SE8107520L - 7-acylaminocefalosporansyraderivat och forfarande for framstellning derav - Google Patents

7-acylaminocefalosporansyraderivat och forfarande for framstellning derav

Info

Publication number: SE8107520L
Authority: SE; Sweden
Prior art keywords: alkyl; acid derivatives; derivatives; protected; procedures
Prior art date: 1980-12-15

Application number

SE8107520A

Other languages

Unknown language ( )

English (en)

Swedish (sv)

Inventor

T Teraji

K Takai

S Nishino

I Ueda

F Shimojo

T Takaya

H Takasugi

Original Assignee

Fujisawa Pharmaceutical Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1980-12-15

Filing date

1981-12-15

Publication date

1982-06-16

1980-12-23 Priority claimed from JP18329980A external-priority patent/JPS57106684A/ja

1981-12-15 Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co

1982-06-16 Publication of SE8107520L publication Critical patent/SE8107520L/

Links

239000002253 acid Substances 0.000 title abstract 2
238000000034 method Methods 0.000 title abstract 2
125000000217 alkyl group Chemical group 0.000 abstract 8
125000005194 alkoxycarbonyloxy group Chemical group 0.000 abstract 2
125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 2
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 2
FZEVMBJWXHDLDB-ZCFIWIBFSA-N (6r)-5-thia-1-azabicyclo[4.2.0]oct-2-en-8-one Chemical compound S1CC=CN2C(=O)C[C@H]21 FZEVMBJWXHDLDB-ZCFIWIBFSA-N 0.000 abstract 1
SXBDXXFTJVHSAF-ZCFIWIBFSA-N (6r)-5-thia-1-azabicyclo[4.2.0]oct-3-en-8-one Chemical compound S1C=CCN2C(=O)C[C@H]21 SXBDXXFTJVHSAF-ZCFIWIBFSA-N 0.000 abstract 1
125000004423 acyloxy group Chemical group 0.000 abstract 1
125000003545 alkoxy group Chemical group 0.000 abstract 1
230000000845 anti-microbial effect Effects 0.000 abstract 1
125000005333 aroyloxy group Chemical group 0.000 abstract 1
125000000852 azido group Chemical group *N=[N+]=[N-] 0.000 abstract 1
125000005201 cycloalkylcarbonyloxy group Chemical group 0.000 abstract 1
125000000623 heterocyclic group Chemical group 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
125000005633 phthalidyl group Chemical group 0.000 abstract 1
125000001424 substituent group Chemical group 0.000 abstract 1
125000000446 sulfanediyl group Chemical group *S* 0.000 abstract 1
125000000475 sulfinyl group Chemical group [*:2]S([*:1])=O 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Cephalosporin Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

SE8107520A 1980-12-15 1981-12-15 7-acylaminocefalosporansyraderivat och forfarande for framstellning derav SE8107520L (sv)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
GB8040108		1980-12-15
JP18329980A JPS57106684A (en)	1980-12-23	1980-12-23	Syn-isomer of 7-substituted-3-cephem-4-carboxylic acid ester and its preparation
GB8041516		1980-12-30
GB8108135		1981-03-16

Publications (1)

Publication Number	Publication Date
SE8107520L true SE8107520L (sv)	1982-06-16

Family

ID=27449218

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE8107520A SE8107520L (sv)	1980-12-15	1981-12-15	7-acylaminocefalosporansyraderivat och forfarande for framstellning derav

Country Status (11)

