UA85220C2 - Эмульсия перфторорганических соединений медицинского назначения и способ ее получения - Google Patents
Эмульсия перфторорганических соединений медицинского назначения и способ ее полученияInfo
- Publication number
- UA85220C2 UA85220C2 UAA200610353A UAA200610353A UA85220C2 UA 85220 C2 UA85220 C2 UA 85220C2 UA A200610353 A UAA200610353 A UA A200610353A UA A200610353 A UAA200610353 A UA A200610353A UA 85220 C2 UA85220 C2 UA 85220C2
- Authority
- UA
- Ukraine
- Prior art keywords
- emulsion
- perfluororganic
- compounds
- mixture
- inventive
- Prior art date
Links
- 239000000839 emulsion Substances 0.000 title abstract 6
- 150000001875 compounds Chemical class 0.000 title abstract 5
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 abstract 4
- 239000008280 blood Substances 0.000 abstract 3
- 210000004369 blood Anatomy 0.000 abstract 3
- 239000006185 dispersion Substances 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 2
- WTWWXOGTJWMJHI-UHFFFAOYSA-N perflubron Chemical compound FC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)Br WTWWXOGTJWMJHI-UHFFFAOYSA-N 0.000 abstract 2
- 229960001217 perflubron Drugs 0.000 abstract 2
- 150000003904 phospholipids Chemical class 0.000 abstract 2
- 150000003512 tertiary amines Chemical class 0.000 abstract 2
- 206010021143 Hypoxia Diseases 0.000 abstract 1
- 239000000654 additive Substances 0.000 abstract 1
- 230000000996 additive effect Effects 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 230000001146 hypoxic effect Effects 0.000 abstract 1
- 230000000302 ischemic effect Effects 0.000 abstract 1
- 238000002483 medication Methods 0.000 abstract 1
- 210000000056 organ Anatomy 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 229950008618 perfluamine Drugs 0.000 abstract 1
- -1 perfluordecalin Chemical class 0.000 abstract 1
- JAJLKEVKNDUJBG-UHFFFAOYSA-N perfluorotripropylamine Chemical compound FC(F)(F)C(F)(F)C(F)(F)N(C(F)(F)C(F)(F)C(F)(F)F)C(F)(F)C(F)(F)C(F)(F)F JAJLKEVKNDUJBG-UHFFFAOYSA-N 0.000 abstract 1
- 210000002381 plasma Anatomy 0.000 abstract 1
- 210000002966 serum Anatomy 0.000 abstract 1
- 230000001954 sterilising effect Effects 0.000 abstract 1
- 238000004659 sterilization and disinfection Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0026—Blood substitute; Oxygen transporting formulations; Plasma extender
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/02—Halogenated hydrocarbons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/08—Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Hematology (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Dermatology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2004106722/15A RU2259819C1 (ru) | 2004-03-01 | 2004-03-01 | Эмульсия перфторорганических соединений медицинского назначения и способ её получения |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA85220C2 true UA85220C2 (ru) | 2009-01-12 |
Family
ID=34993426
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200610353A UA85220C2 (ru) | 2004-03-01 | 2005-02-07 | Эмульсия перфторорганических соединений медицинского назначения и способ ее получения |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7842730B2 (ru) |
| EP (1) | EP1736148A4 (ru) |
| JP (1) | JP2007525536A (ru) |
| CN (1) | CN101014326B (ru) |
| CA (1) | CA2557833A1 (ru) |
| EA (1) | EA010315B1 (ru) |
| RU (1) | RU2259819C1 (ru) |
| UA (1) | UA85220C2 (ru) |
