TR200101434T2 - Organofosfor terkipler ve kullanımları - Google Patents

Organofosfor terkipler ve kullanımları

Info

Publication number
TR200101434T2
TR200101434T2 TR2001/01434T TR200101434T TR200101434T2 TR 200101434 T2 TR200101434 T2 TR 200101434T2 TR 2001/01434 T TR2001/01434 T TR 2001/01434T TR 200101434 T TR200101434 T TR 200101434T TR 200101434 T2 TR200101434 T2 TR 200101434T2
Authority
TR
Turkey
Prior art keywords
formula
compositions
group
cycloalkyl
carbon atoms
Prior art date
Application number
TR2001/01434T
Other languages
English (en)
Inventor
Jomaa Hassan
Original Assignee
Jomaa Pharmaka Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jomaa Pharmaka Gmbh filed Critical Jomaa Pharmaka Gmbh
Publication of TR200101434T2 publication Critical patent/TR200101434T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06—Antimalarials
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3808—Acyclic saturated acids which can have further substituents on alkyl
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576—Six-membered rings
    • C07F9/58—Pyridine rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Bu bulus (I) formül organofosfor terkiplere iliskindir; bu formülde A (II) genel formülüne karsilik gelir; (II) formülünde C3, C4, C5 grubundan seçilen bir veya birden fazla karbon atomu ile ilgili yer degistirenleri yok sayabilir ve B1 ila B10'dan en az bir yer degistiren C3-8 sikloalkil (C0-9) alkil grubudur; burada hem C3-8 sikloalkil grubu hem C0-9 alkil grubu bir veya birden fazla çift bagi haiz olabilir ve sikloalkil grubun bir veya iki karbon atomu azot, oksijen veya sülfür atomlariyla yer degistirebilir. Bulus ayrica sözü geçen terkipleri içeren farmasötik preparatlara ve bunlarin insan ve hayvanlardaki enfeksiyonlu süreçlerin terapisi ve profilaksisinde kullanimina iliskindir.
TR2001/01434T 1998-11-25 1999-11-20 Organofosfor terkipler ve kullanımları TR200101434T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19854403A DE19854403A1 (de) 1998-11-25 1998-11-25 Phosphororganische Verbindungen und ihre Verwendung

Publications (1)

Publication Number Publication Date
TR200101434T2 true TR200101434T2 (tr) 2001-10-22

Family

ID=7888998

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2001/01434T TR200101434T2 (tr) 1998-11-25 1999-11-20 Organofosfor terkipler ve kullanımları

Country Status (22)

Country Link
US (1) US6534489B1 (tr)
EP (1) EP1133500B1 (tr)
JP (1) JP2002530412A (tr)
KR (1) KR20010093112A (tr)
CN (1) CN1328563A (tr)
AP (1) AP2001002150A0 (tr)
AT (1) ATE223921T1 (tr)
AU (1) AU754378B2 (tr)
BR (1) BR9915671A (tr)
CA (1) CA2352317A1 (tr)
CZ (1) CZ20011820A3 (tr)
DE (2) DE19854403A1 (tr)
EA (1) EA200100584A1 (tr)
HK (1) HK1042304B (tr)
IL (1) IL142777A0 (tr)
NO (1) NO20012542L (tr)
OA (1) OA11803A (tr)
PL (1) PL348871A1 (tr)
SK (1) SK7102001A3 (tr)
TR (1) TR200101434T2 (tr)
WO (1) WO2000031085A1 (tr)
ZA (1) ZA200103670B (tr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1297352A (zh) * 1998-04-14 2001-05-30 哈桑·朱马 有机磷化合物在治疗和预防性治疗感染中的应用
WO2001093872A1 (de) * 2000-06-08 2001-12-13 Jomaa Pharmaka Gmbh Verwendung von phosphororganischen hydroxamsäurederivaten zur herstellung von arzneimitteln
WO2001094358A1 (de) * 2000-06-08 2001-12-13 Jomaa Pharmaka Gmbh Phosphororganische hydroamsäurederivate als herbizide
WO2002078714A1 (de) * 2001-03-30 2002-10-10 Jomaa Pharmaka Gmbh Magensaftresistente formulierungen zur applikation von antiinfektiös wirkenden verbindungen, die den 2-c-methylerythrose-4-stoffwechselweg hemmen, sowie ihren salzen und estern
DE10356410A1 (de) * 2003-11-24 2005-06-23 Bioagency Ag Phosphororganische Verbindungen und deren Verwendung
EP3967312A1 (en) 2014-09-12 2022-03-16 UNION therapeutics A/S Antibacterial use of halogenated salicylanilides
GB201509326D0 (en) 2015-05-29 2015-07-15 Antibio Tx Aps Novel use
CN107722035B (zh) * 2017-11-03 2020-03-10 宁夏大学 一类青蒿素-哌嗪衍生物及其制法和在制备抗肝癌药物中的应用
US11419834B2 (en) 2019-02-25 2022-08-23 Rhode Island Hospital Methods for treating diseases or infections caused by or associated with H. pylori using a halogenated salicylanilide
CN112426531B (zh) * 2020-12-04 2023-04-07 深圳市中医院 一种药物组合物在制备治疗肾脏疾病药物中的用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1580899A (en) * 1976-07-27 1980-12-10 Fujisawa Pharmaceutical Co Hydroxyaminohydrocarbonphosphonic acid derivatives and production and use thereof
US4206156A (en) * 1976-07-27 1980-06-03 Fujisawa Pharmaceutical Company, Limited Hydroxyaminohydrocarbonphosphonic acids
US4268503A (en) 1978-09-14 1981-05-19 Fujisawa Pharmaceutical Co., Ltd. Antibacterial composition
US4693742A (en) * 1983-12-20 1987-09-15 Rohm And Hass Company Herbicidal hydroxyamino phosphonic acids and derivatives
JPS61106504A (ja) 1984-10-30 1986-05-24 Teijin Ltd 除草剤
CN1297352A (zh) 1998-04-14 2001-05-30 哈桑·朱马 有机磷化合物在治疗和预防性治疗感染中的应用

Also Published As

Publication number Publication date
BR9915671A (pt) 2001-08-14
CZ20011820A3 (cs) 2001-08-15
EP1133500A1 (de) 2001-09-19
KR20010093112A (ko) 2001-10-27
HK1042304A1 (en) 2002-08-09
CN1328563A (zh) 2001-12-26
DE19854403A1 (de) 2000-05-31
JP2002530412A (ja) 2002-09-17
AU754378B2 (en) 2002-11-14
NO20012542D0 (no) 2001-05-23
OA11803A (en) 2005-08-10
ATE223921T1 (de) 2002-09-15
AP2001002150A0 (en) 2001-06-30
CA2352317A1 (en) 2000-06-02
EA200100584A1 (ru) 2001-12-24
EP1133500B1 (de) 2002-09-11
NO20012542L (no) 2001-07-24
AU1652300A (en) 2000-06-13
DE59902692D1 (de) 2002-10-17
HK1042304B (zh) 2003-07-04
WO2000031085A1 (de) 2000-06-02
PL348871A1 (en) 2002-06-17
IL142777A0 (en) 2002-03-10
ZA200103670B (en) 2002-05-07
SK7102001A3 (en) 2001-12-03
US6534489B1 (en) 2003-03-18

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