SK178698A3 - Treating urinary incontinence using (s)-oxybutynin and (s)-desethyloxybutynin - Google Patents

Treating urinary incontinence using (s)-oxybutynin and (s)-desethyloxybutynin Download PDF

Info

Publication number: SK178698A3
Authority: SK; Slovakia
Prior art keywords: oxybutynin; pharmaceutically acceptable; deethyloxybutynin; acceptable salt; deo
Prior art date: 1996-06-28

Application number

SK1786-98A

Other languages

English (en)

Slovak (sk)

Inventor

Gunnar Aberg

John R Mccullough

Original Assignee

Sepracor Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-06-28

Filing date

1997-06-27

Publication date

1999-09-10

1997-06-27 Application filed by Sepracor Inc filed Critical Sepracor Inc

1999-09-10 Publication of SK178698A3 publication Critical patent/SK178698A3/sk

Links

206010046543 Urinary incontinence Diseases 0.000 title claims abstract description 12
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SNIBJKHIKIIGPR-HXUWFJFHSA-N 4-(ethylamino)but-2-ynyl (2s)-2-cyclohexyl-2-hydroxy-2-phenylacetate Chemical compound C1([C@@](O)(C(=O)OCC#CCNCC)C=2C=CC=CC=2)CCCCC1 SNIBJKHIKIIGPR-HXUWFJFHSA-N 0.000 title abstract 3
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/06—Anti-spasmodics

Landscapes

Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Urology & Nephrology (AREA)
Engineering & Computer Science (AREA)
Emergency Medicine (AREA)
Epidemiology (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

SK1786-98A 1996-06-28 1997-06-27 Treating urinary incontinence using (s)-oxybutynin and (s)-desethyloxybutynin SK178698A3 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US08/671,976 US5736577A (en)	1995-01-31	1996-06-28	Methods and compositions for treating urinary incontinence using optically pure (S)-oxybutynin
PCT/US1997/011570 WO1998000126A1 (en)	1996-06-28	1997-06-27	Treating urinary incontinence using (s)-oxybutynin and (s)-desethyloxybutynin

Publications (1)

Publication Number	Publication Date
SK178698A3 true SK178698A3 (en)	1999-09-10

Family

ID=24696647

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK1786-98A SK178698A3 (en)	1996-06-28	1997-06-27	Treating urinary incontinence using (s)-oxybutynin and (s)-desethyloxybutynin

Country Status (14)

Country	Link
US (1)	US5736577A (pt)
EP (1)	EP0914113A1 (pt)
JP (1)	JP2000513724A (pt)
AU (1)	AU732568B2 (pt)
BR (1)	BR9710031A (pt)
CA (1)	CA2257121C (pt)
CZ (1)	CZ428398A3 (pt)
NO (1)	NO985896D0 (pt)
NZ (1)	NZ333282A (pt)
PL (1)	PL190483B1 (pt)
RU (1)	RU2195276C2 (pt)
SK (1)	SK178698A3 (pt)
UA (1)	UA61916C2 (pt)
WO (1)	WO1998000126A1 (pt)

