TR201200588A2 - Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler. - Google Patents
Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler.Info
- Publication number
- TR201200588A2 TR201200588A2 TR2012/00588A TR201200588A TR201200588A2 TR 201200588 A2 TR201200588 A2 TR 201200588A2 TR 2012/00588 A TR2012/00588 A TR 2012/00588A TR 201200588 A TR201200588 A TR 201200588A TR 201200588 A2 TR201200588 A2 TR 201200588A2
- Authority
- TR
- Turkey
- Prior art keywords
- polymorphs
- mixtures
- processes
- preparing sodium
- sodium ibandronate
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 2
- -1 sodium ibandronate monohydrate Chemical class 0.000 title 1
- NASFKTWZWDYFER-UHFFFAOYSA-N sodium;hydrate Chemical compound O.[Na] NASFKTWZWDYFER-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
Abstract
Bu buluş [1-hidroksi-3-(metilpentilamino)propil den]bis-1,1-fosfonik asit monosodyum monohidrat'ın polimorflarının veya polimorf karışımlarının hazırlanması için geliştirilen prosesler ile ilgilidir.
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2012/00588A TR201200588A2 (tr) | 2012-01-18 | 2012-01-18 | Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler. |
| PCT/TR2012/000214 WO2013109198A1 (en) | 2012-01-18 | 2012-12-14 | Processes for the preparation of sodium ibandronate monohydrate polymorphs a, b and mixture of polymorphs a with b |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2012/00588A TR201200588A2 (tr) | 2012-01-18 | 2012-01-18 | Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR201200588A2 true TR201200588A2 (tr) | 2012-07-23 |
Family
ID=47004341
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2012/00588A TR201200588A2 (tr) | 2012-01-18 | 2012-01-18 | Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler. |
Country Status (2)
| Country | Link |
|---|---|
| TR (1) | TR201200588A2 (tr) |
| WO (1) | WO2013109198A1 (tr) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN109608492B (zh) * | 2018-12-19 | 2021-02-09 | 深圳市第二人民医院 | 一种用于骨质疏松的二膦酸化合物及其制备方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3623397A1 (de) | 1986-07-11 | 1988-01-14 | Boehringer Mannheim Gmbh | Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
| CN101111504B (zh) | 2005-02-01 | 2011-12-21 | 霍夫曼-拉罗奇有限公司 | 伊班膦酸盐多晶型物a |
| CA2594717C (en) * | 2005-02-01 | 2015-01-20 | F. Hoffmann-La Roche Ag | Ibandronate polymorph b |
| WO2007074475A2 (en) * | 2005-12-27 | 2007-07-05 | Natco Pharma Limited | Novel polymorphic forms of ibandronate |
| WO2008014510A2 (en) * | 2006-07-28 | 2008-01-31 | Dr. Reddy's Laboratories Limited | Crystalline form a of ibandronic acid and process for the preparation |
-
2012
- 2012-01-18 TR TR2012/00588A patent/TR201200588A2/tr unknown
- 2012-12-14 WO PCT/TR2012/000214 patent/WO2013109198A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2013109198A1 (en) | 2013-07-25 |
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