TR201720672A2 - İvabradi̇ni̇n kontrollü salimli farmasöti̇k kompozi̇syonlari - Google Patents

İvabradi̇ni̇n kontrollü salimli farmasöti̇k kompozi̇syonlari Download PDF

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Publication number
TR201720672A2
TR201720672A2 TR2017/20672A TR201720672A TR201720672A2 TR 201720672 A2 TR201720672 A2 TR 201720672A2 TR 2017/20672 A TR2017/20672 A TR 2017/20672A TR 201720672 A TR201720672 A TR 201720672A TR 201720672 A2 TR201720672 A2 TR 201720672A2
Authority
TR
Turkey
Prior art keywords
controlled release
ivabradine
pharmaceutical compositions
release pharmaceutical
polymorph
Prior art date
Application number
TR2017/20672A
Other languages
English (en)
Inventor
Güner Di̇cle
Palantöken Arzu
Türkyilmaz Ali̇
Original Assignee
Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi filed Critical Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi
Priority to TR2017/20672A priority Critical patent/TR201720672A2/tr
Priority to PCT/TR2018/050818 priority patent/WO2019209208A2/en
Publication of TR201720672A2 publication Critical patent/TR201720672A2/tr

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Mevcut buluş, ivabradin veya farmasötik olarak kabul edilebilir bir tuzunu, solvatını veya polimorfunu ve en az bir kontrollü salım ajan içeren kontrollü salımlı farmasötik kompozisyonlarla ilgilidir.
TR2017/20672A 2017-12-18 2017-12-18 İvabradi̇ni̇n kontrollü salimli farmasöti̇k kompozi̇syonlari TR201720672A2 (tr)

Priority Applications (2)

Application Number Priority Date Filing Date Title
TR2017/20672A TR201720672A2 (tr) 2017-12-18 2017-12-18 İvabradi̇ni̇n kontrollü salimli farmasöti̇k kompozi̇syonlari
PCT/TR2018/050818 WO2019209208A2 (en) 2017-12-18 2018-12-17 Controlled-release pharmaceutical compositions of ivabradine

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
TR2017/20672A TR201720672A2 (tr) 2017-12-18 2017-12-18 İvabradi̇ni̇n kontrollü salimli farmasöti̇k kompozi̇syonlari

Publications (1)

Publication Number Publication Date
TR201720672A2 true TR201720672A2 (tr) 2019-07-22

Family

ID=67900851

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2017/20672A TR201720672A2 (tr) 2017-12-18 2017-12-18 İvabradi̇ni̇n kontrollü salimli farmasöti̇k kompozi̇syonlari

Country Status (2)

Country Link
TR (1) TR201720672A2 (tr)
WO (1) WO2019209208A2 (tr)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010128525A2 (en) * 2009-05-04 2010-11-11 Dinesh Shantilal Patel A formulation of ivabradine for treating the cardiovascular disease
PL2579859T3 (pl) * 2010-06-14 2015-12-31 Ratiopharm Gmbh Kompozycja stała zawierająca iwabradynę
CN102908327B (zh) * 2011-08-05 2015-03-11 江苏恒瑞医药股份有限公司 伊伐布雷定或其可药用盐的缓释制剂

Also Published As

Publication number Publication date
WO2019209208A3 (en) 2020-01-16
WO2019209208A2 (en) 2019-10-31

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