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AU2018299A (en) *	1997-12-31	1999-07-19	Sepracor, Inc.	(s)-procyclidine for treating urinary incontinence
US20010038855A1 (en) *	1998-06-05	2001-11-08	Desjardin Michael A.	Dosage form for administering prescribed dose
AU767877B2 (en) *	1999-05-20	2003-11-27	Sepracor, Inc.	Methods for treatment of asthma using S-oxybutynin
WO2000076490A2 (en) *	1999-06-10	2000-12-21	Sepracor Inc.	Methods and compositions for treating urinary frequency and urgency using optically pure (s)-oxybutynin
US6248359B1 (en)	2000-01-05	2001-06-19	Laboratorios Phoenix U.S.A., Inc.	Multi-tablet oxybutynin system for treating incontinence
US7029694B2 (en) *	2000-04-26	2006-04-18	Watson Laboratories, Inc.	Compositions and methods for transdermal oxybutynin therapy
US7179483B2 (en) *	2000-04-26	2007-02-20	Watson Pharmaceuticals, Inc.	Compositions and methods for transdermal oxybutynin therapy
US20030124177A1 (en) *	2000-04-26	2003-07-03	Watson Pharmaceuticals, Inc.	Compositions and methods for transdermal oxybutynin therapy
CN101843601A (zh) *	2000-04-26	2010-09-29	沃特森药物公司	最小化与奥昔布宁疗法有关的副作用
ATE485837T1 (de) *	2000-08-03	2010-11-15	Antares Pharma Ipl Ag	Zusammensetzung zur transdermalen und/oder transmukosalen verabreichung von wirkstoffen, die ausreichende therapeutische spiegel garantiert
US7198801B2 (en) *	2000-08-03	2007-04-03	Antares Pharma Ipl Ag	Formulations for transdermal or transmucosal application
US20070225379A1 (en) *	2001-08-03	2007-09-27	Carrara Dario Norberto R	Transdermal delivery of systemically active central nervous system drugs
US8980290B2 (en)	2000-08-03	2015-03-17	Antares Pharma Ipl Ag	Transdermal compositions for anticholinergic agents
DE10041478A1 (de)	2000-08-24	2002-03-14	Sanol Arznei Schwarz Gmbh	Neue pharmazeutische Zusammensetzung
US6545046B2 (en)	2000-08-30	2003-04-08	Theramax Inc.	Method for enhanced delivery of oxybutynin and compositions thereof
DE10103262A1 (de) *	2001-01-25	2002-08-01	Axel Schmidt-Dossi	Arzneimittel gegen Blasenfunktionsstörung
WO2002076426A2 (en) *	2001-03-27	2002-10-03	Galen (Chemicals) Limited	Intravaginal drug delivery devices for the administration of an antimicrobial agent
JP2004532874A (ja) *	2001-04-03	2004-10-28	アリックスセラピューティクス	抗コリン作用性化合物および使用法
US20030027856A1 (en) *	2001-06-29	2003-02-06	Aberg A.K. Gunnar	Tolterodine metabolites
DE10146275A1 (de)	2001-09-18	2003-04-24	Gruenenthal Gmbh	Kombination ausgewählter Opioide mit Muscarin-Antagonisten zur Therapie der Harninkontinenz
MXPA04003806A (es) *	2001-11-05	2005-04-08	Upjohn Co	Aerosol antimuscarinico.
US7921999B1 (en)	2001-12-20	2011-04-12	Watson Laboratories, Inc.	Peelable pouch for transdermal patch and method for packaging
EP1386604A1 (en) *	2002-07-30	2004-02-04	Schwarz Pharma Ag	Improved transdermal delivery system
ATE534373T1 (de)	2003-10-10	2011-12-15	Antares Pharma Ipl Ag	Transdermale pharmazeutische formulierung zur minimierung von rückständen auf der haut
US7425340B2 (en) *	2004-05-07	2008-09-16	Antares Pharma Ipl Ag	Permeation enhancing compositions for anticholinergic agents
US8067399B2 (en)	2005-05-27	2011-11-29	Antares Pharma Ipl Ag	Method and apparatus for transdermal or transmucosal application of testosterone
CN101426475A (zh) *	2006-04-21	2009-05-06	安塔雷斯制药Ipl股份公司	使用用于经皮或经粘膜应用的制剂治疗热潮红的方法
WO2008067991A2 (en) *	2006-12-08	2008-06-12	Antares Pharma Ipl Ag	Skin-friendly drug complexes for transdermal administration
US8415390B2 (en)	2008-05-30	2013-04-09	Microdose Therapeutx, Inc.	Methods and compositions for administration of oxybutynin
US9119777B2 (en)	2008-05-30	2015-09-01	Microdose Therapeutx, Inc.	Methods and compositions for administration of oxybutynin
BRPI0812000A2 (pt) *	2007-05-30	2014-11-18	Microdose Therapeutx Inc	Métodos e composições para administração de oxibutinina
JP5782635B2 (ja) *	2011-01-12	2015-09-24	有限会社センチュリーテック	搬送装置
JP7776442B2 (ja)	2020-05-05	2025-11-26	アプニメッド，インコーポレイテッド（デラウェア）	（ｒ）－オキシブチニン塩酸塩の多形形態
EP3909570A1 (de) *	2020-05-15	2021-11-17	Farco-Pharma GmbH	Oxybutynin für die intravesikale anwendung
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NL124473C (pt) *	1960-07-26
JPH0755904B2 (ja) *	1986-05-14	1995-06-14	小玉株式会社	膀胱疾患治療剤
MX9202350A (es) *	1991-05-20	1992-11-01	Alza Corp	Composiciones de incrementador de penetracion a la piel que usan monolinoleato de glicerol.
JP3688293B2 (ja) *	1993-09-29	2005-08-24	アルザ・コーポレーション	モノグリセリド／乳酸エステル透過促進剤
US5677346A (en) *	1995-01-31	1997-10-14	Sepracor, Inc.	Treating urinary incontinence using (S)-desethyloxybutynin
US5532278A (en) *	1995-01-31	1996-07-02	Sepracor, Inc.	Methods and compositions for treating urinary incontinence using optically pure (S)-oxybutynin

