TR200000529T2 - İçinde eksipiyan olmayan granüller - Google Patents

İçinde eksipiyan olmayan granüller

Info

Publication number
TR200000529T2
TR200000529T2 TR2000/00529T TR200000529T TR200000529T2 TR 200000529 T2 TR200000529 T2 TR 200000529T2 TR 2000/00529 T TR2000/00529 T TR 2000/00529T TR 200000529 T TR200000529 T TR 200000529T TR 200000529 T2 TR200000529 T2 TR 200000529T2
Authority
TR
Turkey
Prior art keywords
granules
excipients
prepare
kinds
same time
Prior art date
Application number
TR2000/00529T
Other languages
English (en)
Inventor
Willem Groenendaal Jan
Original Assignee
Dsm N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dsm N.V. filed Critical Dsm N.V.
Publication of TR200000529T2 publication Critical patent/TR200000529T2/tr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682Processes
    • A61K9/1688Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient

Landscapes

  • Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Içinde eksipiyan olmayan, her türlü farmakolojik formülasyonlara uygun granüller elde edilmistir. Ayni zamanda sözü edilen granülleri tercihen hava jet sistemi olan bir eleme aygiti kullanilarak hazirlamak için bir islem elde edilmistir.
TR2000/00529T 1997-08-29 1998-08-27 İçinde eksipiyan olmayan granüller TR200000529T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP97202651 1997-08-29

Publications (1)

Publication Number Publication Date
TR200000529T2 true TR200000529T2 (tr) 2000-08-21

Family

ID=8228682

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2000/00529T TR200000529T2 (tr) 1997-08-29 1998-08-27 İçinde eksipiyan olmayan granüller

Country Status (5)

