TR200607613A2 - Lipaz inhibitörü içeren farmasötik formülasyonlar - Google Patents
Lipaz inhibitörü içeren farmasötik formülasyonlarInfo
- Publication number
- TR200607613A2 TR200607613A2 TR2006/07613A TR200607613A TR200607613A2 TR 200607613 A2 TR200607613 A2 TR 200607613A2 TR 2006/07613 A TR2006/07613 A TR 2006/07613A TR 200607613 A TR200607613 A TR 200607613A TR 200607613 A2 TR200607613 A2 TR 200607613A2
- Authority
- TR
- Turkey
- Prior art keywords
- pharmaceutical formulations
- formulations containing
- lipase inhibitors
- containing lipase
- orlistat
- Prior art date
Links
- 229940127470 Lipase Inhibitors Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 102100031416 Gastric triacylglycerol lipase Human genes 0.000 abstract 1
- 208000008589 Obesity Diseases 0.000 abstract 1
- 108050006759 Pancreatic lipases Proteins 0.000 abstract 1
- 102000019280 Pancreatic lipases Human genes 0.000 abstract 1
- 238000009472 formulation Methods 0.000 abstract 1
- 230000002496 gastric effect Effects 0.000 abstract 1
- 108010091264 gastric triacylglycerol lipase Proteins 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 235000020824 obesity Nutrition 0.000 abstract 1
- AHLBNYSZXLDEJQ-FWEHEUNISA-N orlistat Chemical compound CCCCCCCCCCC[C@H](OC(=O)[C@H](CC(C)C)NC=O)C[C@@H]1OC(=O)[C@H]1CCCCCC AHLBNYSZXLDEJQ-FWEHEUNISA-N 0.000 abstract 1
- 229960001243 orlistat Drugs 0.000 abstract 1
- 229940116369 pancreatic lipase Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1682—Processes
- A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Child & Adolescent Psychology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Bu buluş obesite tedavisinde kullanılan mide ve pankreas lipaz inhibitörü etkinliğine sahip orlistat'ı içeren oral yolla alınmaya uygun bir farmasötik dozaj formülasyonunu tarif etmektedir.
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2006/07613A TR200607613A2 (tr) | 2006-12-29 | 2006-12-29 | Lipaz inhibitörü içeren farmasötik formülasyonlar |
| PCT/TR2007/000152 WO2008082373A2 (en) | 2006-12-29 | 2007-12-28 | Pharmaceutical formulations comprising lipase inhibitor |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2006/07613A TR200607613A2 (tr) | 2006-12-29 | 2006-12-29 | Lipaz inhibitörü içeren farmasötik formülasyonlar |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR200607613A2 true TR200607613A2 (tr) | 2008-07-21 |
Family
ID=39589103
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2006/07613A TR200607613A2 (tr) | 2006-12-29 | 2006-12-29 | Lipaz inhibitörü içeren farmasötik formülasyonlar |
Country Status (2)
| Country | Link |
|---|---|
| TR (1) | TR200607613A2 (tr) |
| WO (1) | WO2008082373A2 (tr) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0901602B8 (pt) * | 2009-04-03 | 2021-05-25 | Ems S/A | formulação farmacêuticas |
| MX342962B (es) * | 2009-09-18 | 2016-06-07 | Teva Pharmaceuticals Holdings Mexico S A De C V | Composicion farmaceutica para bajar de peso y procedimiento para obtener la misma. |
| CN114767634A (zh) * | 2022-03-14 | 2022-07-22 | 大邦(湖南)生物制药有限公司 | 一种奥利司他微丸及其制备方法、奥利司他胶囊 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6004996A (en) * | 1997-02-05 | 1999-12-21 | Hoffman-La Roche Inc. | Tetrahydrolipstatin containing compositions |
| WO2000009123A1 (en) * | 1998-08-14 | 2000-02-24 | F. Hoffmann-La Roche Ag | Pharmaceutical compositions containing lipase inhibitors and chitosan |
| AR025587A1 (es) * | 1999-09-13 | 2002-12-04 | Hoffmann La Roche | Formulaciones en dispersion que contienen inhibidores de lipasa |
-
2006
- 2006-12-29 TR TR2006/07613A patent/TR200607613A2/tr unknown
-
2007
- 2007-12-28 WO PCT/TR2007/000152 patent/WO2008082373A2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2008082373A2 (en) | 2008-07-10 |
| WO2008082373A3 (en) | 2008-12-18 |
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