SE9302396D0 - A novel compound form - Google Patents

A novel compound form

Info

Publication number
SE9302396D0
SE9302396D0 SE19939302396A SE9302396A SE9302396D0 SE 9302396 D0 SE9302396 D0 SE 9302396D0 SE 19939302396 A SE19939302396 A SE 19939302396A SE 9302396 A SE9302396 A SE 9302396A SE 9302396 D0 SE9302396 D0 SE 9302396D0
Authority
SE
Sweden
Prior art keywords
novel compound
compound form
crystallinity
manufacture
useful
Prior art date
Application number
SE19939302396A
Other languages
English (en)
Swedish (sv)
Inventor
Aake *Kaellstroem Lars
Annelie *Nygren Monica
Original Assignee
Ab Astra
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20390588&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SE9302396(D0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority to SE19939302396A priority Critical patent/SE9302396D0/xx
Application filed by Ab Astra filed Critical Ab Astra
Publication of SE9302396D0 publication Critical patent/SE9302396D0/xx
Priority to TW083105710A priority patent/TW504509B/zh
Priority to HR940385A priority patent/HRP940385B1/xx
Priority to IL11019094A priority patent/IL110190A/xx
Priority to SA94150058A priority patent/SA94150058B1/ar
Priority to IS4186A priority patent/IS2075B/is
Priority to MYPI94001774A priority patent/MY113274A/en
Priority to ZA944933A priority patent/ZA944933B/xx
Priority to EG40794A priority patent/EG21437A/xx
Priority to MA23567A priority patent/MA23257A1/fr
Priority to NZ268693A priority patent/NZ268693A/en
Priority to CN94192733A priority patent/CN1064680C/zh
Priority to SI9430414T priority patent/SI0707580T1/xx
Priority to HU9503873A priority patent/HU226861B1/hu
Priority to AU71981/94A priority patent/AU679766B2/en
Priority to EP94921154A priority patent/EP0707580B1/fr
Priority to JP50400595A priority patent/JP3635432B2/ja
Priority to SK22-96A priority patent/SK281230B6/sk
Priority to AT94921154T priority patent/ATE212628T1/de
Priority to DE0707580T priority patent/DE707580T1/de
Priority to DK94921154T priority patent/DK0707580T3/da
Priority to PT94921154T priority patent/PT707580E/pt
Priority to TNTNSN94079A priority patent/TNSN94079A1/fr
Priority to ES94921154T priority patent/ES2100136T3/es
Priority to DE69429774T priority patent/DE69429774T2/de
Priority to RU96102079A priority patent/RU2139868C1/ru
Priority to BR9406940A priority patent/BR9406940A/pt
Priority to UA96010059A priority patent/UA43343C2/uk
Priority to US08/313,342 priority patent/US5900424A/en
Priority to CZ199669A priority patent/CZ288933B6/cs
Priority to EP01117362A priority patent/EP1164132A3/fr
Priority to HK98109227.9A priority patent/HK1008329B/en
Priority to KR1019960700051A priority patent/KR100353783B1/ko
Priority to CA002166794A priority patent/CA2166794C/fr
Priority to YU43694A priority patent/YU49193B/sh
Priority to SG1996004887A priority patent/SG52464A1/en
Priority to PCT/SE1994/000680 priority patent/WO1995001977A1/fr
Priority to PL94312440A priority patent/PL175999B1/pl
Priority to MX9405217A priority patent/MX9405217A/es
Priority to EE9400405A priority patent/EE03127B1/xx
Priority to DZ940071A priority patent/DZ1792A1/fr
Priority to NO960068A priority patent/NO308702B1/no
Priority to FI960101A priority patent/FI114154B/fi
Priority to GR970300015T priority patent/GR970300015T1/el
Priority to JP2001293480A priority patent/JP3878826B2/ja

