SV2017005441A - Antagonista de a2a de dosis baja para el tratamiento de tdah y la enfermedad de parkinson - Google Patents
Antagonista de a2a de dosis baja para el tratamiento de tdah y la enfermedad de parkinsonInfo
- Publication number
- SV2017005441A SV2017005441A SV2017005441A SV2017005441A SV2017005441A SV 2017005441 A SV2017005441 A SV 2017005441A SV 2017005441 A SV2017005441 A SV 2017005441A SV 2017005441 A SV2017005441 A SV 2017005441A SV 2017005441 A SV2017005441 A SV 2017005441A
- Authority
- SV
- El Salvador
- Prior art keywords
- parkinson
- antagonist
- disease
- low dose
- adhd treatment
- Prior art date
Links
- 208000018737 Parkinson disease Diseases 0.000 title abstract 2
- 239000005557 antagonist Substances 0.000 title abstract 2
- 208000006096 Attention Deficit Disorder with Hyperactivity Diseases 0.000 title 1
- 208000036864 Attention deficit/hyperactivity disease Diseases 0.000 title 1
- 230000006735 deficit Effects 0.000 abstract 1
- 229940126601 medicinal product Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4436—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Psychology (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
- Coloring Foods And Improving Nutritive Qualities (AREA)
Abstract
LA PRESENTE INVENCIÓN SE REFIERE A DOSIS ESPECÍFICAS DE UN ANTAGONISTA DE A2A PARA UTILIZARLO COMO UN MEDICAMENTO Y, EN PARTICULAR, QUE SEAN ÚTILES PARA EL TRATAMIENTO DE LA ENFERMEDAD DE PARKINSON Y DEL TRASTORNO POR DÉFICIT DE ATENCIÓN CON HIPERACTIVIDAD
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA201400704 | 2014-12-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SV2017005441A true SV2017005441A (es) | 2017-08-25 |
Family
ID=58731664
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SV2017005441A SV2017005441A (es) | 2014-12-03 | 2017-05-12 | Antagonista de a2a de dosis baja para el tratamiento de tdah y la enfermedad de parkinson |
Country Status (25)
| Country | Link |
|---|---|
| US (2) | US20160158211A1 (es) |
| EP (1) | EP3226863A1 (es) |
| JP (1) | JP2017536400A (es) |
| KR (1) | KR20170090430A (es) |
| CN (1) | CN106999480A (es) |
| AU (1) | AU2015357197A1 (es) |
| BR (1) | BR112017011777A2 (es) |
| CA (1) | CA2966582A1 (es) |
| CL (1) | CL2017001407A1 (es) |
| CO (1) | CO2017004785A2 (es) |
| CR (1) | CR20170221A (es) |
| DO (1) | DOP2017000121A (es) |
| EA (1) | EA201790973A1 (es) |
| EC (1) | ECSP17030050A (es) |
| IL (1) | IL252355A0 (es) |
| MA (1) | MA41090A (es) |
| MX (1) | MX2017007027A (es) |
| NI (1) | NI201700066A (es) |
| PE (1) | PE20170926A1 (es) |
| PH (1) | PH12017500923A1 (es) |
| SG (1) | SG11201704370XA (es) |
| SV (1) | SV2017005441A (es) |
| TN (1) | TN2017000174A1 (es) |
| TW (1) | TW201632186A (es) |
| WO (1) | WO2016087429A1 (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GEP20237548B (en) | 2018-07-05 | 2023-10-10 | Incyte Corp | Fused pyrazine derivatives as a2a /a2b inhibitors |
| US20200345725A1 (en) | 2019-01-11 | 2020-11-05 | Omeros Corporation | Methods and Compositions for Treating Cancer |