| WO (1) | WO2005089739A1 (ru) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008082321A1 (fr) * | 2006-12-28 | 2008-07-10 | Germanov, Evgeny Pavlovich | Émulsions de composés organiques perfluorés médicinaux, procédé de préparation et procédé d'utilisation |
| RU2393849C2 (ru) * | 2006-12-28 | 2010-07-10 | Общество с ограниченной ответственностью "Биология и фармакология перфторсоединений" | Эмульсия перфторорганических соединений медицинского назначения, способ ее приготовления и способ ее применения |
| JP5340954B2 (ja) * | 2007-11-16 | 2013-11-13 | テクノガード株式会社 | 薬物含有脂肪乳剤およびその製造方法 |
| US8063020B2 (en) * | 2007-12-22 | 2011-11-22 | Simpkins Cuthbert O | Resuscitation fluid |
| RU2406537C2 (ru) * | 2009-02-13 | 2010-12-20 | Государственное учреждение Научно-исследовательский институт биомедицинской химии им. В.Н. Ореховича РАМН | Способ получения эмульсии на основе растительных фосфолипидов |
| CA2756685C (en) * | 2009-04-15 | 2019-12-24 | Tenax Therapeutics, Inc. | Emulsions of perfluorocarbons |
| WO2012003406A2 (en) * | 2010-07-01 | 2012-01-05 | The Board Of Trustees Of The Leland Stanford Junior University | Apparatus and methods to treat or prevent kidney and urologic disease |
| GB2482911A (en) * | 2010-08-20 | 2012-02-22 | Sphere Fluidics Ltd | Microdroplet emulsion system |
| CN103361298A (zh) * | 2012-03-27 | 2013-10-23 | 中国科学院大连化学物理研究所 | 一种适用于猪胰岛的分离提取液及其制备和应用 |
| RU2518313C2 (ru) * | 2012-05-17 | 2014-06-10 | Сергей Иванович Воробьев | Перфторуглеродный кровезаменитель - газотранспортный заменитель донорской крови: состав и средство лечения |
| CN105248412A (zh) * | 2015-10-30 | 2016-01-20 | 暨南大学 | 一种乳化氟碳液在制备肺器官保存液中的应用 |
| RU2696874C2 (ru) * | 2016-11-23 | 2019-08-07 | Федеральное государственное бюджетное учреждение науки Институт теоретической и экспериментальной биофизики Российской академии наук (ИТЭБ РАН) | 1,20-Дибром-3,6,9,12,15,18-гексаоксаперфтор-4,7,10,11,14,17-гексаметилэйкозан в качестве исходного соединения для эмульсий медико-биологического назначения и способ его получения |
| RU2707553C2 (ru) * | 2016-11-23 | 2019-11-28 | Федеральное государственное бюджетное учреждение науки Институт теоретической и экспериментальной биофизики Российской академии наук (ИТЭБ РАН) | α,ω-ДИБРОМПОЛИОКСАПЕРФТОРАЛКАНЫ, СПОСОБ ИХ ПОЛУЧЕНИЯ И ЭМУЛЬСИИ МЕДИКО-БИОЛОГИЧЕСКОГО НАЗНАЧЕНИЯ НА ИХ ОСНОВЕ |
| CN108849861A (zh) * | 2018-09-30 | 2018-11-23 | 南京麦荻泉生物科技有限公司 | 一种含有氟碳乳剂型器官保存液 |
| RU2745290C2 (ru) * | 2019-04-12 | 2021-03-23 | Ирина Николаевна Кузнецова | Эмульсия перфторуглеродных соединений медико-биологического назначения и способ её получения |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3778381A (en) | 1972-04-24 | 1973-12-11 | Allied Chem | Fluorocarbon microemulsions |
| JPS5835485B2 (ja) * | 1976-02-03 | 1983-08-03 | 株式会社ミドリ十字 | 酸素運搬輸液 |
| US4794000A (en) * | 1987-01-08 | 1988-12-27 | Synthetic Blood Corporation | Coacervate-based oral delivery system for medically useful compositions |
| DE3785054T2 (de) * | 1986-01-24 | 1993-07-08 | Childrens Hosp Medical Center | Stabile emulsionen von stark fluorierten, organischen verbindungen. |
| US4866096A (en) | 1987-03-20 | 1989-09-12 | Air Products And Chemicals, Inc. | Stable fluorochemical aqueous emulsions |
| US5171755A (en) * | 1988-04-29 | 1992-12-15 | Hemagen/Pfc | Emulsions of highly fluorinated organic compounds |
| DE4019062A1 (de) * | 1989-08-30 | 1991-03-07 | Kali Chemie Ag | Stabilisierung von perfluorcarbonemulsionen und als emulsionsstabilisierende zusaetze verwendbare perfluorierte heterocyclische verbindungen |
