TH129940A - Lactam group replaced with piperidinyl that acts as a modulator of GPR119 (PIPERIDINYL-SUBSTITUTED LACTAMS AS GPR119 MODULATORS). - Google Patents
Lactam group replaced with piperidinyl that acts as a modulator of GPR119 (PIPERIDINYL-SUBSTITUTED LACTAMS AS GPR119 MODULATORS).Info
- Publication number
- TH129940A TH129940A TH1201005976A TH1201005976A TH129940A TH 129940 A TH129940 A TH 129940A TH 1201005976 A TH1201005976 A TH 1201005976A TH 1201005976 A TH1201005976 A TH 1201005976A TH 129940 A TH129940 A TH 129940A
- Authority
- TH
- Thailand
- Prior art keywords
- piperidinyl
- gpr119
- modulator
- modulators
- acts
- Prior art date
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Abstract
DC60 (16/11/55) สารประกอบชนิดต่างๆ ที่มีสูตรโครงสร้างที่ (I) (สูตรเคมี) (I) และเกลือที่เป็นที่ยอมรับทางเภสัชกรรมชนิดต่างๆ ของสารประกอบดังกล่าว ซึ่ง X1, X2, L, R3, R4, R5, R6, R6a, R7, R9, R9a และ n มีความหมายตามที่ให้ไว้ในเอกสารสิทธิบัตร คือ มอ ดูเลเตอร์ของ GPR119 และมีประโยชน์ในการรักษาหรือป้องกันโรคต่างๆ เช่น แต่ไม่จำกัดเพียง โรคเบาหวานชนิดที่ 2 อาการของโรคเบาหวาน ภาวะแทรกซ้อนจากโรคเบาหวาน โรคอ้วนลงพุง โรคอ้วน ภาวะไขมันในเลือดสูง และภาวะอื่นๆ ที่เกี่ยวข้องDC60 (16/11/55) Various compounds having the structural formula (I) (chemical formula) (I) and various pharmaceutically accepted salts of such compounds, where X1, X2, L, R3, R4, R5, R6, R6a, R7, R9, R9a and n have the meanings given in the patent documents, namely modulators of GPR119 and are useful in treating or preventing diseases such as, but not limited to, type 2 diabetes, symptoms of diabetes, complications of diabetes, central obesity, obesity, hyperlipidemia and other related conditions.
Claims (1)
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TH129940A true TH129940A (en) | 2013-11-28 |
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