TR199801713T2 - Yeni eritromisin t�revleri, bunlar�n haz�rlanmas�na y�nelik metodlar - Google Patents

Yeni eritromisin t�revleri, bunlar�n haz�rlanmas�na y�nelik metodlar

Info

Publication number: TR199801713T2
Authority: TR; Turkey
Prior art keywords: preparation; methods; erythromycin derivatives; new erythromycin; formula
Prior art date: 1996-02-28

Application number

TR1998/01713T

Other languages

English (en)

Turkish (tr)

Inventor

Agouridas Constantin

Chantot Jeon-Fran�Ois

Original Assignee

Hoechst Marion Roussel

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-02-28

Filing date

1997-02-27

Publication date

1998-12-21

1997-02-27 Application filed by Hoechst Marion Roussel filed Critical Hoechst Marion Roussel

1998-12-21 Publication of TR199801713T2 publication Critical patent/TR199801713T2/xx

Links

ULGZDMOVFRHVEP-RWJQBGPGSA-N Erythromycin Chemical class O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ULGZDMOVFRHVEP-RWJQBGPGSA-N 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 2
KXDHJXZQYSOELW-UHFFFAOYSA-N Carbamic acid Chemical group NC(O)=O KXDHJXZQYSOELW-UHFFFAOYSA-N 0.000 abstract 1
-1 SO2 radical Chemical class 0.000 abstract 1
150000005840 aryl radicals Chemical group 0.000 abstract 1
230000003115 biocidal effect Effects 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
125000004430 oxygen atom Chemical group O* 0.000 abstract 1
150000003254 radicals Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Molecular Biology (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Oncology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Communicable Diseases (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)

TR1998/01713T 1996-02-28 1997-02-27 Yeni eritromisin t�revleri, bunlar�n haz�rlanmas�na y�nelik metodlar TR199801713T2 (xx)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR9602472A FR2745290B1 (fr)	1996-02-28	1996-02-28	Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number	Publication Date
TR199801713T2 true TR199801713T2 (xx)	1998-12-21

Family

ID=9489659

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
TR1998/01713T TR199801713T2 (xx)	1996-02-28	1997-02-27	Yeni eritromisin t�revleri, bunlar�n haz�rlanmas�na y�nelik metodlar

Country Status (31)