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Contacts (AREA)
  • Conductive Materials (AREA)
  • Electroplating Methods And Accessories (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Fats And Perfumes (AREA)
  • Glass Compositions (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Powder Metallurgy (AREA)
  • Medicinal Preparation (AREA)
SE19939302396A 1993-07-09 1993-07-09 A novel compound form SE9302396D0 (sv)

Priority Applications (45)

Application Number Priority Date Filing Date Title
SE19939302396A SE9302396D0 (sv) 1993-07-09 1993-07-09 A novel compound form
TW083105710A TW504509B (en) 1993-07-09 1994-06-23 A novel form of magnesium omeprazole, its preparation process and pharmaceutical composition comprising the same
HR940385A HRP940385B1 (en) 1993-07-09 1994-07-01 Novel compound form
IL11019094A IL110190A (en) 1993-07-09 1994-07-01 Magnesium omeprazole with crystallinity higher than 70% process for its preparation and its use in the manufacture of medicaments for inhibiting gastric acid secretion and for obtaining gastric mucosa protective activity
SA94150058A SA94150058B1 (ar) 1993-07-09 1994-07-04 مركب ملح مغنسيوم الاومبرازول
IS4186A IS2075B (is) 1993-07-09 1994-07-05 Aðferð til að framleiða magnesíumómeprasól
MA23567A MA23257A1 (fr) 1993-07-09 1994-07-07 Nouvelle forme de compose demagnesium d'omeprazole etson utilisation .
EG40794A EG21437A (en) 1993-07-09 1994-07-07 Method for preparing magnesium omeprazole compounds useful for inhibiting gastric acid sectretion
MYPI94001774A MY113274A (en) 1993-07-09 1994-07-07 Omeprazole magnesium salt form
ZA944933A ZA944933B (en) 1993-07-09 1994-07-07 A novel compound form
PL94312440A PL175999B1 (pl) 1993-07-09 1994-07-08 Omeprazol magnezowy i sposób wytwarzania omeprazolu magnezowego oraz kompozycja farmaceutyczna go zawierająca
MX9405217A MX9405217A (es) 1993-07-09 1994-07-08 Proceso para la fabricacion de sal de magnesio de omeprazol, productoobtenido a partir del mismo y composicion farmaceutica que contiene dichoproducto.
PT94921154T PT707580E (pt) 1993-07-09 1994-07-08 Omeprazole magnesio
UA96010059A UA43343C2 (uk) 1993-07-09 1994-07-08 Магнієва сіль омепразолу, спосіб її одержання, фармацевтична композиція, спосіб лікування
SI9430414T SI0707580T1 (en) 1993-07-09 1994-07-08 Magnesium omeprazole
HU9503873A HU226861B1 (en) 1993-07-09 1994-07-08 Magnesium salt of omeprazole
AU71981/94A AU679766B2 (en) 1993-07-09 1994-07-08 Magnesium omeprazole
EP94921154A EP0707580B1 (fr) 1993-07-09 1994-07-08 Omeprazole de magnesium
JP50400595A JP3635432B2 (ja) 1993-07-09 1994-07-08 オメプラゾールマグネシウムの製法
