UA91733C2 - Способ получения кристаллической формы орлистата - Google Patents
Способ получения кристаллической формы орлистатаInfo
- Publication number
- UA91733C2 UA91733C2 UAA200809715A UAA200809715A UA91733C2 UA 91733 C2 UA91733 C2 UA 91733C2 UA A200809715 A UAA200809715 A UA A200809715A UA A200809715 A UAA200809715 A UA A200809715A UA 91733 C2 UA91733 C2 UA 91733C2
- Authority
- UA
- Ukraine
- Prior art keywords
- orlistat
- crystalline forms
- preparing crystalline
- preparing
- crystalline form
- Prior art date
Links
- AHLBNYSZXLDEJQ-FWEHEUNISA-N orlistat Chemical compound CCCCCCCCCCC[C@H](OC(=O)[C@H](CC(C)C)NC=O)C[C@@H]1OC(=O)[C@H]1CCCCCC AHLBNYSZXLDEJQ-FWEHEUNISA-N 0.000 title abstract 4
- 229960001243 orlistat Drugs 0.000 title abstract 4
- 238000004519 manufacturing process Methods 0.000 title abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/02—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D305/10—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings having one or more double bonds between ring members or between ring members and non-ring members
- C07D305/12—Beta-lactones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Child & Adolescent Psychology (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
Данное изобретение относится к способу получения кристаллических форм орлистата, в частности, орлистата кристаллической формы II, как описано в WO 2005/026140.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP05028489A EP1803714A1 (en) | 2005-12-27 | 2005-12-27 | Process for preparing crystalline forms of orlistat |
| PCT/EP2006/012544 WO2007073937A2 (en) | 2005-12-27 | 2006-12-27 | Process for preparing crystalline forms of orlistat |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA91733C2 true UA91733C2 (ru) | 2010-08-25 |
Family
ID=36354129
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200809715A UA91733C2 (ru) | 2005-12-27 | 2006-12-27 | Способ получения кристаллической формы орлистата |
Country Status (5)
| Country | Link |
|---|---|
| EP (2) | EP1803714A1 (ru) |
| EA (1) | EA015940B1 (ru) |
| NO (1) | NO20083269L (ru) |
| UA (1) | UA91733C2 (ru) |
| WO (1) | WO2007073937A2 (ru) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1803714A1 (en) | 2005-12-27 | 2007-07-04 | KRKA, tovarna zdravil, d.d., Novo mesto | Process for preparing crystalline forms of orlistat |
| PL2002825T3 (pl) * | 2007-06-14 | 2013-12-31 | Krka | Kompozycje farmaceutyczne zawierające orlistat |
| WO2009040827A1 (en) * | 2007-09-24 | 2009-04-02 | Biocon Limited | A process for obtaining tetrahydrolipstatin |
| EP2141236A1 (en) | 2008-07-03 | 2010-01-06 | KRKA, D.D., Novo Mesto | Process for production of lipstatin and microorganisms therefore |
| US20120022274A1 (en) * | 2009-01-22 | 2012-01-26 | Umesh Sannachikkanna | Crystalline Form of Orlistat and a Process Thereof |
| KR102679975B1 (ko) | 2017-07-12 | 2024-06-28 | 메이오 파운데이션 포 메디칼 에쥬케이션 앤드 리써치 | 지방독성 손상을 저감하기 위한 화합물 |
| WO2021072773A1 (zh) * | 2019-10-18 | 2021-04-22 | 山东新时代药业有限公司 | 一种奥利司他胶囊及其制备方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6004996A (en) * | 1997-02-05 | 1999-12-21 | Hoffman-La Roche Inc. | Tetrahydrolipstatin containing compositions |
| EP1028115B1 (en) * | 1999-01-29 | 2002-11-20 | F. Hoffmann-La Roche Ag | Purification of lipstatin |
| CN100423715C (zh) * | 2000-07-28 | 2008-10-08 | 霍夫曼-拉罗奇有限公司 | 新型药物组合物 |
| CA2417607C (en) * | 2000-08-09 | 2008-01-29 | Christine Feinle | Lipase inhibitors for the treatment of dyspepsia |
