TR201722323A2 - Dabi̇gatranin oral farmasöti̇k kompozi̇syonlari - Google Patents
Dabi̇gatranin oral farmasöti̇k kompozi̇syonlariInfo
- Publication number
- TR201722323A2 TR201722323A2 TR2017/22323A TR201722323A TR201722323A2 TR 201722323 A2 TR201722323 A2 TR 201722323A2 TR 2017/22323 A TR2017/22323 A TR 2017/22323A TR 201722323 A TR201722323 A TR 201722323A TR 201722323 A2 TR201722323 A2 TR 201722323A2
- Authority
- TR
- Turkey
- Prior art keywords
- pharmaceutical compositions
- dabigatran
- oral pharmaceutical
- dabigatran etexilate
- componenet
- Prior art date
Links
- YBSJFWOBGCMAKL-UHFFFAOYSA-N dabigatran Chemical group N=1C2=CC(C(=O)N(CCC(O)=O)C=3N=CC=CC=3)=CC=C2N(C)C=1CNC1=CC=C(C(N)=N)C=C1 YBSJFWOBGCMAKL-UHFFFAOYSA-N 0.000 title 1
- 229960003850 dabigatran Drugs 0.000 title 1
- 239000008203 oral pharmaceutical composition Substances 0.000 title 1
- 229960000288 dabigatran etexilate Drugs 0.000 abstract 2
- KSGXQBZTULBEEQ-UHFFFAOYSA-N dabigatran etexilate Chemical compound C1=CC(C(N)=NC(=O)OCCCCCC)=CC=C1NCC1=NC2=CC(C(=O)N(CCC(=O)OCC)C=3N=CC=CC=3)=CC=C2N1C KSGXQBZTULBEEQ-UHFFFAOYSA-N 0.000 abstract 2
- 239000012458 free base Substances 0.000 abstract 1
- 150000007524 organic acids Chemical class 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Mevcut buluş, dabigatran eteksilat serbest bazını veya dabigatran eteksilatın farmasötik olarak kabul edilebilir tuzlarını içeren bir birinci bileşen ve bir organik asit içeren bir ikinci bileşen içeren oral uygulama için farmasötik kompozisyonlarla ilgilidir.
Priority Applications (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2017/22323A TR201722323A2 (tr) | 2017-12-27 | 2017-12-27 | Dabi̇gatranin oral farmasöti̇k kompozi̇syonlari |
| PCT/TR2018/050901 WO2019132839A1 (en) | 2017-12-27 | 2018-12-26 | Oral pharmaceutical compositions of dabigatran |
| EP18877293.3A EP3731822A1 (en) | 2017-12-27 | 2018-12-26 | Oral pharmaceutical compositions of dabigatran |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2017/22323A TR201722323A2 (tr) | 2017-12-27 | 2017-12-27 | Dabi̇gatranin oral farmasöti̇k kompozi̇syonlari |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR201722323A2 true TR201722323A2 (tr) | 2019-07-22 |
Family
ID=66476807
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2017/22323A TR201722323A2 (tr) | 2017-12-27 | 2017-12-27 | Dabi̇gatranin oral farmasöti̇k kompozi̇syonlari |
Country Status (3)
| Country | Link |
|---|---|
| EP (1) | EP3731822A1 (tr) |
| TR (1) | TR201722323A2 (tr) |
| WO (1) | WO2019132839A1 (tr) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112266475B (zh) * | 2020-11-05 | 2022-02-22 | 中国科学院长春应用化学研究所 | 一种二氧化碳聚酯多元醇、全生物降解二氧化碳基聚氨酯及其制备方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE121699A1 (es) | 1997-02-18 | 1999-12-08 | Boehringer Ingelheim Pharma | Heterociclos biciclicos disustituidos como inhibidores de la trombina |
| CA2476054C (en) | 2002-03-07 | 2011-11-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Pharmaceutical composition for the oral administration of 3-[(2-{[4-(hexyloxycarbonylamino-imino-methyl)-phenylamino)-methyl}-1-methyl-1h-benzimidazol-5-carbonyl)-pyridin-2-yl-amino)-propionic acid ethyl ester and the salts thereof |