Country	Link
US (1)	US6096714A (2)
EP (1)	EP0885234B1 (2)
JP (1)	JP4102440B2 (2)
KR (1)	KR100486053B1 (2)
CN (1)	CN1168734C (2)
AP (1)	AP952A (2)
AR (1)	AR005999A1 (2)
AT (1)	ATE217633T1 (2)
AU (1)	AU716204B2 (2)
BG (1)	BG63207B1 (2)
BR (1)	BR9707709B1 (2)
CZ (1)	CZ293893B6 (2)
DE (1)	DE69712610T2 (2)
DK (1)	DK0885234T3 (2)
EA (1)	EA001376B1 (2)
EE (1)	EE9800265A (2)
ES (1)	ES2176698T3 (2)
FR (1)	FR2745290B1 (2)
HU (1)	HU227567B1 (2)
IL (1)	IL125622A (2)
NO (1)	NO983955L (2)
NZ (1)	NZ331600A (2)
OA (1)	OA10845A (2)
PL (1)	PL191736B1 (2)
PT (1)	PT885234E (2)
SK (1)	SK118498A3 (2)
TR (1)	TR199801713T2 (2)
UA (1)	UA58504C2 (2)
WO (1)	WO1997031929A1 (2)
YU (1)	YU37098A (2)
ZA (1)	ZA971659B (2)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA989835B (en) *	1997-10-29	1999-05-05	Taisho Pharmaceutical Co Ltd	Erythromycin a derivatives
WO1999021870A1 (en) *	1997-10-29	1999-05-06	Taisho Pharmaceutical Co., Ltd.	Erythromycin a 11, 12-carbamate derivatives
JP4573925B2 (ja) *	1998-07-09	2010-11-04	アベンティス・ファーマ・ソシエテ・アノニム	新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用
FR2792637B1 (fr) *	1999-04-26	2001-06-01	Hoechst Marion Roussel Inc	Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2780977B1 (fr) *	1998-07-09	2000-09-01	Hoechst Marion Roussel Inc	Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2781484B1 (fr) *	1998-07-21	2001-08-10	Hoechst Marion Roussel Inc	Nouveaux derives de la 6-deoxy erythromycine, leur procede de preparation et leur application comme medicaments
CA2359708C (en)	1999-01-27	2005-10-25	Pfizer Products Inc.	Ketolide antibiotics
EA200100983A1 (ru) *	1999-05-24	2002-10-31	Пфайзер Продактс Инк.	Производные 13-метилэритромицина
WO2001010880A1 (fr) *	1999-08-06	2001-02-15	Taisho Pharmaceutical Co., Ltd.	Derives d'erythromycine a
WO2001010879A1 (fr) *	1999-08-06	2001-02-15	Taisho Pharmaceutical Co., Ltd.	Derives d'erythromycine a
WO2001010878A1 (fr) *	1999-08-06	2001-02-15	Taisho Pharmaceutical Co., Ltd.	Derives d'erythromycine a
EP1146051A3 (en) *	2000-04-10	2001-10-31	Pfizer Products Inc.	Erythromycin A derivatives
US20020115621A1 (en) *	2000-08-07	2002-08-22	Wei-Gu Su	Macrolide antibiotics
ITMI20021726A1 (it) *	2002-08-01	2004-02-02	Zambon Spa	Macrolidi ad attivita' antiinfiammatoria.
ES2552682T3 (es)	2003-03-10	2015-12-01	Merck Sharp & Dohme Corp.	Agentes antibacterianos novedosos
WO2005007143A2 (en) *	2003-07-14	2005-01-27	The Board Of Trustees Of The University Of Illinois	Use of makrolides and ketolides for the treatment of tuberculosis
WO2007069264A2 (en) *	2005-12-15	2007-06-21	Alembic Limited	Reference standards for determining the purity of telithromycin and processes therefor
CN105732745A (zh)	2007-10-25	2016-07-06	森普拉制药公司	大环内酯类抗菌剂的制备方法
AU2009308182B2 (en) *	2008-10-24	2016-05-19	Cempra Pharmaceuticals, Inc.	Biodefenses using triazole-containing macrolides
US9937194B1 (en)	2009-06-12	2018-04-10	Cempra Pharmaceuticals, Inc.	Compounds and methods for treating inflammatory diseases
US9480679B2 (en)	2009-09-10	2016-11-01	Cempra Pharmaceuticals, Inc.	Methods for treating malaria, tuberculosis and MAC diseases
DK2550286T3 (en)	2010-03-22	2016-02-29	Cempra Pharmaceuticals Inc	CRYSTALLINE FORMS OF A MACROLID AND APPLICATIONS THEREOF
CN105198944B (zh)	2010-05-20	2018-06-01	森普拉制药公司	制备大环内酯和酮内酯及其中间体的方法
EP2613630A4 (en)	2010-09-10	2014-01-15	Cempra Pharmaceuticals Inc	HYDROGEN BOND FOR THE PREPARATION OF FLUOROCHETOLIDES FOR THE TREATMENT OF DISEASES
MX2014011537A (es)	2012-03-27	2015-02-10	Cempra Pharmaceuticals Inc	Formulaciones parenterales para la administracion de antibioticos macrolidos.
HK1217665A1 (zh)	2013-03-14	2017-01-20	森普拉制药公司	用於治療呼吸道疾病的方法及其製劑
RU2015138797A (ru)	2013-03-15	2017-04-24	Семпра Фармасьютикалс, Инк.	Конвергентные способы получения макролидных антибактериальных агентов

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US487411A (en) *		1892-12-06		Island
IL114589A (en) *	1990-11-21	1999-12-22	Roussel Uclaf	Intermediates for the preparation of erythromycin derivatives
US5444031A (en) *	1993-01-21	1995-08-22	Calgon Carbon Corporation	Process for making catalytic carbon
FR2727969B1 (fr) *	1994-12-09	1997-01-17	Roussel Uclaf	Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