| FR2679150A1 (fr) * | 1991-07-17 | 1993-01-22 | Atta | Preparations comprenant un fluorocarbure ou compose hautement fluore et un compose organique lipophile-fluorophile, et leurs utilisations. |
| AU2441592A (en) * | 1991-08-08 | 1993-03-02 | Leigh D. Segel | Fluorocarbon blood substitute |
| DE4127442C2 (de) * | 1991-08-17 | 1996-08-22 | Udo Dr Gros | Wäßrige Dispersion Fluorcarbon enthaltender Phospholipid-Vesikel und ein Verfahren zu ihrer Herstellung |
| US5344393A (en) * | 1992-02-28 | 1994-09-06 | Alliance Pharmaceutical Corp. | Use of synthetic oxygen carriers to facilitate oxygen delivery |
| US5628930A (en) * | 1992-10-27 | 1997-05-13 | Alliance Pharmaceutical Corp. | Stabilization of fluorocarbon emulsions |
| RU2088217C1 (ru) | 1993-05-07 | 1997-08-27 | Институт биофизики клетки РАН | Эмульсия перфторорганических соединений с газотранспортными свойствами |
| US5733526A (en) * | 1995-12-14 | 1998-03-31 | Alliance Pharmaceutical Corp. | Hydrocarbon oil/fluorochemical preparations and methods of use |
| RU2162692C1 (ru) * | 1999-06-24 | 2001-02-10 | Воробьев Сергей Иванович | Состав на основе эмульсии перфторорганических соединений для медико-биологических целей |
| RU2161122C1 (ru) * | 1999-09-10 | 2000-12-27 | Институт молекулярной генетики РАН | Способ ускорения окисления оксида азота (no) в гетерогенной среде |
| WO2002007717A1 (en) * | 2000-07-20 | 2002-01-31 | Otkrytoe Aktsionernoe Obschestvo Nauchno-Proizvodstvennaya Firma 'perftoran' | Emulsion of perfluororganic compounds for medical purposes, method for producing said emulsion and methods for curing and preventing diseases with the aid of the emulsion |
| RU2200582C2 (ru) * | 2001-04-02 | 2003-03-20 | Воробьев Сергей Иванович | Способ стерилизации перфторуглеродных кровезаменителей и различных сред на основе перфторуглеродных эмульсий |
| RU2199311C2 (ru) | 2001-04-26 | 2003-02-27 | Воробьев Сергей Иванович | Состав перфторуглеродного кровезаменителя на основе эмульсии перфторорганических соединений для медико-биологических целей |
| RU2200544C1 (ru) * | 2001-06-29 | 2003-03-20 | Воробьев Сергей Иванович | Способ получения стерильных перфторуглеродных эмульсий для искусственных перфторуглеродных кровезаменителей |
-
2004
- 2004-03-01 RU RU2004106722/15A patent/RU2259819C1/ru not_active IP Right Cessation
-
2005
- 2005-02-07 JP JP2007501743A patent/JP2007525536A/ja not_active Ceased
- 2005-02-07 EP EP05726945A patent/EP1736148A4/de not_active Withdrawn
- 2005-02-07 CN CN200580013930XA patent/CN101014326B/zh not_active Expired - Fee Related
- 2005-02-07 US US10/591,411 patent/US7842730B2/en not_active Expired - Fee Related
- 2005-02-07 EA EA200601598A patent/EA010315B1/ru not_active IP Right Cessation
- 2005-02-07 WO PCT/RU2005/000058 patent/WO2005089739A1/ru not_active Ceased
- 2005-02-07 UA UAA200610353A patent/UA85220C2/ru unknown
- 2005-02-07 CA CA002557833A patent/CA2557833A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| RU2004106722A (ru) | 2005-08-10 |
| EA010315B1 (ru) | 2008-08-29 |
| US7842730B2 (en) | 2010-11-30 |
| EA200601598A1 (ru) | 2006-12-29 |
| CA2557833A1 (en) | 2005-09-29 |
| CN101014326B (zh) | 2010-09-01 |
| US20070197475A1 (en) | 2007-08-23 |
| CN101014326A (zh) | 2007-08-08 |
| WO2005089739A1 (fr) | 2005-09-29 |
| EP1736148A4 (de) | 2008-04-30 |
| EP1736148A1 (de) | 2006-12-27 |
| JP2007525536A (ja) | 2007-09-06 |
| RU2259819C1 (ru) | 2005-09-10 |
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