| TWI829857B (zh) | 2019-01-29 | 2024-01-21 | 美商英塞特公司 | 作為a2a / a2b抑制劑之吡唑并吡啶及三唑并吡啶 |
| CN114917350B (zh) * | 2022-06-21 | 2023-06-13 | 重庆医科大学附属第二医院 | Cftr增强剂在注意缺陷与多动障碍中的应用及产品 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2551611C (en) * | 2003-12-26 | 2013-06-25 | Kyowa Kirin Co., Ltd. | Thiazole derivatives for treating or preventing parkinson's disease |
| NZ590793A (en) * | 2008-07-23 | 2012-07-27 | Kyowa Hakko Kirin Co Ltd | Therapeutic agent for migraine |
| TWI548411B (zh) * | 2009-04-28 | 2016-09-11 | Kyowa Hakko Kirin Co Ltd | Exercise disorder treatment |
| UA110097C2 (uk) * | 2009-09-02 | 2015-11-25 | Терапевтичний агент для лікування розладів настрою | |
| UA113383C2 (xx) * | 2009-09-02 | 2017-01-25 | Терапевтичний агент для лікування тривожних розладів |
-
2015
- 2015-11-30 MA MA041090A patent/MA41090A/fr unknown
- 2015-12-01 TW TW104140137A patent/TW201632186A/zh unknown
- 2015-12-01 CA CA2966582A patent/CA2966582A1/en not_active Withdrawn
- 2015-12-01 BR BR112017011777A patent/BR112017011777A2/pt not_active Application Discontinuation
- 2015-12-01 CN CN201580064814.4A patent/CN106999480A/zh not_active Withdrawn
- 2015-12-01 CR CR20170221A patent/CR20170221A/es unknown
- 2015-12-01 JP JP2017529636A patent/JP2017536400A/ja not_active Withdrawn
- 2015-12-01 PE PE2017000864A patent/PE20170926A1/es not_active Application Discontinuation
- 2015-12-01 US US14/955,148 patent/US20160158211A1/en not_active Abandoned
- 2015-12-01 EP EP15802121.2A patent/EP3226863A1/en not_active Withdrawn
- 2015-12-01 KR KR1020177015211A patent/KR20170090430A/ko not_active Withdrawn
- 2015-12-01 EA EA201790973A patent/EA201790973A1/ru unknown
- 2015-12-01 TN TN2017000174A patent/TN2017000174A1/en unknown
- 2015-12-01 MX MX2017007027A patent/MX2017007027A/es unknown
- 2015-12-01 AU AU2015357197A patent/AU2015357197A1/en not_active Withdrawn
- 2015-12-01 SG SG11201704370XA patent/SG11201704370XA/en unknown
- 2015-12-01 WO PCT/EP2015/078181 patent/WO2016087429A1/en not_active Ceased
-
2017
- 2017-05-12 CO CONC2017/0004785A patent/CO2017004785A2/es unknown
- 2017-05-12 SV SV2017005441A patent/SV2017005441A/es unknown
- 2017-05-16 DO DO2017000121A patent/DOP2017000121A/es unknown
- 2017-05-16 EC ECIEPI201730050A patent/ECSP17030050A/es unknown
- 2017-05-17 IL IL252355A patent/IL252355A0/en unknown
- 2017-05-18 PH PH12017500923A patent/PH12017500923A1/en unknown
- 2017-06-01 NI NI201700066A patent/NI201700066A/es unknown
- 2017-06-02 CL CL2017001407A patent/CL2017001407A1/es unknown
- 2017-11-10 US US15/809,378 patent/US20180125835A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| PE20170926A1 (es) | 2017-07-13 |
| JP2017536400A (ja) | 2017-12-07 |
| CN106999480A (zh) | 2017-08-01 |
| TN2017000174A1 (en) | 2018-10-19 |
| CO2017004785A2 (es) | 2017-08-31 |
| TW201632186A (zh) | 2016-09-16 |
| MX2017007027A (es) | 2017-08-24 |
| MA41090A (fr) | 2017-10-10 |
| NI201700066A (es) | 2018-01-04 |
| US20160158211A1 (en) | 2016-06-09 |
| BR112017011777A2 (pt) | 2018-02-20 |
| EA201790973A1 (ru) | 2017-10-31 |
| DOP2017000121A (es) | 2017-07-15 |
| CR20170221A (es) | 2017-10-05 |