1996
- 1996-02-28 FR FR9602472A patent/FR2745290B1/fr not_active Expired - Lifetime
1997
- 1997-02-25 AR ARP970100760A patent/AR005999A1/es unknown
- 1997-02-26 ZA ZA9701659A patent/ZA971659B/xx unknown
- 1997-02-27 EE EE9800265A patent/EE9800265A/xx unknown
- 1997-02-27 IL IL12562297A patent/IL125622A/xx not_active IP Right Cessation
- 1997-02-27 PT PT97907141T patent/PT885234E/pt unknown
- 1997-02-27 EP EP97907141A patent/EP0885234B1/fr not_active Expired - Lifetime
- 1997-02-27 KR KR10-1998-0706733A patent/KR100486053B1/ko not_active Expired - Lifetime
- 1997-02-27 EA EA199800768A patent/EA001376B1/ru not_active IP Right Cessation
- 1997-02-27 ES ES97907141T patent/ES2176698T3/es not_active Expired - Lifetime
- 1997-02-27 AT AT97907141T patent/ATE217633T1/de active
- 1997-02-27 DE DE69712610T patent/DE69712610T2/de not_active Expired - Lifetime
- 1997-02-27 US US09/125,959 patent/US6096714A/en not_active Ceased
- 1997-02-27 AP APAP/P/1998/001318A patent/AP952A/en active
- 1997-02-27 CN CNB971926255A patent/CN1168734C/zh not_active Expired - Lifetime
- 1997-02-27 BR BRPI9707709-7A patent/BR9707709B1/pt not_active IP Right Cessation
- 1997-02-27 DK DK97907141T patent/DK0885234T3/da active
- 1997-02-27 WO PCT/FR1997/000351 patent/WO1997031929A1/fr not_active Ceased
- 1997-02-27 PL PL328608A patent/PL191736B1/pl unknown
- 1997-02-27 HU HU9902576A patent/HU227567B1/hu unknown
- 1997-02-27 SK SK1184-98A patent/SK118498A3/sk unknown
- 1997-02-27 UA UA98095031A patent/UA58504C2/uk unknown
- 1997-02-27 TR TR1998/01713T patent/TR199801713T2/xx unknown
- 1997-02-27 JP JP53067197A patent/JP4102440B2/ja not_active Expired - Lifetime
- 1997-02-27 CZ CZ19982587A patent/CZ293893B6/cs not_active IP Right Cessation
- 1997-02-27 NZ NZ331600A patent/NZ331600A/xx unknown
- 1997-02-27 AU AU19298/97A patent/AU716204B2/en not_active Expired
1998
- 1998-08-12 BG BG102691A patent/BG63207B1/bg unknown
- 1998-08-27 NO NO983955A patent/NO983955L/no not_active Application Discontinuation
- 1998-08-28 OA OA9800150A patent/OA10845A/fr unknown
- 1998-08-28 YU YU37098A patent/YU37098A/sh unknown