| DE10337697A1 (de) | 2003-08-16 | 2005-03-24 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Tablette enthaltend 3-[(2-{[4-(Hexyloxycarbonylamino-imino-methyl)-phenyl-amino]-methyl}-1-methyl-1H-benzimidazol-5-carbonyl)-pyridin-2-yl-amino]-propionsäure-ethylester oder dessen Salze |
| DE102005020002A1 (de) | 2005-04-27 | 2006-11-02 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Physiologisch verträgliche Salze von 3-[(2-{[4-(Hexyloxycarbonylamino-imino-methyl)-phenylamino]-methyl}-1-methyl-1H-benzimidazol-5-carbonyl)-pyridin-2-yl-amino]-propionsäure-ethylester |
| PL2588090T3 (pl) | 2010-07-01 | 2017-12-29 | Krka, Tovarna Zdravil, D.D., Novo Mesto | Doustne farmaceutyczne postacie dawkowania zawierające eteksylan dabigatranu i jego farmaceutycznie dopuszczalne sole |
| US9006448B2 (en) | 2010-12-06 | 2015-04-14 | Msn Laboratories Private Limited | Process for the preparation of benzimidazole derivatives and its salts |
| HUE056194T2 (hu) | 2012-02-21 | 2022-01-28 | Towa Pharmaceutical Europe S L | Dabigatrán-etexilát orális gyógyszerészeti készítményei |
| IN2013CH05441A (tr) * | 2013-11-26 | 2015-05-29 | Aurobindo Pharma Ltd | |
| IN2014MU01042A (tr) * | 2014-03-26 | 2015-10-02 | Cadila Healthcare Ltd | |
| KR20170070635A (ko) * | 2015-12-14 | 2017-06-22 | 한미약품 주식회사 | 다비가트란 이텍실레이트를 함유하는 복합 캡슐제 |
-
2017
- 2017-12-27 TR TR2017/22323A patent/TR201722323A2/tr unknown
-
2018
- 2018-12-26 EP EP18877293.3A patent/EP3731822A1/en not_active Withdrawn
- 2018-12-26 WO PCT/TR2018/050901 patent/WO2019132839A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2019132839A1 (en) | 2019-07-04 |
| EP3731822A1 (en) | 2020-11-04 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JOP20200122A1 (ar) | مركبات مفيدة لتثبيط cdk7 | |
| SA519410865B1 (ar) | مركب حلقي شبيه بكُومارين بوصفه مثبط mek واستخدامه | |
| NZ780890A (en) | Pharmaceutical compositions comprising meloxicam | |
| EA201201263A1 (ru) | Фармацевтическая композиция, содержащая этексилат дабигатрана | |
| EA201792592A1 (ru) | Фармацевтические препараты, содержащие тенофовир и эмтрицитабин | |
| CY1124251T1 (el) | Παραγωγα καρβοξαμιδιου | |
| EA201201202A1 (ru) | Пероральная фармацевтическая композиция, содержащая этексилат дабигатрана | |
| IN2013CH05441A (tr) | ||
| PH12017500029A1 (en) | 4,5-dihydroisoxazole derivatives as nampt inhibitors | |
| IN2014MN02245A (tr) | ||
| IL264880A (en) | Preparations for oral administration of active substances | |
| MX387731B (es) | Composiciones farmacéuticas orales de mesalazina. | |
| MX2016013431A (es) | Composiciones farmaceuticas que comprenden agentes antibacterianos. | |
| IN2014MU01042A (tr) | ||
| MX2023012198A (es) | Composiciones de amantadina, preparaciones de estas y metodos de uso. | |
| WO2016142821A3 (en) | Compositions containing a thrombin inhibitor | |
| NZ740587A (en) | Fluoroindole derivatives as muscarinic m1 receptor positive allosteric modulators | |
| MX385513B (es) | Composiciones farmaceuticas que comprenden safinamida. | |
| TR201722323A2 (tr) | Dabi̇gatranin oral farmasöti̇k kompozi̇syonlari | |
| WO2020032885A3 (en) | Capsule-in-capsule compositions of dabigatran etexilate | |
| WO2019004980A3 (en) | SOLID ORAL PHARMACEUTICAL COMPOSITIONS OF DABIGATRAN DEXILATE | |
| IN2014MU00859A (tr) | ||
| TR201722186A2 (tr) | Dabi̇gatranin farmasöti̇k kompozi̇syonlari | |
| WO2019151966A3 (en) | Pharmaceutical tablet compositions of dabigatran | |
| IN2013MU03421A (tr) |