| IL162323A0 (en) * | 2001-12-04 | 2005-11-20 | Biogal Pharmaceutical Co | Preparation of orlistat and orlistat crystalline forms |
| ES2329474T3 (es) * | 2003-09-12 | 2009-11-26 | Ranbaxy Laboratories Limited | Proceso para la preparacion de formas cristalinas del orlistat. |
| EP1803714A1 (en) | 2005-12-27 | 2007-07-04 | KRKA, tovarna zdravil, d.d., Novo mesto | Process for preparing crystalline forms of orlistat |
-
2005
- 2005-12-27 EP EP05028489A patent/EP1803714A1/en not_active Withdrawn
-
2006
- 2006-12-27 WO PCT/EP2006/012544 patent/WO2007073937A2/en not_active Ceased
- 2006-12-27 UA UAA200809715A patent/UA91733C2/ru unknown
- 2006-12-27 EP EP06841172.7A patent/EP1973893B1/en not_active Revoked
- 2006-12-27 EA EA200801573A patent/EA015940B1/ru not_active IP Right Cessation
-
2008
- 2008-07-23 NO NO20083269A patent/NO20083269L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007073937A3 (en) | 2007-08-23 |
| EP1973893A2 (en) | 2008-10-01 |
| EA200801573A1 (ru) | 2008-10-30 |
| EP1973893B1 (en) | 2015-04-29 |
| WO2007073937A2 (en) | 2007-07-05 |
| EP1803714A1 (en) | 2007-07-04 |
| NO20083269L (no) | 2008-09-19 |
| EA015940B1 (ru) | 2011-12-30 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| MX2010002836A (es) | Bortezomib y proceso para la produccion del mismo. | |
| IL187586A0 (en) | Method for producing dihydroquinazolines | |
| TW200722079A (en) | Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein | |
| MY150538A (en) | Process for the manufacture of dihydropteridinones | |
| WO2009039307A3 (en) | Hydrogels and methods for producing and using the same | |
| WO2006136357A3 (de) | Kristalline modifikationen des pyraclostrobins | |
| MY147732A (en) | Process for the preparation of 2-substituted-5- (1-alkylthio) alkylpyridines | |
| TW200720232A (en) | Crystalline solid forms of tigecycline and methods of preparing same | |
| EP1908749A4 (en) | PROCESS FOR PREPARING ISOCYANATE, ISOCYANATE MADE ACCORDING TO IT AND USE OF ISOCYANATE | |
| UA89390C2 (ru) | Способ получения аннелированных производных пиперазин-2-она та соответствующие промежуточные продукты | |
| TW200617019A (en) | A process for the preparation of 7α-alkylated 19-norsteroids | |
| MX2007011668A (es) | Mezclas de caucho de silicona de reticulacion por adicion autoadhesivas, metodo para la produccion de las mismas, metodo para producir partes moldeadas compuestas y uso de las mismas. | |
| MY158910A (en) | Surface modified silicic acid semi-gels | |
| IL180551A0 (en) | Use of substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines in the treatment of nausea and vomiting | |
| EG25069A (en) | Process for urea production and related plant. | |
| MX2009008422A (es) | Proceso para la preparacion de alquilpiridinas de 5-(1-alquiltio)2-sustituidas. | |
| TW200732410A (en) | Sprayable acoustic compositions | |
| WO2007141593A3 (en) | Process for the preparation of metoprolol and its salts | |
| NO20083269L (no) | Prosess for a anvende krystallinsk orlistatmetoder | |
| MX2007010143A (es) | Formas cristalinas de intermedio de linezolid. | |
| EG24992A (en) | Process for urea production and related plant. | |
| EG25292A (en) | Process for the production of anilines. | |
| TW200730521A (en) | Triazine compounds having amino-and carboxyl-containing substituents | |
| MY146610A (en) | Process of producing bleach boosters | |
| TW200637832A (en) | Process for preparing amorphous valsartan |