Also Published As

Publication number	Publication date
CZ258798A3 (cs)	1998-12-16
FR2745290B1 (fr)	1998-04-03
ATE217633T1 (de)	2002-06-15
AP9801318A0 (en)	1998-09-30
DK0885234T3 (da)	2002-08-26
ES2176698T3 (es)	2002-12-01
NO983955D0 (no)	1998-08-27
KR19990087324A (ko)	1999-12-27
JP2000505469A (ja)	2000-05-09
AU1929897A (en)	1997-09-16
NO983955L (no)	1998-08-27
AU716204B2 (en)	2000-02-24
US6096714A (en)	2000-08-01
BG63207B1 (bg)	2001-06-29
WO1997031929A1 (fr)	1997-09-04
HUP9902576A1 (hu)	1999-12-28
IL125622A (en)	2003-10-31
BG102691A (en)	1999-06-30
DE69712610T2 (de)	2002-11-28
PL191736B1 (pl)	2006-06-30
HUP9902576A3 (en)	2001-03-28
PL328608A1 (en)	1999-02-01
CN1168734C (zh)	2004-09-29
AR005999A1 (es)	1999-07-21
KR100486053B1 (ko)	2005-06-16
JP4102440B2 (ja)	2008-06-18
EP0885234B1 (fr)	2002-05-15
FR2745290A1 (fr)	1997-08-29
EE9800265A (et)	1999-02-15
CN1212700A (zh)	1999-03-31
HU227567B1 (en)	2011-08-29
DE69712610D1 (de)	2002-06-20
EA199800768A1 (ru)	1999-02-25
SK118498A3 (en)	1999-07-12
UA58504C2 (uk)	2003-08-15
BR9707709A (pt)	1999-04-06
YU37098A (sh)	1999-07-28
BR9707709B1 (pt)	2014-10-14
NZ331600A (en)	1999-08-30
ZA971659B (en)	1998-02-26
AP952A (en)	2001-03-29
CZ293893B6 (cs)	2004-08-18
OA10845A (fr)	2003-02-05
PT885234E (pt)	2002-10-31
EP0885234A1 (fr)	1998-12-23
IL125622A0 (en)	1999-04-11
EA001376B1 (ru)	2001-02-26

Publication	Publication Date	Title
TR199801713T2 (xx)	1998-12-21	Yeni eritromisin t�revleri, bunlar�n haz�rlanmas�na y�nelik metodlar
AU5047793A (en)	1994-05-19	New derivatives of erythromycin, their preparation process, their use as medicaments
MY106250A (en)	1995-04-29	Azolylmethylcyclopentane benzylidene fungicide.
IL73893A0 (en)	1985-03-31	11-beta arylestradienes,their production,and pharmaceutical preparations containing same
IE883430L (en)	1989-05-17	Novel fluorocytidine derivatives
ATE32077T1 (de)	1988-02-15	7-amino-azolo(1,5-a>-pyrimidine und diese enthaltende fungizide.
AU4387296A (en)	1996-07-19	Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens
ZA875059B (en)	1988-02-24	Solutions of oxazaphosphorins having improved stability and process for the preparation thereof
IE892794L (en)	1990-03-01	Disubstituted benzylamines, their preparation process, their¹use as medicine and their synthesising agents
YU120991A (sh)	1994-01-20	Postupak za dobivanje cikličnih sulfata
AU2321688A (en)	1989-04-18	Compositions comprising 1-oxo- or thiohydrocarbyl substituted azacycloalkanes
TR200001222T2 (tr)	2000-09-21	Yeni tetrasiklikler, bunların üretimi için işlem ve bu birleşikleri içeren farmasötik preparasyonlar.
EP0974598A3 (fr)	2003-12-17	Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments
TR200000942T2 (tr)	2000-09-21	8-Azabisayklo(3.2.1) oktan-3-metanamin türevleri, hazırlanmaları ve terapötik uygulamaları.
SE8602854D0 (sv)	1986-06-26	New saccharides, their preparation and pharmaceutical compositions containing them
ES8705853A1 (es)	1987-05-16	Un procedimiento para la produccion de derivados de benzoilurea
JPS6431752A (en)	1989-02-02	Amide derivative and skin external preparation containing said derivative
MY104777A (en)	1994-05-31	Benzoxazine dyes
TR199900095T2 (xx)	1999-03-22	Yeni eritromisin t�revleri, haz�rlama metodu, ila� olarak kullan�m�.
MY100938A (en)	1991-05-31	Arylkylimidazole derivatives.
AU5759598A (en)	1998-07-31	Organosilicon compounds containing urea groups, their preparation and their use
TR200100178T2 (tr)	2002-10-21	Yeni 6-deoksi eritromisin türevleri, bunların hazırlanmasına yönelik metod
TR199801839T2 (2)	1998-12-21
TW334463B (en)	1998-06-21	4-methyl-1-pentene polymer compositions the polymer compositions have high permeability to gas and have improved flexibility and mechanical properties
ES481741A1 (es)	1980-02-16	Procedimiento para la obtencion de o-(amino alquil) oximas diaromaticas.