UA85201C2 - Производные дифенилацетидинона, которые являются ингибиторами абсорбции холестерола, способ их получения, фармацевтическая композиция на их основе - Google Patents
Производные дифенилацетидинона, которые являются ингибиторами абсорбции холестерола, способ их получения, фармацевтическая композиция на их основеInfo
- Publication number
- UA85201C2 UA85201C2 UAA200605758A UAA200605758A UA85201C2 UA 85201 C2 UA85201 C2 UA 85201C2 UA A200605758 A UAA200605758 A UA A200605758A UA A200605758 A UAA200605758 A UA A200605758A UA 85201 C2 UA85201 C2 UA 85201C2
- Authority
- UA
- Ukraine
- Prior art keywords
- preparation
- cholesterol absorption
- pharmaceutical composition
- inhibitory activity
- composition based
- Prior art date
Links
- 230000001906 cholesterol absorption Effects 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- VDOXIAUNJCHYRC-UHFFFAOYSA-N 1,3-diphenylazetidin-2-one Chemical class O=C1C(C=2C=CC=CC=2)CN1C1=CC=CC=C1 VDOXIAUNJCHYRC-UHFFFAOYSA-N 0.000 title 1
- 230000002401 inhibitory effect Effects 0.000 title 1
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000012453 solvate Substances 0.000 abstract 2
- 208000031226 Hyperlipidaemia Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Соединения формулы (І) (группы которых определены в описании), их фармацевтически приемлемые соли, сольваты, сольваты таких солей или пролекарства и их применение как ингибиторов абсорбции холестерола для лечения гиперлипидемии. Описаны также способ их получения и фармацевтические композиции, которые их содержат.(І)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0329780A GB0329780D0 (en) | 2003-12-23 | 2003-12-23 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA85201C2 true UA85201C2 (ru) | 2009-01-12 |
Family
ID=30776337
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200605758A UA85201C2 (ru) | 2003-12-23 | 2004-12-21 | Производные дифенилацетидинона, которые являются ингибиторами абсорбции холестерола, способ их получения, фармацевтическая композиция на их основе |
Country Status (4)
| Country | Link |
|---|---|
| CN (1) | CN101065354A (ru) |
| GB (1) | GB0329780D0 (ru) |
| UA (1) | UA85201C2 (ru) |
| ZA (1) | ZA200605161B (ru) |
-
2003
- 2003-12-23 GB GB0329780A patent/GB0329780D0/en not_active Ceased
-
2004
- 2004-12-21 CN CN 200480038465 patent/CN101065354A/zh active Pending
- 2004-12-21 UA UAA200605758A patent/UA85201C2/ru unknown
-
2006
- 2006-06-22 ZA ZA200605161A patent/ZA200605161B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN101065354A (zh) | 2007-10-31 |
| GB0329780D0 (en) | 2004-01-28 |
| ZA200605161B (en) | 2007-12-27 |
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