TR201200588A2 - Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler. - Google Patents

Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler.

Info

Publication number
TR201200588A2
TR201200588A2 TR2012/00588A TR201200588A TR201200588A2 TR 201200588 A2 TR201200588 A2 TR 201200588A2 TR 2012/00588 A TR2012/00588 A TR 2012/00588A TR 201200588 A TR201200588 A TR 201200588A TR 201200588 A2 TR201200588 A2 TR 201200588A2
Authority
TR
Turkey
Prior art keywords
polymorphs
mixtures
processes
preparing sodium
sodium ibandronate
Prior art date
Application number
TR2012/00588A
Other languages
English (en)
Inventor
Aslan Tuncer
Koçak Ender
Original Assignee
Koçak Farma İlaç Ve Ki̇mya Sanayi̇ Anoni̇m Şi̇rketi̇
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Koçak Farma İlaç Ve Ki̇mya Sanayi̇ Anoni̇m Şi̇rketi̇ filed Critical Koçak Farma İlaç Ve Ki̇mya Sanayi̇ Anoni̇m Şi̇rketi̇
Priority to TR2012/00588A priority Critical patent/TR201200588A2/tr
Publication of TR201200588A2 publication Critical patent/TR201200588A2/tr
Priority to PCT/TR2012/000214 priority patent/WO2013109198A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)

Abstract

Bu buluş [1-hidroksi-3-(metilpentilamino)propil den]bis-1,1-fosfonik asit monosodyum monohidrat'ın polimorflarının veya polimorf karışımlarının hazırlanması için geliştirilen prosesler ile ilgilidir.
TR2012/00588A 2012-01-18 2012-01-18 Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler. TR201200588A2 (tr)

Priority Applications (2)

Application Number Priority Date Filing Date Title
TR2012/00588A TR201200588A2 (tr) 2012-01-18 2012-01-18 Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler.
PCT/TR2012/000214 WO2013109198A1 (en) 2012-01-18 2012-12-14 Processes for the preparation of sodium ibandronate monohydrate polymorphs a, b and mixture of polymorphs a with b

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
TR2012/00588A TR201200588A2 (tr) 2012-01-18 2012-01-18 Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler.

Publications (1)

Publication Number Publication Date
TR201200588A2 true TR201200588A2 (tr) 2012-07-23

Family

ID=47004341

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2012/00588A TR201200588A2 (tr) 2012-01-18 2012-01-18 Sodyum ibandronat monohidrat polimorflarini ve polimorflu karışımlarını hazırlamak için prosesler.

Country Status (2)

Country Link
TR (1) TR201200588A2 (tr)
WO (1) WO2013109198A1 (tr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109608492B (zh) * 2018-12-19 2021-02-09 深圳市第二人民医院 一种用于骨质疏松的二膦酸化合物及其制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3623397A1 (de) 1986-07-11 1988-01-14 Boehringer Mannheim Gmbh Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel
CN101111504B (zh) 2005-02-01 2011-12-21 霍夫曼-拉罗奇有限公司 伊班膦酸盐多晶型物a
CA2594717C (en) * 2005-02-01 2015-01-20 F. Hoffmann-La Roche Ag Ibandronate polymorph b
WO2007074475A2 (en) * 2005-12-27 2007-07-05 Natco Pharma Limited Novel polymorphic forms of ibandronate
WO2008014510A2 (en) * 2006-07-28 2008-01-31 Dr. Reddy's Laboratories Limited Crystalline form a of ibandronic acid and process for the preparation

Also Published As

Publication number Publication date
WO2013109198A1 (en) 2013-07-25

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