UA93530C2 - Композиция c пролонгированным высвобождением активного вещества, способ ee получения и применения - Google Patents
Композиция c пролонгированным высвобождением активного вещества, способ ee получения и примененияInfo
- Publication number
- UA93530C2 UA93530C2 UAA200808585A UAA200808585A UA93530C2 UA 93530 C2 UA93530 C2 UA 93530C2 UA A200808585 A UAA200808585 A UA A200808585A UA A200808585 A UAA200808585 A UA A200808585A UA 93530 C2 UA93530 C2 UA 93530C2
- Authority
- UA
- Ukraine
- Prior art keywords
- active ingredient
- composition
- sustained release
- preparation
- esters
- Prior art date
Links
- 239000004480 active ingredient Substances 0.000 title abstract 3
- 239000000203 mixture Substances 0.000 title abstract 3
- 238000013268 sustained release Methods 0.000 title abstract 2
- 239000012730 sustained-release form Substances 0.000 title abstract 2
- 238000000034 method Methods 0.000 title 1
- SMZOUWXMTYCWNB-UHFFFAOYSA-N 2-(2-methoxy-5-methylphenyl)ethanamine Chemical compound COC1=CC=C(C)C=C1CCN SMZOUWXMTYCWNB-UHFFFAOYSA-N 0.000 abstract 2
- NIXOWILDQLNWCW-UHFFFAOYSA-N 2-Propenoic acid Natural products OC(=O)C=C NIXOWILDQLNWCW-UHFFFAOYSA-N 0.000 abstract 2
- CERQOIWHTDAKMF-UHFFFAOYSA-N Methacrylic acid Chemical compound CC(=C)C(O)=O CERQOIWHTDAKMF-UHFFFAOYSA-N 0.000 abstract 2
- 239000007931 coated granule Substances 0.000 abstract 2
- 238000000576 coating method Methods 0.000 abstract 2
- 229920001577 copolymer Polymers 0.000 abstract 2
- 150000002148 esters Chemical class 0.000 abstract 2
- 125000001453 quaternary ammonium group Chemical group 0.000 abstract 2
- 239000002417 nutraceutical Substances 0.000 abstract 1
- 235000021436 nutraceutical agent Nutrition 0.000 abstract 1
- 239000002245 particle Substances 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/28—Compounds containing heavy metals
- A61K31/285—Arsenic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
- A61K33/24—Heavy metals; Compounds thereof
- A61K33/26—Iron; Compounds thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Inorganic Chemistry (AREA)
- Hematology (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Zoology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Фармацевтическая, нутрицевтическая или ветеринарная композиция, которая содержит, по меньшей мере, одну гранулу, покрытую оболочкой, с пролонгированным высвобождением активного вещества, причем указанная гранула, покрытая оболочкой, состоит из частицы, содержащей указанное активное вещество, покрытое, по меньшей мере, двумя оболочками, содержащими комбинацию эксципиентов, которая состоит из, по меньшей мере, одного сополимера (а) сложных эфиров акриловой кислоты и метакриловой кислоты, в котором молярное содержание групп четвертичного аммония ниже или равно 8 %, в ассоциации со вторым сополимером (b) сложных эфиров акриловой кислоты и метакриловой кислоты, в котором молярное содержание групп четвертичного аммония выше 8 %, в массовом соотношении (а)/(b), который составляет от 60/40 до 80/20, и при
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0512189A FR2894143B1 (fr) | 2005-12-01 | 2005-12-01 | Composition a liberation prolongee de l'actif, son procede de preparation et son utilisation. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA93530C2 true UA93530C2 (ru) | 2011-02-25 |
