UA93355C2 - Композиция субероиланилид-гидроксаминовой кислоты и способы ee получения - Google Patents
Композиция субероиланилид-гидроксаминовой кислоты и способы ee полученияInfo
- Publication number
- UA93355C2 UA93355C2 UAA200701731A UAA200701731A UA93355C2 UA 93355 C2 UA93355 C2 UA 93355C2 UA A200701731 A UAA200701731 A UA A200701731A UA A200701731 A UAA200701731 A UA A200701731A UA 93355 C2 UA93355 C2 UA 93355C2
- Authority
- UA
- Ukraine
- Prior art keywords
- hydroxamic acid
- suberoylanilide hydroxamic
- formulation
- producing same
- present
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 4
- WAEXFXRVDQXREF-UHFFFAOYSA-N vorinostat Chemical compound ONC(=O)CCCCCCC(=O)NC1=CC=CC=C1 WAEXFXRVDQXREF-UHFFFAOYSA-N 0.000 title abstract 2
- 229960000237 vorinostat Drugs 0.000 title abstract 2
- 238000009472 formulation Methods 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 239000004480 active ingredient Substances 0.000 abstract 1
- 238000004090 dissolution Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000002245 particle Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Данное изобретение касается фармацевтической композиции с конкретным профилем растворимости, которая в качестве активного ингредиента содержит субероиланилид-гидроксаминовую кислоту с конкретным распределением размеров частичек. Данное изобретение также касается способа получения указанной фармацевтической композиции.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US68287505P | 2005-05-20 | 2005-05-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA93355C2 true UA93355C2 (ru) | 2011-02-10 |
Family
ID=37946173
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200701731A UA93355C2 (ru) | 2005-05-20 | 2006-05-16 | Композиция субероиланилид-гидроксаминовой кислоты и способы ee получения |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP2229941A1 (ru) |
| CN (1) | CN101080223B (ru) |
| AR (1) | AR095159A2 (ru) |
| NO (1) | NO20070952L (ru) |
| RU (1) | RU2354362C2 (ru) |
| UA (1) | UA93355C2 (ru) |
| ZA (1) | ZA200700636B (ru) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8883851B2 (en) | 2008-10-15 | 2014-11-11 | Generics [Uk] Limited | Process for the preparation of vorinostat |
| JP2012509929A (ja) * | 2008-11-26 | 2012-04-26 | ジェネリクス・(ユーケー)・リミテッド | 多型 |
| CN102344392B (zh) * | 2010-08-03 | 2015-05-27 | 杭州容立医药科技有限公司 | 一种蛋白脱乙酰酶抑制剂伏立诺他的精制方法 |
| CN102643214B (zh) * | 2011-02-21 | 2016-08-03 | 杭州容立医药科技有限公司 | 伏立诺他ⅰ晶形大晶粒的制备方法及制剂 |
| CN103159646B (zh) * | 2013-03-19 | 2014-10-22 | 广东药学院 | 一种异羟肟酸类化合物及其制备方法和应用 |
| CN107362148B (zh) * | 2017-07-27 | 2020-04-21 | 东曜药业有限公司 | 一种治疗肿瘤的药物组合物及其制备方法和应用 |
| CN108929246B (zh) * | 2018-07-09 | 2021-07-02 | 湖南中医药大学 | 一种固态法制备羟肟酸类衍生物的方法 |
| CN110283102B (zh) * | 2019-05-31 | 2022-09-27 | 宿州亿帆药业有限公司 | 一种伏林司他ⅰ晶型的制备方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4522811A (en) | 1982-07-08 | 1985-06-11 | Syntex (U.S.A.) Inc. | Serial injection of muramyldipeptides and liposomes enhances the anti-infective activity of muramyldipeptides |
| CN101259120B (zh) * | 2002-03-04 | 2012-07-04 | Hdac默克研究有限责任公司 | 辛二酰苯胺异羟肟酸或其可药用盐在制备诱导末期分化的药物的用途 |
| US7456219B2 (en) * | 2002-03-04 | 2008-11-25 | Merck Hdac Research, Llc | Polymorphs of suberoylanilide hydroxamic acid |
-
2006
- 2006-05-16 EP EP10155706A patent/EP2229941A1/en not_active Withdrawn
- 2006-05-16 RU RU2007106072/15A patent/RU2354362C2/ru active Protection Beyond IP Right Term
- 2006-05-16 UA UAA200701731A patent/UA93355C2/ru unknown
- 2006-05-16 CN CN200680000867.0A patent/CN101080223B/zh active Active
-
2007
- 2007-01-23 ZA ZA200700636A patent/ZA200700636B/xx unknown
- 2007-02-20 NO NO20070952A patent/NO20070952L/no not_active Application Discontinuation
-
2014
- 2014-02-05 AR ARP140100385A patent/AR095159A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AR095159A2 (es) | 2015-09-30 |
| ZA200700636B (en) | 2008-10-29 |
| CN101080223B (zh) | 2015-02-11 |
| EP2229941A1 (en) | 2010-09-22 |
| RU2007106072A (ru) | 2008-08-27 |
| RU2354362C2 (ru) | 2009-05-10 |
| NO20070952L (no) | 2007-03-20 |
| CN101080223A (zh) | 2007-11-28 |
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