Country	Link
US (1)	US4477447A (cs)
AT (1)	AT376983B (cs)
DE (1)	DE3149578A1 (cs)
DK (1)	DK554481A (cs)
ES (1)	ES8303422A1 (cs)
FR (1)	FR2496106B1 (cs)
GB (1)	GB2092575B (cs)
GR (1)	GR76690B (cs)
IT (1)	IT1142096B (cs)
NL (1)	NL8105658A (cs)
SE (1)	SE8107520L (cs)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4703046A (en) *	1978-09-08	1987-10-27	Fujisawa Pharmaceutical Co., Ltd.	Cephem compounds and processes for preparation thereof
EP0136266A3 (de) *	1983-09-22	1986-03-26	Ciba-Geigy Ag	7beta-Acylamido-3-cephem-4-carbonsäureester, Verfahren zu ihrer Herstellung, pharmazeutische Präparate, welche diese Verbindungen enthalten, und Verwendung von letzteren
US4914091A (en) *	1984-04-02	1990-04-03	American Cyanamid Company	Esters of cephalosporin derivitives
US5389625A (en) *	1989-10-28	1995-02-14	Kyoto Pharmaceutical Industries, Ltd.	Cephalosporin compounds
EP2753326A4 (en)	2011-09-09	2015-04-15	Cubist Pharm Inc	METHOD FOR THE TREATMENT OF INTRAPULMONARY INFECTIONS
US8809314B1 (en)	2012-09-07	2014-08-19	Cubist Pharmacueticals, Inc.	Cephalosporin compound
US8476425B1 (en)	2012-09-27	2013-07-02	Cubist Pharmaceuticals, Inc.	Tazobactam arginine compositions
NZ700372A (en)	2013-03-15	2016-01-29	Merck Sharp & Dohme	Ceftolozane antibiotic compositions
US20140274993A1 (en)	2013-03-15	2014-09-18	Cubist Pharmaceuticals, Inc.	Ceftolozane-tazobactam pharmaceutical compositions
US9872906B2 (en)	2013-03-15	2018-01-23	Merck Sharp & Dohme Corp.	Ceftolozane antibiotic compositions
EP3043797B1 (en)	2013-09-09	2020-04-08	Merck Sharp & Dohme Corp.	Treating infections with ceftolozane/tazobactam in subjects having impaired renal function
US8906898B1 (en)	2013-09-27	2014-12-09	Calixa Therapeutics, Inc.	Solid forms of ceftolozane

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2714880A1 (de) *	1977-04-02	1978-10-26	Hoechst Ag	Cephemderivate und verfahren zu ihrer herstellung
US4370326A (en) *	1977-09-13	1983-01-25	Fujisawa Pharmaceutical Co., Ltd.	Cephem compounds and composition
MA18686A1 (fr) *	1978-07-07	1980-10-01	Ciba Geigy Ag	Composes aminothiazoliques
DE2967053D1 (en) *	1978-09-12	1984-07-19	Fujisawa Pharmaceutical Co	Starting compounds for preparing cephem compounds and processes for their preparation
JPS5543011A (en) *	1978-09-20	1980-03-26	Shionogi & Co Ltd	7-halothiazolylalkoxyiminoacetamido-3-cephem compound
GB2111043B (en) *	1980-12-12	1985-02-06	Ciba Geigy Ag	Novel cephalosporin esters
AU8166182A (en) *	1981-03-23	1982-09-30	Kyoto Yakuhin Kogyo K.K.	Cephalosporin derivatives
JPS57193489A (en) *	1981-05-21	1982-11-27	Fujisawa Pharmaceut Co Ltd	Syn-isomer of 7-substituted-3-cephem-4-carboxylic acid ester and its preparation

1981
- 1981-12-14 DK DK554481A patent/DK554481A/da not_active Application Discontinuation
- 1981-12-14 IT IT8125581A patent/IT1142096B/it active
- 1981-12-14 ES ES507942A patent/ES8303422A1/es not_active Expired
- 1981-12-15 GR GR66790A patent/GR76690B/el unknown
- 1981-12-15 NL NL8105658A patent/NL8105658A/nl not_active Application Discontinuation
- 1981-12-15 FR FR8123457A patent/FR2496106B1/fr not_active Expired
- 1981-12-15 SE SE8107520A patent/SE8107520L/ not_active Application Discontinuation
- 1981-12-15 DE DE19813149578 patent/DE3149578A1/de not_active Withdrawn
- 1981-12-15 GB GB8137724A patent/GB2092575B/en not_active Expired
- 1981-12-15 AT AT0536881A patent/AT376983B/de not_active IP Right Cessation
1982
- 1982-02-24 US US06/351,858 patent/US4477447A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
ES507942A0 (es)	1983-02-01
DE3149578A1 (de)	1982-09-09
DK554481A (da)	1982-06-16
FR2496106A1 (fr)	1982-06-18
US4477447A (en)	1984-10-16
IT1142096B (it)	1986-10-08
AT376983B (de)	1985-01-25
IT8125581A0 (it)	1981-12-14
GB2092575A (en)	1982-08-18
GB2092575B (en)	1985-07-03
ATA536881A (de)	1984-06-15
ES8303422A1 (es)	1983-02-01
NL8105658A (nl)	1982-07-01
FR2496106B1 (fr)	1985-07-19
GR76690B (cs)	1984-08-24