| US20180125835A1 (en) | 2018-05-10 |
| CL2017001407A1 (es) | 2018-01-05 |
| SG11201704370XA (en) | 2017-06-29 |
| KR20170090430A (ko) | 2017-08-07 |
| IL252355A0 (en) | 2017-07-31 |
| WO2016087429A1 (en) | 2016-06-09 |
| CA2966582A1 (en) | 2016-06-09 |
| ECSP17030050A (es) | 2017-08-31 |
| EP3226863A1 (en) | 2017-10-11 |
| PH12017500923A1 (en) | 2017-11-20 |
| AU2015357197A1 (en) | 2017-05-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CR20130377A (es) | Métodos y productos de fármaco para tratar enfermedad de alzheimer | |
| CR20160275A (es) | Derivados del sulphamoylpyrrolamide y uso como medicamento para el tratamiento de la hepatitis b | |
| BR112017009497A2 (pt) | polinucleotídeos de aadc para o tratamento da doença de parkinson | |
| SV2017005419A (es) | Triazolopirazinonas como inhibidores de pde1 | |
| DOP2015000241A (es) | Compuestos de biaril-amida como inhibidores de cinasa | |
| MX2016001587A (es) | Inhibidores de kdm1a para el tratamiento de enfermedades. | |
| DOP2017000049A (es) | Compuestos tricíclicos que contienen nitrógeno para el tratamiento de la infección por neisseria gonorrhoeae | |
| MX2019013808A (es) | Compuestos desestabilizadores de microtubulina para usarse en el tratamiento del cancer. | |
| DOP2016000170A (es) | Compuestos derivados de hidroxiformamida y usos del mismo | |
| SV2017005412A (es) | Compuestos de 1-alquil-6-oxo-1,6-dihidropiridin-3-ilo y usos de los mismos | |
| NI201600070A (es) | Inhibidores tetracíclicos de autotaxina | |
| MX2014011855A (es) | Sistemas y metodos para tratar una respuesta farmacodinamica adversa inducida por opioides. | |
| CL2016000019A1 (es) | Compuestos derivados de dihidroxifenilo deuterado o una sal de los mismos; composición farmacéutica que los comprende y su uso para el tratamiento de trastornos mediados por neurotransmisores tales como hipotensión, trastornos del sueño, enfermedad de alzheimer y depresión. | |
| CR20170090A (es) | Derivados de terahidroquinolina como inhibidores del bromodominio | |
| BR112016015997A2 (pt) | ?composições farmacêuticas que compreendem 15- hepe e métodos para tratar asma e distúrbios pulmonares com o uso das mesmas? | |
| SV2017005441A (es) | Antagonista de a2a de dosis baja para el tratamiento de tdah y la enfermedad de parkinson | |
| ECSP16086247A (es) | (s)-pirlindole y sus sales farmacéuticamente aceptables para uso en medicina | |
| MX2017001461A (es) | Terapia de combinacion. | |
| MX364528B (es) | Witanólidos útiles para el tratamiento de enfermedades neurodegenerativas. | |
| MX377995B (es) | Moléculas de unión al receptor bag3 para uso como un medicamento. | |
| BR112017016333A2 (pt) | compostos anticâncer | |
| ECSP16086232A (es) | (r) -pirlindole y sus sales farmacéuticamente aceptables para uso en medicina | |
| MX384637B (es) | Compuestos oxadiazoespíricos para el tratamiento del abuso y la adicción a las drogas. | |
| ECSP16094286A (es) | Compuestos, composición farmacéutica y su uso en el tratamiento de enfermedades neurodegenerativas | |
| GT201600190A (es) | Compuestos químicos |