A SE431330B (sv) | 1975-07-28 | 1976-07-27 | Forfarande for framstellning av tripeptidderivat, vilka har cns-aktivitet |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US4018912A (sv) |
| JP (1) | JPS6033854B2 (sv) |
| BE (1) | BE844603A (sv) |
| CA (1) | CA1062250A (sv) |
| CH (1) | CH621111A5 (sv) |
| DE (1) | DE2633976A1 (sv) |
| FR (1) | FR2319378A1 (sv) |
| GB (1) | GB1523685A (sv) |
| SE (2) | SE431330B (sv) |
| SU (1) | SU632299A3 (sv) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4093713A (en) * | 1977-02-28 | 1978-06-06 | Ayerst Mckenna & Harrison Ltd. | Dipeptide derivatives with central nervous system activity and preparation thereof |
| DE3226241A1 (de) * | 1982-07-14 | 1984-01-26 | Basf Ag, 6700 Ludwigshafen | N-acylderivate von peptiden, ihre herstellung und verwendung bei der bekaempfung von krankheiten und mittel dafuer |
| DE3226242A1 (de) * | 1982-07-14 | 1984-01-26 | Basf Ag, 6700 Ludwigshafen | N-acylderivate von dipeptiden, ihre herstellung und verwendung bei der therapie von krankheiten und mittel dafuer |
| US5190924A (en) * | 1991-02-13 | 1993-03-02 | Boc Health Care, Inc. | Peptide amides and amide dimers useful as muscle relaxants |
| US6767897B2 (en) * | 1994-05-04 | 2004-07-27 | Innapharma, Inc. | Therapeutic uses of tri-, tetra-, penta-, and polypeptides |
| US5767083A (en) * | 1994-05-04 | 1998-06-16 | Innapharma, Inc. | Tri-, tetra-, penta-, and polypeptides and their therapeutic use as an antidepressant agent |
| US5589460A (en) * | 1994-05-04 | 1996-12-31 | Innapharma, Inc. | Tri-, tetra-, penta-, and polypeptides and their therapeutic use as an antidepressant agent |
| US6489300B1 (en) * | 1997-07-31 | 2002-12-03 | Eugene D. Thorsett | Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 |
| DE19813849A1 (de) * | 1998-03-27 | 1999-09-30 | Degussa | Verfahren zur einstufigen Umsalzung und Aufreinigung von Oligopeptiden |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1033904A (en) * | 1962-03-30 | 1966-06-22 | Geigy Ag J R | Process for the production of a new nonapeptidamide |
| NL6707845A (sv) * | 1966-06-11 | 1967-12-12 | ||
| BE787908A (fr) * | 1971-08-24 | 1973-02-23 | Abbott Lab | Medicament antidepressif et antiparkinsonien |
| US3888840A (en) * | 1973-02-07 | 1975-06-10 | American Home Prod | Novel hydrazinocarboxamide derivatives and preparation thereof |
-
1975
- 1975-07-28 US US05/599,450 patent/US4018912A/en not_active Expired - Lifetime
-
1976
- 1976-06-28 CA CA255,845A patent/CA1062250A/en not_active Expired
- 1976-07-22 CH CH940676A patent/CH621111A5/fr not_active IP Right Cessation
- 1976-07-27 SU SU762385906A patent/SU632299A3/ru active
- 1976-07-27 SE SE7608484A patent/SE431330B/sv unknown
- 1976-07-27 FR FR7622908A patent/FR2319378A1/fr active Granted
- 1976-07-27 GB GB31222/76A patent/GB1523685A/en not_active Expired
- 1976-07-28 BE BE169315A patent/BE844603A/xx not_active IP Right Cessation
- 1976-07-28 JP JP51091263A patent/JPS6033854B2/ja not_active Expired
- 1976-07-28 DE DE19762633976 patent/DE2633976A1/de not_active Ceased
-
1980
- 1980-09-02 SE SE8006119A patent/SE8006119L/sv not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| JPS6033854B2 (ja) | 1985-08-05 |
| SE431330B (sv) | 1984-01-30 |
| CA1062250A (en) | 1979-09-11 |
| US4018912A (en) | 1977-04-19 |
| BE844603A (fr) | 1977-01-28 |
| FR2319378A1 (fr) | 1977-02-25 |
| DE2633976A1 (de) | 1977-02-10 |
| SU632299A3 (ru) | 1978-11-05 |
| GB1523685A (en) | 1978-09-06 |
| FR2319378B1 (sv) | 1979-05-04 |
| CH621111A5 (sv) | 1981-01-15 |
| JPS5223070A (en) | 1977-02-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| NAV | Patent application has lapsed |
Ref document number: 8006119-5 |