1996
- 1996-06-28 US US08/671,976 patent/US5736577A/en not_active Expired - Fee Related
1997
- 1997-06-27 JP JP10504448A patent/JP2000513724A/ja not_active Withdrawn
- 1997-06-27 EP EP97931531A patent/EP0914113A1/en not_active Withdrawn
- 1997-06-27 BR BR9710031A patent/BR9710031A/pt not_active IP Right Cessation
- 1997-06-27 PL PL97330752A patent/PL190483B1/pl not_active IP Right Cessation
- 1997-06-27 RU RU99101790/14A patent/RU2195276C2/ru not_active IP Right Cessation
- 1997-06-27 CZ CZ984283A patent/CZ428398A3/cs unknown
- 1997-06-27 SK SK1786-98A patent/SK178698A3/sk unknown
- 1997-06-27 UA UA99010429A patent/UA61916C2/uk unknown
- 1997-06-27 NZ NZ333282A patent/NZ333282A/en unknown
- 1997-06-27 CA CA002257121A patent/CA2257121C/en not_active Expired - Fee Related
- 1997-06-27 AU AU35137/97A patent/AU732568B2/en not_active Ceased
- 1997-06-27 WO PCT/US1997/011570 patent/WO1998000126A1/en not_active Ceased
1998
- 1998-12-16 NO NO985896A patent/NO985896D0/no unknown

Also Published As

Publication number	Publication date
NO985896L (no)	1998-12-16
UA61916C2 (en)	2003-12-15
BR9710031A (pt)	1999-08-10
NZ333282A (en)	2000-06-23
CA2257121A1 (en)	1998-01-08
PL330752A1 (en)	1999-05-24
AU732568B2 (en)	2001-04-26
CZ428398A3 (cs)	1999-06-16
US5736577A (en)	1998-04-07
CA2257121C (en)	2006-10-24
AU3513797A (en)	1998-01-21
NO985896D0 (no)	1998-12-16
WO1998000126A1 (en)	1998-01-08
JP2000513724A (ja)	2000-10-17
PL190483B1 (pl)	2005-12-30
EP0914113A1 (en)	1999-05-12
RU2195276C2 (ru)	2002-12-27

Publication	Publication Date	Title
SK178698A3 (en)	1999-09-10	Treating urinary incontinence using (s)-oxybutynin and (s)-desethyloxybutynin
KR100390271B1 (ko)	2003-10-04	(s)-옥시부티닌과(s)-데스에틸옥시부티닌을이용한요실금치료
US5532278A (en)	1996-07-02	Methods and compositions for treating urinary incontinence using optically pure (S)-oxybutynin
US6310103B1 (en)	2001-10-30	S(−)-tolterodine in the treatment of urinary and gastrointestinal disorders
US6123961A (en)	2000-09-26	Treating urinary incontinence with (R)-desethyloxybutynin and (R)-oxybutynin
EP1286591B1 (en)	2010-10-06	Treating smooth muscle hyperactivity with (r)-oxybutynin and (r)- desethyloxybutynin
US6432446B2 (en)	2002-08-13	Non-arrhythmogenic metabolite of oxybutynin
KR100476550B1 (ko)	2005-07-12	(s)-옥시부티닌과(s)-데스에틸옥시부티닌을이용한요실금치료
WO1998001125A2 (en)	1998-01-15	Dextrorotatory isomers of oxybutynin and desethyloxybutynin in the treatment of gastrointestinal hyperactivity
HK1113909A (en)	2008-10-17	Treating smooth muscle hyperactivity with (r)-oxybutynin and (r)-desethyloxybutynin