SK22-96A SK281230B6 (sk) 1993-07-09 1994-07-08 Magnézium omeprazol, spôsob jeho výroby, farmaceutické prípravky s jeho obsahom a jeho použitie
AT94921154T ATE212628T1 (de) 1993-07-09 1994-07-08 Magnesium-omeprazol
DE0707580T DE707580T1 (de) 1993-07-09 1994-07-08 Magnesium-omeprazol
DK94921154T DK0707580T3 (da) 1993-07-09 1994-07-08 Magnesiumomeprazol
NZ268693A NZ268693A (en) 1993-07-09 1994-07-08 Magnesium omeprazole having a degree of crystallinity greater than 70%
TNTNSN94079A TNSN94079A1 (fr) 1993-07-09 1994-07-08 Une nouvelle forme de compose
ES94921154T ES2100136T3 (es) 1993-07-09 1994-07-08 Omeprazol de magnesio.
DE69429774T DE69429774T2 (de) 1993-07-09 1994-07-08 Magnesium-omeprazol
RU96102079A RU2139868C1 (ru) 1993-07-09 1994-07-08 Магниевая соль омепразола, способ ее получения, фармацевтическая композиция, способ лечения
BR9406940A BR9406940A (pt) 1993-07-09 1994-07-08 Magnésio-omeprazol processo para a preparação de magnésio-omeprazol composição farmacêutica formulação farmacêutica para a administração oral forumulação de tablete uso do magnesio-omeprazol processo para a inibição da secreção de ácido gástrico em mamiferos e no homem e processo para o tratamento das doenças relacionadas com o ácido gastrico em mamiferos e no homem
CN94192733A CN1064680C (zh) 1993-07-09 1994-07-08 奥美拉唑镁的制备方法
US08/313,342 US5900424A (en) 1993-07-09 1994-07-08 Omeprazole magnesium salt form
CZ199669A CZ288933B6 (cs) 1993-07-09 1994-07-08 Magnezium omeprazol
EP01117362A EP1164132A3 (fr) 1993-07-09 1994-07-08 Omeprazole de magnésium cristallin
HK98109227.9A HK1008329B (en) 1993-07-09 1994-07-08 Magnesium omeprazole
KR1019960700051A KR100353783B1 (ko) 1993-07-09 1994-07-08 마그네슘오메프라졸
CA002166794A CA2166794C (fr) 1993-07-09 1994-07-08 Derive magnesien d'omeprazole
YU43694A YU49193B (sh) 1993-07-09 1994-07-08 Magnezijum omeprazol i postupak za dobijanje ovog jedinjenja
SG1996004887A SG52464A1 (en) 1993-07-09 1994-07-08 A novel compound form
PCT/SE1994/000680 WO1995001977A1 (fr) 1993-07-09 1994-07-08 Omeprazole de magnesium
EE9400405A EE03127B1 (et) 1993-07-09 1994-11-17 Kristalne magneesiumomeprasool, selle valmistamise protsess, seda sisaldavad ravimpreparaadid ja nende kasutamine
DZ940071A DZ1792A1 (fr) 1993-07-09 1994-11-27 Une nouvelle forme de composé.
NO960068A NO308702B1 (no) 1993-07-09 1996-01-05 Magnesiumomeprazol, fremgangsmÕte for fremstilling derav, farmasøytisk preparat inneholdende magnesiumomeprazol og anvendelse derav
FI960101A FI114154B (fi) 1993-07-09 1996-01-09 Menetelmä terapeuttisesti käyttökelpoisen magnesiumomepratsolin valmistamiseksi
GR970300015T GR970300015T1 (en) 1993-07-09 1997-05-30 Magnesium omeprazole
JP2001293480A JP3878826B2 (ja) 1993-07-09 2001-09-26 オメプラゾールマグネシウム

