UA105164C2 - Substituted 8-[6-amino-3-pyridyl]xanthines - Google Patents
Substituted 8-[6-amino-3-pyridyl]xanthinesInfo
- Publication number
- UA105164C2 UA105164C2 UAA200900239A UAA200900239A UA105164C2 UA 105164 C2 UA105164 C2 UA 105164C2 UA A200900239 A UAA200900239 A UA A200900239A UA A200900239 A UAA200900239 A UA A200900239A UA 105164 C2 UA105164 C2 UA 105164C2
- Authority
- UA
- Ukraine
- Prior art keywords
- xanthines
- pyridyl
- amino
- substituted
- compositions
- Prior art date
Links
- DIVYESOURJTWDY-UHFFFAOYSA-N 8-(6-aminopyridin-3-yl)-3,7-dihydropurine-2,6-dione Chemical class C1=NC(N)=CC=C1C(N1)=NC2=C1C(=O)NC(=O)N2 DIVYESOURJTWDY-UHFFFAOYSA-N 0.000 title abstract 2
- 108050000203 Adenosine receptors Proteins 0.000 abstract 1
- 102000009346 Adenosine receptors Human genes 0.000 abstract 1
- 101150078577 Adora2b gene Proteins 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000008177 pharmaceutical agent Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
- C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US80503006P | 2006-06-16 | 2006-06-16 | |
| PCT/US2007/013849 WO2007149277A2 (fr) | 2006-06-16 | 2007-06-13 | 8-[6-amino-3-pyridyl]xanthines substituées |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA105164C2 true UA105164C2 (en) | 2014-04-25 |
Family
ID=38833978
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200900239A UA105164C2 (en) | 2006-06-16 | 2007-06-13 | Substituted 8-[6-amino-3-pyridyl]xanthines |
Country Status (4)
| Country | Link |
|---|---|
| CN (1) | CN101466382A (fr) |
| UA (1) | UA105164C2 (fr) |
| WO (1) | WO2007149277A2 (fr) |
| ZA (1) | ZA200900259B (fr) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5460690B2 (ja) | 2008-03-26 | 2014-04-02 | アドヴィナス・セラピューティックス・リミテッド | アデノシンレセプターアンタゴニストとしてのヘテロ環化合物 |
| AU2010222289B2 (en) | 2009-03-13 | 2013-07-11 | Advinus Therapeutics Private Limited | Substituted fused pyrimidine compounds |
| EP2499142B1 (fr) | 2009-11-09 | 2016-09-21 | Advinus Therapeutics Limited | Composés pyrimidine fusionnés substitués, leur préparation et leurs utilisations |
| CN103261200B (zh) | 2010-09-13 | 2016-03-30 | 阿迪维纳斯疗法有限公司 | 作为a2b腺苷受体拮抗剂的前药的嘌呤化合物、它们的制备方法及医药用途 |
| MX2021008094A (es) | 2019-01-11 | 2021-09-21 | Omeros Corp | Metodos y composiciones para el tratamiento del cancer. |
| BR112023023996A2 (pt) * | 2021-05-18 | 2024-01-30 | Adovate Llc | Xantinas de piridil contendo amida cíclica como antagonistas de a2b |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4938949A (en) | 1988-09-12 | 1990-07-03 | University Of New York | Treatment of damaged bone marrow and dosage units therefor |
| KR101222364B1 (ko) * | 2003-08-25 | 2013-01-15 | 트로비스 파마슈티칼스 엘엘씨 | 치환된 8-헤테로아릴 크산틴 |
-
2007
- 2007-06-13 WO PCT/US2007/013849 patent/WO2007149277A2/fr not_active Ceased
- 2007-06-13 CN CNA2007800222077A patent/CN101466382A/zh active Pending
- 2007-06-13 UA UAA200900239A patent/UA105164C2/ru unknown
-
2009
- 2009-01-13 ZA ZA200900259A patent/ZA200900259B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007149277A3 (fr) | 2008-02-21 |
| CN101466382A (zh) | 2009-06-24 |
| WO2007149277A2 (fr) | 2007-12-27 |
| ZA200900259B (en) | 2010-09-29 |
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