UA84443C2 - Кристаллическая форма 2,3-диметил-8-(2,6-диметилбензиламино)-n-гидроксиэтилимидазо[1,2-а]пиридин-6-карбоксамид мезилата (варианты), способ их получения, фармацевтическая композиция и способ лечения желудочно-кишечных расстройств - Google Patents

Кристаллическая форма 2,3-диметил-8-(2,6-диметилбензиламино)-n-гидроксиэтилимидазо[1,2-а]пиридин-6-карбоксамид мезилата (варианты), способ их получения, фармацевтическая композиция и способ лечения желудочно-кишечных расстройств

Info

Publication number: UA84443C2
Authority: UA; Ukraine
Prior art keywords: dimethylbenzylamino; imidazo; hydroxyethyl; pyridine; dimethyl
Prior art date: 2003-12-18

Application number

UAA200605707A

Other languages

English (en)

Ukrainian (uk)

Inventor

Ларс Лилльеквист

Мария Линдквист

Петер Нордберг

Урсула Петерссон

Тесфаи Себгату

Original Assignee

Астразенека Аб

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-12-18

Filing date

2004-12-16

Publication date

2008-10-27

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=30768770&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA84443(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2004-12-16 Application filed by Астразенека Аб filed Critical Астразенека Аб

2008-10-27 Publication of UA84443C2 publication Critical patent/UA84443C2/ru

Links

238000000034 method Methods 0.000 title abstract 3
QCHUWMQLRFKFDK-UHFFFAOYSA-N 8-[(2,6-dimethylphenyl)methylamino]-n-(2-hydroxyethyl)-2,3-dimethylimidazo[1,2-a]pyridine-6-carboxamide;methanesulfonic acid Chemical compound CS(O)(=O)=O.C=1C(C(=O)NCCO)=CN2C(C)=C(C)N=C2C=1NCC1=C(C)C=CC=C1C QCHUWMQLRFKFDK-UHFFFAOYSA-N 0.000 title abstract 2
208000018522 Gastrointestinal disease Diseases 0.000 title abstract 2
239000008194 pharmaceutical composition Substances 0.000 title abstract 2
150000001875 compounds Chemical class 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Pulmonology (AREA)
Hospice & Palliative Care (AREA)
Otolaryngology (AREA)
Epidemiology (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

UAA200605707A 2003-12-18 2004-12-16 Кристаллическая форма 2,3-диметил-8-(2,6-диметилбензиламино)-n-гидроксиэтилимидазо[1,2-а]пиридин-6-карбоксамид мезилата (варианты), способ их получения, фармацевтическая композиция и способ лечения желудочно-кишечных расстройств UA84443C2 (ru)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
SE0303451A SE0303451D0 (sv)	2003-12-18	2003-12-18	New compounds
PCT/SE2004/001909 WO2005058895A1 (en)	2003-12-18	2004-12-16	Novel crystalline forms of 2, 3 dimethyl-8- (2, 6-dimethylbenzylamino) -n-hydroxyethyl-imidazo [1, 2-a] pyridine-6-carboxamide mesylate salt.

Publications (1)

Publication Number	Publication Date
UA84443C2 true UA84443C2 (ru)	2008-10-27

Family

ID=30768770

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
UAA200605707A UA84443C2 (ru)	2003-12-18	2004-12-16	Кристаллическая форма 2,3-диметил-8-(2,6-диметилбензиламино)-n-гидроксиэтилимидазо[1,2-а]пиридин-6-карбоксамид мезилата (варианты), способ их получения, фармацевтическая композиция и способ лечения желудочно-кишечных расстройств

Country Status (24)

Country	Link
US (1)	US7459463B2 (ru)
EP (1)	EP1697360B1 (ru)
JP (2)	JP2007514744A (ru)
KR (1)	KR20060125803A (ru)
CN (1)	CN1894246B (ru)
AR (1)	AR046956A1 (ru)
AT (1)	ATE499371T1 (ru)
AU (1)	AU2004299435B2 (ru)
BR (1)	BRPI0417640A (ru)
CA (1)	CA2549144A1 (ru)
CO (1)	CO5721004A2 (ru)
DE (1)	DE602004031556D1 (ru)
ES (1)	ES2359829T3 (ru)
IL (1)	IL175957A0 (ru)
MX (1)	MXPA06006708A (ru)
MY (1)	MY140450A (ru)
NO (1)	NO20063309L (ru)
RU (1)	RU2376306C2 (ru)
SE (1)	SE0303451D0 (ru)
TW (1)	TW200526659A (ru)
UA (1)	UA84443C2 (ru)
UY (1)	UY28676A1 (ru)
WO (1)	WO2005058895A1 (ru)
ZA (1)	ZA200604633B (ru)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2005041961A1 (en) *	2003-11-03	2005-05-12	Astrazeneca Ab	Imidazo [1,2-a] pyridine derivatives for the treatment of silent gastro-esophageal reflux
FI20086158A0 (fi)	2008-12-03	2008-12-03	Mikael Dahlstroem	Imidatsopyridiinijohdannaiset
JP2024530045A (ja)	2021-11-05	2024-08-14	シンクルス・ファーマ・ホールディング・アクチエボラグ	リナプラザングルレート塩酸塩の多形