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE19939302396A SE9302396D0 (sv) 1993-07-09 1993-07-09 A novel compound form

Publications (1)

Publication Number Publication Date
SE9302396D0 true SE9302396D0 (sv) 1993-07-09

Family

ID=20390588

Family Applications (1)

Application Number Title Priority Date Filing Date
SE19939302396A SE9302396D0 (sv) 1993-07-09 1993-07-09 A novel compound form

Country Status (41)

Country Link
US (1) US5900424A (fr)
EP (2) EP0707580B1 (fr)
JP (2) JP3635432B2 (fr)
KR (1) KR100353783B1 (fr)
CN (1) CN1064680C (fr)
AT (1) ATE212628T1 (fr)
AU (1) AU679766B2 (fr)
BR (1) BR9406940A (fr)
CA (1) CA2166794C (fr)
CZ (1) CZ288933B6 (fr)
DE (2) DE69429774T2 (fr)
DK (1) DK0707580T3 (fr)
DZ (1) DZ1792A1 (fr)
EE (1) EE03127B1 (fr)
EG (1) EG21437A (fr)
ES (1) ES2100136T3 (fr)
FI (1) FI114154B (fr)
GR (1) GR970300015T1 (fr)
HR (1) HRP940385B1 (fr)
HU (1) HU226861B1 (fr)
IL (1) IL110190A (fr)
IS (1) IS2075B (fr)
MA (1) MA23257A1 (fr)
MX (1) MX9405217A (fr)
MY (1) MY113274A (fr)
NO (1) NO308702B1 (fr)
NZ (1) NZ268693A (fr)
PL (1) PL175999B1 (fr)
PT (1) PT707580E (fr)
RU (1) RU2139868C1 (fr)
SA (1) SA94150058B1 (fr)
SE (1) SE9302396D0 (fr)
SG (1) SG52464A1 (fr)
SI (1) SI0707580T1 (fr)
SK (1) SK281230B6 (fr)
TN (1) TNSN94079A1 (fr)
TW (1) TW504509B (fr)
UA (1) UA43343C2 (fr)
WO (1) WO1995001977A1 (fr)
YU (1) YU49193B (fr)
ZA (1) ZA944933B (fr)

Families Citing this family (95)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6875872B1 (en) * 1993-05-28 2005-04-05 Astrazeneca Compounds
SE9301830D0 (sv) * 1993-05-28 1993-05-28 Ab Astra New compounds
SE9302395D0 (sv) * 1993-07-09 1993-07-09 Ab Astra New pharmaceutical formulation
SE9302396D0 (sv) * 1993-07-09 1993-07-09 Ab Astra A novel compound form
BR9508261A (pt) * 1994-07-08 1997-12-23 Astra Ab Formulação oral entericamente revestida uso da mesma processo para preparer a formulação inibir a secreção de ácido gástrico em mamíferos e no ser humano e tratar doenças relacionadas ao ácido gástrico em maníferos e no ser humano e pacote de empola de pressão transversal
DK1078628T3 (da) 1994-07-08 2009-02-23 Astrazeneca Ab Tabletteret flerenhedsdoseringsform
SE9500478D0 (sv) * 1995-02-09 1995-02-09 Astra Ab New pharmaceutical formulation and process
US5840737A (en) 1996-01-04 1998-11-24 The Curators Of The University Of Missouri Omeprazole solution and method for using same
US6699885B2 (en) * 1996-01-04 2004-03-02 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and methods of using same
US6489346B1 (en) * 1996-01-04 2002-12-03 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US6645988B2 (en) * 1996-01-04 2003-11-11 Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
SE9600070D0 (sv) * 1996-01-08 1996-01-08 Astra Ab New oral pharmaceutical dosage forms
SE508669C2 (sv) * 1996-04-26 1998-10-26 Astra Ab Nytt förfarande
US6623759B2 (en) * 1996-06-28 2003-09-23 Astrazeneca Ab Stable drug form for oral administration with benzimidazole derivatives as active ingredient and process for the preparation thereof
TW385306B (en) * 1996-11-14 2000-03-21 Takeda Chemical Industries Ltd Method for producing crystals of benzimidazole derivatives
SE510666C2 (sv) * 1996-12-20 1999-06-14 Astra Ab Nya Kristallmodifikationer
SE9702000D0 (sv) * 1997-05-28 1997-05-28 Astra Ab New pharmaceutical formulation
SE510650C2 (sv) 1997-05-30 1999-06-14 Astra Ab Ny förening
US6747155B2 (en) 1997-05-30 2004-06-08 Astrazeneca Ab Process
US6174548B1 (en) 1998-08-28 2001-01-16 Andrx Pharmaceuticals, Inc. Omeprazole formulation
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US6048981A (en) * 1998-04-22 2000-04-11 Torcan Chemical Ltd. Magnesium omeprazole and process for its preparation
DE19843413C1 (de) * 1998-08-18 2000-03-30 Byk Gulden Lomberg Chem Fab Neue Salzform von Pantoprazol
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US6403616B1 (en) 1998-11-18 2002-06-11 Astrazeneca Ab Chemical process and pharmaceutical formulation
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