TR201902178T4 - Akti̇ni̇k keratozun tedavi̇si̇ne yöneli̇k düşük dozaj yi̇ti̇li̇ği̇ne sahi̇p i̇mi̇kui̇mod formülasyonlari ve kisa dozajli reji̇mler. - Google Patents
Akti̇ni̇k keratozun tedavi̇si̇ne yöneli̇k düşük dozaj yi̇ti̇li̇ği̇ne sahi̇p i̇mi̇kui̇mod formülasyonlari ve kisa dozajli reji̇mler. Download PDFInfo
- Publication number
- TR201902178T4 TR201902178T4 TR2019/02178T TR201902178T TR201902178T4 TR 201902178 T4 TR201902178 T4 TR 201902178T4 TR 2019/02178 T TR2019/02178 T TR 2019/02178T TR 201902178 T TR201902178 T TR 201902178T TR 201902178 T4 TR201902178 T4 TR 201902178T4
- Authority
- TR
- Turkey
- Prior art keywords
- dosage
- loss
- imiquimod
- formulations
- actinic keratosis
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 2
- DOUYETYNHWVLEO-UHFFFAOYSA-N imiquimod Chemical compound C1=CC=CC2=C3N(CC(C)C)C=NC3=C(N)N=C21 DOUYETYNHWVLEO-UHFFFAOYSA-N 0.000 abstract 8
- 229960002751 imiquimod Drugs 0.000 abstract 5
- 208000009621 actinic keratosis Diseases 0.000 abstract 3
- 229940060265 aldara Drugs 0.000 abstract 2
- 239000006071 cream Substances 0.000 abstract 2
- 238000001647 drug administration Methods 0.000 abstract 2
- 238000009472 formulation Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
- 230000037317 transdermal delivery Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
ABD Gıda & İlaç Dairesi ("FDA") tarafından onaylandığı üzere, ticari olarak temin edilebilen Aldara® %5 imikuimod kremi için mevcut olarak reçetelendirilenden, daha kısa terapi süreleriyle aktinik keratozu tedavi etmek üzere diğer adı imikuimod olan 1izobütil-1Himidazo[4,5-c]-kinolin-4-amin veya 1-(2-metilpropil)-1H-imidazo[4,5-c]kinolin-4-aminin opikal veya transdermal iletime yönelik farmasötik formülasyonlar ve yöntemler tarif edilmektedir ve açıklanmaktadır. Daha spesifik olarak, aktinik keratozu tedavi etmek üzere Aldara® %5 imikuimod kremi için ABD Gıda & İlaç Dairesi ("FDA") tarafından mevcut olarak onaylanan dozaj rejiminden, hasta kullanımı için kısa ve daha uygun olan bir kabul edilebilir güvenlik profili ve dozaj rejimlerine sahip aktinik keratozun tedavi edilmesine yönelik etkili bir imikuimod dozunu iletmek için daha düşük dozaj yitiliğe sahip imikuimod formülasyonları da tarif edilmekte ve açıklanmaktadır.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13953608P | 2008-12-19 | 2008-12-19 | |
| US20514508P | 2008-12-19 | 2008-12-19 | |
| US14473108P | 2008-12-19 | 2008-12-19 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR201902178T4 true TR201902178T4 (tr) | 2019-04-22 |
Family
ID=67981265
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2019/02178T TR201902178T4 (tr) | 2008-12-19 | 2009-12-11 | Akti̇ni̇k keratozun tedavi̇si̇ne yöneli̇k düşük dozaj yi̇ti̇li̇ği̇ne sahi̇p i̇mi̇kui̇mod formülasyonlari ve kisa dozajli reji̇mler. |
Country Status (1)
| Country | Link |
|---|---|
| TR (1) | TR201902178T4 (tr) |
-
2009
- 2009-12-11 TR TR2019/02178T patent/TR201902178T4/tr unknown
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