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4040632A1 (de) *	1990-12-19	1992-06-25	Kali Chemie Pharma Gmbh	Phenylalkylaminoalkyl-verbindungen sowie verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
SE9700661D0 (sv) *	1997-02-25	1997-02-25	Astra Ab	New compounds
SE512531C2 (sv)	1997-09-04	2000-03-27	Astacarotene Ab	Användning av åtminstone en typ av xantofyller för framställning av ett läkemedel för profylaktisk och/eller terapeutisk förbättring av muskelfunktionsdurationen hos däggdjur och/eller behandling av muskelstörningar eller - sjukdomar hos däggdjur
SE9801526D0 (sv) *	1998-04-29	1998-04-29	Astra Ab	New compounds
SE0003186D0 (sv) *	2000-09-07	2000-09-07	Astrazeneca Ab	New process
SE0100295D0 (sv) *	2001-02-01	2001-02-01	Astrazeneca Ab	New compounds
SE0100297D0 (sv) *	2001-02-01	2001-02-01	Astrazeneca Ab	New compounds
SE0100296D0 (sv) *	2001-02-01	2001-02-01	Astrazeneca Ab	New compounds
CN1491104A (zh) *	2001-02-13	2004-04-21		新型改进释放制剂
JP2005528418A (ja) *	2002-05-07	2005-09-22	アルタナ　ファルマ　アクチエンゲゼルシャフト	気道疾患を治療するための新規組み合わせ

2003
- 2003-12-18 SE SE0303451A patent/SE0303451D0/xx unknown
2004
- 2004-12-15 TW TW093139011A patent/TW200526659A/zh unknown
- 2004-12-16 KR KR1020067011954A patent/KR20060125803A/ko not_active Ceased
- 2004-12-16 AT AT04809082T patent/ATE499371T1/de not_active IP Right Cessation
- 2004-12-16 EP EP04809082A patent/EP1697360B1/en not_active Expired - Lifetime
- 2004-12-16 UA UAA200605707A patent/UA84443C2/ru unknown
- 2004-12-16 MY MYPI20045189A patent/MY140450A/en unknown
- 2004-12-16 JP JP2006545292A patent/JP2007514744A/ja active Pending
- 2004-12-16 WO PCT/SE2004/001909 patent/WO2005058895A1/en not_active Ceased
- 2004-12-16 BR BRPI0417640-5A patent/BRPI0417640A/pt not_active IP Right Cessation
- 2004-12-16 AU AU2004299435A patent/AU2004299435B2/en not_active Ceased
- 2004-12-16 US US10/582,838 patent/US7459463B2/en not_active Expired - Fee Related
- 2004-12-16 CN CN2004800379883A patent/CN1894246B/zh not_active Expired - Fee Related
- 2004-12-16 CA CA002549144A patent/CA2549144A1/en not_active Abandoned
- 2004-12-16 DE DE602004031556T patent/DE602004031556D1/de not_active Expired - Lifetime
- 2004-12-16 ES ES04809082T patent/ES2359829T3/es not_active Expired - Lifetime
- 2004-12-16 MX MXPA06006708A patent/MXPA06006708A/es unknown
- 2004-12-16 RU RU2006123362/04A patent/RU2376306C2/ru not_active IP Right Cessation
- 2004-12-17 UY UY28676A patent/UY28676A1/es unknown
- 2004-12-17 AR ARP040104749A patent/AR046956A1/es not_active Application Discontinuation
2006
- 2006-05-25 IL IL175957A patent/IL175957A0/en unknown
- 2006-06-06 ZA ZA200604633A patent/ZA200604633B/en unknown
- 2006-06-20 CO CO06059763A patent/CO5721004A2/es not_active Application Discontinuation
- 2006-07-17 NO NO20063309A patent/NO20063309L/no not_active Application Discontinuation
2012
- 2012-01-23 JP JP2012010610A patent/JP2012102143A/ja active Pending

Also Published As

Publication number	Publication date
ATE499371T1 (de)	2011-03-15
JP2007514744A (ja)	2007-06-07
AU2004299435A1 (en)	2005-06-30
AR046956A1 (es)	2006-01-04
CN1894246B (zh)	2011-06-22
JP2012102143A (ja)	2012-05-31
ZA200604633B (en)	2007-04-25
ES2359829T3 (es)	2011-05-27
WO2005058895A1 (en)	2005-06-30
RU2376306C2 (ru)	2009-12-20
US7459463B2 (en)	2008-12-02
HK1095810A1 (en)	2007-05-18
MY140450A (en)	2009-12-31
US20070112021A1 (en)	2007-05-17
RU2006123362A (ru)	2008-01-27
UY28676A1 (es)	2005-07-29
TW200526659A (en)	2005-08-16
CA2549144A1 (en)	2005-06-30
SE0303451D0 (sv)	2003-12-18
IL175957A0 (en)	2006-10-05
CO5721004A2 (es)	2007-01-31
CN1894246A (zh)	2007-01-10
DE602004031556D1 (de)	2011-04-07
MXPA06006708A (es)	2006-08-18
AU2004299435B2 (en)	2008-04-17
NO20063309L (no)	2006-09-14
EP1697360B1 (en)	2011-02-23
EP1697360A1 (en)	2006-09-06
BRPI0417640A (pt)	2007-03-27
KR20060125803A (ko)	2006-12-06

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UA86614C2 (ru)	2009-05-12	Соединение, которое имеет активность ингибитора киназ, фармацевтическая композиция, которая включает указанное соединение, и их применение для приготовления лекарственного препарата
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WO2006011050A3 (en)	2006-10-05	Pyridine derivatives
TW200612892A (en)	2006-05-01	Novel compounds
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SI1730144T1 (sl)	2009-12-31	Substituirane spojine 1,4,8-triazaspiro(4.5)dekan-2-on
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