Family
ID=36968738
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200808585A UA93530C2 (ru) | 2005-12-01 | 2006-11-23 | Композиция c пролонгированным высвобождением активного вещества, способ ee получения и применения |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US8834923B2 (ru) |
| EP (1) | EP1954251B1 (ru) |
| JP (1) | JP5674275B2 (ru) |
| KR (1) | KR101332744B1 (ru) |
| CN (1) | CN101321520A (ru) |
| AR (1) | AR057212A1 (ru) |
| AT (1) | ATE548030T1 (ru) |
| AU (1) | AU2006319077B2 (ru) |
| BR (1) | BRPI0619774B1 (ru) |
| CA (1) | CA2632547C (ru) |
| DK (1) | DK1954251T3 (ru) |
| ES (1) | ES2383760T3 (ru) |
| FR (1) | FR2894143B1 (ru) |
| IL (1) | IL191758A (ru) |
| MA (1) | MA29770B1 (ru) |
| NO (1) | NO339720B1 (ru) |
| NZ (1) | NZ566783A (ru) |
| PL (1) | PL1954251T3 (ru) |
| PT (1) | PT1954251E (ru) |
| RS (1) | RS52308B (ru) |
| RU (1) | RU2414211C2 (ru) |
| SI (1) | SI1954251T1 (ru) |
| TN (1) | TNSN08152A1 (ru) |
| TW (1) | TWI374035B (ru) |
| UA (1) | UA93530C2 (ru) |
| WO (1) | WO2007063200A1 (ru) |
| ZA (1) | ZA200801896B (ru) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0613583D0 (en) * | 2006-07-05 | 2006-08-16 | Sericol Ltd | A printing ink |
| CN101912049A (zh) * | 2010-07-27 | 2010-12-15 | 广州市正百饲料科技有限公司 | 包被微量元素预混料及其制备方法 |
| CN103191078B (zh) * | 2012-01-06 | 2018-01-09 | 常州善美药物研究开发中心有限公司 | 一种双膜多药层的高溶解度盐类药物控释片 |
| NL2014348B1 (en) | 2015-02-25 | 2016-10-13 | Univ Delft Tech | Controlled release from particles encapsulated by molecular layer deposition. |
| RU2702690C2 (ru) * | 2015-08-13 | 2019-10-09 | БИОЛИНГУС АйПи ЛЛСи | Способ получения продуктов, содержащих стабилизированные активные вещества, и композиций, содержащих таковые |
| RU2616264C1 (ru) * | 2016-03-28 | 2017-04-13 | Санкт-Петербургское Государственное бюджетное учреждение здравоохранения "Родильный дом N 10" | Способ профилактики железодефицитной анемии у несовершеннолетних беременных женщин |
| RU2623071C1 (ru) * | 2016-09-29 | 2017-06-21 | федеральное государственное бюджетное образовательное учреждение высшего образования "Ставропольский государственный аграрный университет" | Лечебно-профилактический хелатный железосодержащий препарат для сельскохозяйственных животных |
| CN106344534B (zh) * | 2016-09-30 | 2019-07-19 | 广西科技大学 | 硫酸亚铁肠溶滴丸的制备方法 |
| US20200275685A1 (en) * | 2017-11-14 | 2020-09-03 | PIZETA PHARMA S.p.A. | Oral administration form comprising an iron-copper mixture and its use as a food supplement |
| CN109999058A (zh) * | 2019-05-22 | 2019-07-12 | 江阴天江药业有限公司 | 一种胶类中药的烊化方法和产品,以及由该产品制得的固体饮料及其制备方法 |
| WO2024006539A1 (en) * | 2022-07-01 | 2024-01-04 | Vitakey Inc. | Nutraceutical particles |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3622487A1 (de) * | 1986-07-02 | 1988-01-14 | Schering Ag | Arzneimittel mit verzoegerter wirkstoffabgabe |
| IE82916B1 (en) * | 1990-11-02 | 2003-06-11 | Elan Corp Plc | Formulations and their use in the treatment of neurological diseases |
| US5286493A (en) * | 1992-01-27 | 1994-02-15 | Euroceltique, S.A. | Stabilized controlled release formulations having acrylic polymer coating |
| US5478577A (en) * | 1993-11-23 | 1995-12-26 | Euroceltique, S.A. | Method of treating pain by administering 24 hour oral opioid formulations exhibiting rapid rate of initial rise of plasma drug level |
