TW201326134A - 以被取代吡唑基甲醯胺及被以一含氮基團取代之含有一苯基基元之尿素衍生物做為類香草素受體之配位體 - Google Patents

以被取代吡唑基甲醯胺及被以一含氮基團取代之含有一苯基基元之尿素衍生物做為類香草素受體之配位體 Download PDF

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TW201326134A
TW201326134A TW101141482A TW101141482A TW201326134A TW 201326134 A TW201326134 A TW 201326134A TW 101141482 A TW101141482 A TW 101141482A TW 101141482 A TW101141482 A TW 101141482A TW 201326134 A TW201326134 A TW 201326134A
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Taiwan
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methyl
phenyl
pyrazol
fluoro
group
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TW101141482A
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English (en)
Chinese (zh)
Inventor
Robert Frank
Thomas Christoph
Nils Damann
Bernhard Lesch
Gregor Bahrenberg
Derek John Saunders
Hannelore Stockhausen
Yong-Soo Kim
Myeong-Seop Kim
Jee-Woo Lee
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Gruenenthal Gmbh
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Publication of TW201326134A publication Critical patent/TW201326134A/zh

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
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TW101141482A 2011-11-09 2012-11-08 以被取代吡唑基甲醯胺及被以一含氮基團取代之含有一苯基基元之尿素衍生物做為類香草素受體之配位體 TW201326134A (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP11008913 2011-11-09

Publications (1)

Publication Number Publication Date
TW201326134A true TW201326134A (zh) 2013-07-01

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Application Number Title Priority Date Filing Date
TW101141482A TW201326134A (zh) 2011-11-09 2012-11-08 以被取代吡唑基甲醯胺及被以一含氮基團取代之含有一苯基基元之尿素衍生物做為類香草素受體之配位體

Country Status (13)

Country Link
EP (1) EP2776399A1 (sr)
JP (1) JP2014532742A (sr)
KR (1) KR20140096351A (sr)
CN (1) CN103906736A (sr)
AR (1) AR088701A1 (sr)
AU (1) AU2012334066A1 (sr)
BR (1) BR112014010957A2 (sr)
CA (1) CA2854935A1 (sr)
HK (1) HK1202116A1 (sr)
IN (1) IN2014KN00847A (sr)
MX (1) MX2014005611A (sr)
TW (1) TW201326134A (sr)
WO (1) WO2013068462A1 (sr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107108593B (zh) * 2014-11-24 2020-03-24 美迪福伦Dbt有限公司 作为类香草素受体配体ii的基于取代的恶唑和噻唑的羧酰胺和脲衍生物
CN114920697A (zh) * 2022-05-16 2022-08-19 河南应用技术职业学院 杂环基取代的茚满丙酰胺类化合物及其应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999012910A1 (en) * 1997-09-11 1999-03-18 Nissan Chemical Industries, Ltd. Pyrazole compounds and plant disease control agent
KR101347102B1 (ko) * 2005-10-19 2014-01-03 그뤼넨탈 게엠베하 신규한 바닐로이드 수용체 리간드 및 약제를 제조하기 위한이의 용도
WO2008073825A1 (en) * 2006-12-08 2008-06-19 Exelixis, Inc. Lxr and fxr modulators
RU2498982C2 (ru) * 2007-04-16 2013-11-20 Грюненталь Гмбх Новые лиганды ванилоидных рецепторов и их применение для изготовления лекарственных средств
DE102007018151A1 (de) * 2007-04-16 2008-10-23 Günenthal GmbH Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
CA2758289A1 (en) 2009-05-07 2010-11-11 Gruenenthal Gmbh Substituted aromatic carboxamide and urea derivatives as vanilloid receptor ligands
JP5745505B2 (ja) 2009-05-07 2015-07-08 グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング バニロイド受容体リガンドとしての置換フェニル尿素および置換フェニルアミド
JP2014532743A (ja) * 2011-11-09 2014-12-08 グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング バニロイド受容体リガンドとしての、n−環式基で置換されたフェニル部分を担持する置換ピラゾリルをベースとするカルボキサミドおよび尿素誘導体

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Publication number Publication date
KR20140096351A (ko) 2014-08-05
CA2854935A1 (en) 2013-05-16
HK1202116A1 (en) 2015-09-18
CN103906736A (zh) 2014-07-02
AR088701A1 (es) 2014-06-25
EP2776399A1 (en) 2014-09-17
MX2014005611A (es) 2014-07-30
WO2013068462A1 (en) 2013-05-16
JP2014532742A (ja) 2014-12-08
BR112014010957A2 (pt) 2017-06-06
IN2014KN00847A (sr) 2015-10-02
AU2012334066A1 (en) 2014-05-22

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