TWI449692B - 吡咯烷化合物(三) - Google Patents

吡咯烷化合物(三) Download PDF

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Publication number
TWI449692B
TWI449692B TW102143870A TW102143870A TWI449692B TW I449692 B TWI449692 B TW I449692B TW 102143870 A TW102143870 A TW 102143870A TW 102143870 A TW102143870 A TW 102143870A TW I449692 B TWI449692 B TW I449692B
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TW
Taiwan
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group
lower alkyl
phenyl
fluorophenyl
pyrrolidin
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TW102143870A
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English (en)
Chinese (zh)
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TW201412708A (zh
Inventor
Muneaki Kurimura
Shinichi Taira
Takahiro Tomoyasu
Nobuaki Ito
Kuninori Tai
Noriaki Takemura
Takayuki Matsuzaki
Yasuhiro Menjo
Shin Miyamura
Yohji Sakurai
Akihito Watanabe
Yasuyo Sakata
Takumi Masumoto
Kohei Akazawa
Haruhiko Sugino
Naoki Amada
Satoshi Ohashi
Tomoichi Shinohara
Hirofumi Sasaki
Chisako Morita
Junko Yamashita
Satoko Nakajima
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Otsuka Pharma Co Ltd
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Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of TW201412708A publication Critical patent/TW201412708A/zh
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TW102143870A 2005-05-13 2006-05-08 吡咯烷化合物(三) TWI449692B (zh)

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Application Number Priority Date Filing Date Title
JP2005141230 2005-05-13

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TW201412708A TW201412708A (zh) 2014-04-01
TWI449692B true TWI449692B (zh) 2014-08-21

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TW102143870A TWI449692B (zh) 2005-05-13 2006-05-08 吡咯烷化合物(三)
TW095116220A TWI410406B (zh) 2005-05-13 2006-05-08 吡咯烷化合物
TW102101997A TWI439452B (zh) 2005-05-13 2006-05-08 吡咯烷化合物(二)

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TW102101997A TWI439452B (zh) 2005-05-13 2006-05-08 吡咯烷化合物(二)

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US (6) US8084442B2 (2)
EP (2) EP2407451B1 (2)
JP (1) JP4776631B2 (2)
KR (2) KR100971850B1 (2)
CN (3) CN103613587A (2)
AR (1) AR054191A1 (2)
AU (2) AU2006244851B2 (2)
BR (1) BRPI0610279A2 (2)
CA (1) CA2608184C (2)
CY (1) CY1114767T1 (2)
DK (1) DK2407451T3 (2)
ES (2) ES2446375T3 (2)
IL (1) IL187311A (2)
IN (1) IN2012DN00758A (2)
MX (1) MX2007014252A (2)
MY (1) MY148653A (2)
PL (1) PL2407451T3 (2)
PT (1) PT2407451E (2)
RU (1) RU2414454C2 (2)
SG (1) SG162722A1 (2)
SI (1) SI2407451T1 (2)
TW (3) TWI449692B (2)
WO (1) WO2006121218A1 (2)
ZA (1) ZA200709691B (2)

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EP1565436B1 (en) 2002-11-27 2012-04-25 Incyte Corporation 3-aminopyrrolidine derivatives as modulators of chemokine receptors
TWI449692B (zh) 2005-05-13 2014-08-21 Otsuka Pharma Co Ltd 吡咯烷化合物(三)
EP1954133A4 (en) * 2005-11-30 2010-11-24 Glaxosmithkline Llc PYRROLIDINANILINE
EP1960355A1 (en) * 2005-11-30 2008-08-27 F.Hoffmann-La Roche Ag 3-amino-1-arylpropyl indoles and aza-substituted indoles
JP5219465B2 (ja) * 2006-11-10 2013-06-26 大塚製薬株式会社 医薬
CN101977907A (zh) 2008-03-20 2011-02-16 弗·哈夫曼-拉罗切有限公司 吡咯烷基衍生物及其用途
EP2496234A1 (en) 2009-11-07 2012-09-12 Merck Patent GmbH Heteroarylaminoquinolines as tgf-beta receptor kinase inhibitors
WO2011131748A2 (en) * 2010-04-21 2011-10-27 Probiodrug Ag Novel inhibitors
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