Country Link
EP (1) EP1023065A1 (tr)
CN (1) CN1268888A (tr)
AU (1) AU9540898A (tr)
TR (1) TR200000529T2 (tr)
WO (1) WO1999011261A1 (tr)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA01009808A (es) 1999-04-01 2002-04-24 Dsm Nv Aglomerados por cristalizacion.
WO2001043766A1 (fr) * 1999-12-14 2001-06-21 Asahi Kasei Kabushiki Kaisha Granules de sulfate de colistine
AT412344B (de) * 2001-04-12 2005-01-25 Sandoz Ag Hydrophobisierte teilchen von k-clavulanat
AT413983B (de) * 2001-04-12 2006-08-15 Sandoz Ag K-clavulanat in der form eines granulates
AT500131A1 (de) * 2002-02-01 2005-11-15 Sandoz Ag Organische verbindungen
AT500134A1 (de) * 2002-02-01 2005-11-15 Sandoz Ag Verfahren zur herstellung eines entmischungsstabilen granulats
AU2003208358A1 (en) * 2002-02-01 2003-09-02 Sandoz Gmbh Demixing-stable granulate
AT500132A1 (de) * 2002-02-06 2005-11-15 Sandoz Ag Organische verbindungen
AT500133A1 (de) * 2002-02-06 2005-11-15 Sandoz Ag Verfahren zur herstellung eines entmischungsstabilen granulats
US7534781B2 (en) 2003-03-21 2009-05-19 Dsm Ip Assets B.V. Crystalline amoxicillin trihydrate powder
US20060172987A1 (en) * 2003-03-21 2006-08-03 Dsm Ip Assets B.V. Amoxicillin trihydrate
WO2006003152A1 (en) * 2004-06-30 2006-01-12 Dsm Ip Assets B.V. GRANULES COMPRISING A ß-LACTAM ANTIBIOTIC
DE602006014531D1 (de) 2005-03-03 2010-07-08 Janssen Pharmaceutica Nv Substituierte oxadiazaspiro-ä5.5ü-undecanonderivate und ihre verwendung als neurokininantagonisten
NZ556628A (en) 2005-03-08 2009-09-25 Janssen Pharmaceutica Nv Diaza-spiro-[4.4]-nonane derivatives as neurokinin (NK1) antagonists
FI20080352A0 (fi) * 2008-05-09 2008-05-09 Atacama Labs Oy Prosessi korkean lääkepitoisuuden tabletin valmistamiseksi
FI20060990A0 (fi) * 2006-11-10 2006-11-10 Iprbox Oy Rakeita, tabletteja ja rakeistusmenetelmä
FI20080351A0 (fi) * 2008-05-09 2008-05-09 Atacama Labs Oy Prosessi matalan lääkepitoisuuden tabletin valmistamiseksi
FI20080348A0 (fi) * 2008-02-15 2008-05-09 Atacama Labs Oy Uudenlainen farmaseuttinen formulaatio
FI20080355A0 (fi) * 2008-05-09 2008-05-09 Atacama Labs Oy Prosessi metforminia käsittävien tablettien valmistamiseksi
FI20080353A0 (fi) * 2008-05-09 2008-05-09 Atacama Labs Oy Prosessi erittäin korkean lääkepitoisuuden tabletin valmistamiseksi
FI20070521A7 (fi) 2006-11-10 2008-05-11 Atacama Labs Oy Rakeita, tabletteja ja rakeistusmenetelmä
US8951562B2 (en) * 2006-11-10 2015-02-10 Atacama Labs Oy Method and apparatus or dry granulation
FI20080346A0 (fi) * 2008-05-09 2008-05-09 Atacama Labs Oy Prosessi lisäaineita sisältävän tabletin valmistamiseksi
WO2008089920A1 (en) 2007-01-26 2008-07-31 Dsm Ip Assets B.V. Process for the manufacture of substituted 2-cyano cinnamic esters
PT2271348T (pt) 2008-03-28 2018-04-16 Paratek Pharm Innc Formulação de comprimido oral de composto de tetraciclina
WO2009135946A1 (en) 2008-05-09 2009-11-12 Atacama Labs Oy Method and apparatus for dry granulation
IT1394597B1 (it) 2008-11-05 2012-07-05 Politi Granulazione a secco in flusso di gas.
US20150238425A1 (en) * 2012-08-28 2015-08-27 Dsm Sinochem Pharmaceuticals Netherlands B.V. Mini-tablets
BE1021312B1 (nl) * 2014-07-30 2015-10-28 Nordic Specialty Pharma Bvba Dicloxacillin capsule
CN105832694A (zh) * 2016-03-25 2016-08-10 海南汤臣史克生物科技有限公司 一种青霉素类药物胶囊及其制法
CN106088893B (zh) * 2016-07-28 2017-11-28 谭芳 隐藏式闭门器
EP4025353B1 (en) 2019-09-06 2024-11-06 Novo Nordisk A/S Method and equipment for fractionation of granules for use in pharmaceutical compositions

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2251250C3 (de) * 1972-10-19 1981-06-25 Hoechst Ag, 6230 Frankfurt Verfahren zur Herstellung hochdosierter Antibiotica-Tabletten
JPS6238A (ja) * 1985-03-12 1987-01-06 Sankyo Co Ltd 混合ビタミン凍結乾燥製剤の製法
DE3887179T2 (de) * 1987-03-02 1994-06-16 Brocades Pharma Bv Pharmazeutische Zusammensetzung, pharmazeutisches Granulat und Verfahren zu ihrer Herstellung.
DE3927810A1 (de) * 1989-08-23 1991-02-28 Basf Ag Riboflavingranulate
GB9009473D0 (en) * 1990-04-27 1990-06-20 Beecham Group Plc Pharmaceutical formulation
GB9109862D0 (en) * 1991-05-08 1991-07-03 Beecham Lab Sa Pharmaceutical formulations
GB9408117D0 (en) * 1994-04-23 1994-06-15 Smithkline Beecham Corp Pharmaceutical formulations
TWI225402B (en) * 1996-03-13 2004-12-21 Biochemie Gmbh Auxiliary-free agglomerates

Also Published As

Publication number Publication date
CN1268888A (zh) 2000-10-04
EP1023065A1 (en) 2000-08-02
WO1999011261A1 (en) 1999-03-11
AU9540898A (en) 1999-03-22

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