TR200907227A2 - Çözünürlüğü yüksek stabil mikronize granüller. - Google Patents
Çözünürlüğü yüksek stabil mikronize granüller.Info
- Publication number
- TR200907227A2 TR200907227A2 TR2009/07227A TR200907227A TR200907227A2 TR 200907227 A2 TR200907227 A2 TR 200907227A2 TR 2009/07227 A TR2009/07227 A TR 2009/07227A TR 200907227 A TR200907227 A TR 200907227A TR 200907227 A2 TR200907227 A2 TR 200907227A2
- Authority
- TR
- Turkey
- Prior art keywords
- high solubility
- stable micronized
- micronized granules
- granules
- stable
- Prior art date
Links
- 239000008187 granular material Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 abstract 1
- FABPRXSRWADJSP-MEDUHNTESA-N moxifloxacin Chemical compound COC1=C(N2C[C@H]3NCCC[C@H]3C2)C(F)=CC(C(C(C(O)=O)=C2)=O)=C1N2C1CC1 FABPRXSRWADJSP-MEDUHNTESA-N 0.000 abstract 1
- 229960003702 moxifloxacin Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Mevcut buluş, çözünürlük ve stabilite özellikleri geliştirilmiş moksifloksasin bileşimlerine, bu bileşimlerin hazırlanma yöntemine ve tıbbi kullanımına ilişkindir.
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2009/07227A TR200907227A2 (tr) | 2009-09-18 | 2009-09-18 | Çözünürlüğü yüksek stabil mikronize granüller. |
| PCT/TR2010/000181 WO2011034514A2 (en) | 2009-09-18 | 2010-09-06 | Stable micronized granules having high solubility |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2009/07227A TR200907227A2 (tr) | 2009-09-18 | 2009-09-18 | Çözünürlüğü yüksek stabil mikronize granüller. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR200907227A2 true TR200907227A2 (tr) | 2011-04-21 |
Family
ID=43759215
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2009/07227A TR200907227A2 (tr) | 2009-09-18 | 2009-09-18 | Çözünürlüğü yüksek stabil mikronize granüller. |
Country Status (2)
| Country | Link |
|---|---|
| TR (1) | TR200907227A2 (tr) |
| WO (1) | WO2011034514A2 (tr) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI1106900A2 (pt) * | 2011-12-26 | 2013-11-05 | Ems Sa | Composição farmacêutica sólida compreendendo antibótico da familia das quinolonas e processo de sua obtenção |
| GR1008169B (el) * | 2013-03-19 | 2014-04-08 | "Φαρματεν Α.Β.Ε.Ε.", | Φαρμακευτικο σκευασμα περιεχον εναν αντιβακτηριακο παραγοντα φθοριοκινολονης και μεθοδος για την παρασκευη αυτου |
| HUE058207T2 (hu) | 2017-01-31 | 2022-07-28 | Veru Inc | Készítmények és módszerek gonadotropin felszabadító hormon (GNRH) antagonisták elnyújtott idejû felszabadítására |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TR200101310T2 (tr) * | 1998-11-10 | 2001-10-22 | Bayer Aktiengesellschaft | Farmasötik moksifloksasin preparatı. |
| WO2009135646A2 (en) * | 2008-05-05 | 2009-11-12 | Farmaprojects, Sa | Stable pharmaceutical compositions and their processes for preparation suitable for industrial scale |
| ES2391132T3 (es) * | 2008-10-09 | 2012-11-21 | Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi | Uso de disolventes orgánicos en la granulación húmeda de moxifloxacino |
-
2009
- 2009-09-18 TR TR2009/07227A patent/TR200907227A2/tr unknown
-
2010
- 2010-09-06 WO PCT/TR2010/000181 patent/WO2011034514A2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011034514A2 (en) | 2011-03-24 |
| WO2011034514A3 (en) | 2011-11-10 |
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