TH170428A - 6- (5-hydroxy-1h-pyrazol-1-il) derivatives, nicotine amide and their use as a PHD inhibitor. - Google Patents
6- (5-hydroxy-1h-pyrazol-1-il) derivatives, nicotine amide and their use as a PHD inhibitor.Info
- Publication number
- TH170428A TH170428A TH1501005718A TH1501005718A TH170428A TH 170428 A TH170428 A TH 170428A TH 1501005718 A TH1501005718 A TH 1501005718A TH 1501005718 A TH1501005718 A TH 1501005718A TH 170428 A TH170428 A TH 170428A
- Authority
- TH
- Thailand
- Prior art keywords
- compounds
- group
- pyrazol
- hydroxy
- derivatives
- Prior art date
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Abstract
การประดิษฐ์นี้ให้สารประกอบของสูตรโครงสร้างที่ (I) ซึ่งเป็นประโยชน์เป็นสารยับยั้ง PHD องค์ประกอบทางเภสัชกรรมของสารประกอบดังกล่าว วิธีการสำหรับการรักษาภาวะต่าง ๆ ที่ สัมพันธ์กับ HIF กระบวนการสำหรับการทำสารประกอบดังกล่าวและสารมัธยันตร์ของ สารประกอบดังกล่าวThe present invention provides compounds of structural formula (I) which are useful as PHD inhibitors, pharmaceutical compositions of said compounds, methods for treating various conditions associated with HIF, processes for making said compounds and intermediates of said compounds.
Claims (1)
Publications (2)
| Publication Number | Publication Date |
|---|---|
| TH170428A true TH170428A (en) | 2017-11-16 |
| TH1501005718A TH1501005718A (en) | 2017-11-16 |
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