Similar Documents

Publication	Publication Date	Title
HK98486A (en)	1986-12-24	Quinoline carboxylic acid derivatives and their preparation
SE8107520L (sv)	1982-06-16	7-acylaminocefalosporansyraderivat och forfarande for framstellning derav
FR2479229B1 (fr)	1986-01-17	Nouveaux derives des cephalosporines, leur procede de preparation et les medicaments utilisables comme antibiotiques qui contiennent lesdits derives
SE8202961L (sv)	1982-11-13	Cefalosporinderivat och forfarande for deras framstellning
ATE51223T1 (de)	1990-04-15	Derivate der 2-azetidinon-1-sulfonsaeure, ihre herstellung und verwendung.
IE37916B1 (en)	1977-11-09	Trifluoromethylmercaptoacetamidocephalosporins
ES8107224A1 (es)	1981-10-01	Un procedimiento para la preparacion de derivados acidos penem-carboxilicos
PT729455E (pt)	2005-01-31	Arilpiperazinas derivadas de indol como ligados para os receptores 5ht1-like, 5ht1b e 5ht1d
IL80114A0 (en)	1986-12-31	Quinoline derivatives,their manufacture and pharmaceutical compositions containing them
SE8207302L (sv)	1982-12-21	Nya 2-pyrrolidonforeningar och forfarande for framstellning av desamma
FI882477A0 (fi)	1988-05-26	>nya alkansulfonanilidderivat, foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska blandningar.
ES8305366A1 (es)	1983-04-01	"procedimiento para la preparacion de derivados de penem".
ES8105329A1 (es)	1981-06-01	Procedimiento para la obtencion de compuestos de acido ami- notiazolacetamido-3-cefem-4-carboxilico.
ES2132245T3 (es)	1999-08-16	Derivados de 1-azaadamantano como agonistas o antagonistas de 5-ht.
ES8200691A1 (es)	1981-11-01	Procedimiento para la preparacion de nuevas cefalosporinas
SE7907159L (sv)	1980-03-01	3,7-disubstituerade 3-cefem-4-karboxylsyraforeningar och forfarande for deras framstelllning
ATE92927T1 (de)	1993-08-15	1-carboxy-1-vinyloxyiminoaminothiazolcephalosporin-derivate und deren herstellung.
FI872997A0 (fi)	1987-07-07	Amidderivat.
US4013765A (en)	1977-03-22	Compositions and methods for treating bacterial infections with substituted acetamidocephalosporins
US3957770A (en)	1976-05-18	Substituted acetamidocephalosporins
US3998818A (en)	1976-12-21	Trifluoroethylmercapto, -sulfinyl or -sulfonyl acetamidocephalosporins
US3998819A (en)	1976-12-21	Trifluoroethyl-mercapto, -sulfinyl or -sulfonyl acetamidocephalosporins
FI823732A0 (fi)	1982-11-02	Nya 1-furyl-3,4-dihydroisokinoliner, laekemedel innehaollande dessa samt deras framstaellningsfoerfaranden och deras anvaendning
US3963711A (en)	1976-06-15	Cyanomethyl sulfinyl- and sulfonyl-acetamido cephalosporins
US4075338A (en)	1978-02-21	Substituted acetamidocephalosporins

Legal Events

Date

Code

Title

Description

1995-02-28

NAV

Patent application has lapsed

Ref document number: 8107520-2

Format of ref document f/p: F