| DE4332394A1 (de) * | 1993-09-23 | 1995-03-30 | Falk Pharma Gmbh | Budesonid-Pellets mit kontrolliertem Freigabeprofil und Verfahren zu ihrer Herstellung |
| FR2792527B1 (fr) * | 1999-04-22 | 2004-08-13 | Ethypharm Lab Prod Ethiques | Microgranules de ketoprofene, procede de preparation et compositions pharmaceutiques |
| ES2226886T3 (es) * | 1999-08-31 | 2005-04-01 | Grunenthal Gmbh | Forma de administracion de accion retardada que contiene sacarinato de tramadol. |
| DE50008261D1 (de) * | 1999-08-31 | 2004-11-18 | Gruenenthal Gmbh | Retardierte darreichungsform enthaltend tramadolsaccharinat |
| JP2003508420A (ja) * | 1999-09-02 | 2003-03-04 | ノストラム・ファーマスーティカルズ・インコーポレイテッド | 経口投与に適した、制御された放出の経口用量 |
| WO2001045668A2 (en) | 1999-12-20 | 2001-06-28 | Schering Corporation | Stable extended release oral dosage composition comprising pseudoephedrine and desloratadine |
| DE10013029A1 (de) * | 2000-03-17 | 2001-09-20 | Roehm Gmbh | Mehrschichtige Arzneiform für die Colonfreigabe |
| US7070803B2 (en) * | 2000-03-31 | 2006-07-04 | Nycomed Austria Gmbh | Controlled release pharmaceutical composition for oral use containing midodrine and/or active metabolite, desglymidodrine |
| AR030557A1 (es) * | 2000-04-14 | 2003-08-27 | Jagotec Ag | Una tableta en multicapa de liberacion controlada y metodo de tratamiento |
| KR100477874B1 (ko) | 2001-04-10 | 2005-03-22 | 곽해수 | 지방산에스터를 이용한 수용성 철분 미세캡슐 |
| WO2003020241A2 (en) * | 2001-09-05 | 2003-03-13 | Vectura Limited | Functional powders for oral delivery |
| EP1474123A1 (en) | 2002-01-03 | 2004-11-10 | LEK Pharmaceuticals D.D. | Controlled release pharmaceutical formulation containing venlafaxine |
| US20030190355A1 (en) * | 2002-04-05 | 2003-10-09 | Hermelin Marc S. | Modified release minerals |
| DE60335426D1 (de) * | 2002-08-15 | 2011-01-27 | Euro Celtique Sa | Pharmazeutische Zusammensetzungen enthaltend einen Opioidantagonisten |
| US6562378B1 (en) * | 2002-08-16 | 2003-05-13 | Tsar Health Private Ltd. | Nutritional supplement for adolescents |
| WO2005020993A1 (en) * | 2003-08-29 | 2005-03-10 | Lifecycle Pharma A/S | Modified release compositions comprising tacrolimus |
-
2005
- 2005-12-01 FR FR0512189A patent/FR2894143B1/fr not_active Expired - Lifetime
-
2006
- 2006-11-23 US US12/085,501 patent/US8834923B2/en active Active
- 2006-11-23 RS RS20120229A patent/RS52308B/sr unknown
- 2006-11-23 JP JP2008542790A patent/JP5674275B2/ja active Active
- 2006-11-23 UA UAA200808585A patent/UA93530C2/ru unknown
- 2006-11-23 RU RU2008126728/15A patent/RU2414211C2/ru active
- 2006-11-23 CN CNA2006800453522A patent/CN101321520A/zh active Pending
- 2006-11-23 DK DK06831163.8T patent/DK1954251T3/da active
- 2006-11-23 SI SI200631341T patent/SI1954251T1/sl unknown
- 2006-11-23 CA CA2632547A patent/CA2632547C/fr active Active
- 2006-11-23 EP EP06831163A patent/EP1954251B1/fr active Active
- 2006-11-23 PT PT06831163T patent/PT1954251E/pt unknown
- 2006-11-23 PL PL06831163T patent/PL1954251T3/pl unknown
- 2006-11-23 KR KR1020087008548A patent/KR101332744B1/ko active Active
- 2006-11-23 ES ES06831163T patent/ES2383760T3/es active Active
- 2006-11-23 NZ NZ566783A patent/NZ566783A/en unknown
- 2006-11-23 BR BRPI0619774-4A patent/BRPI0619774B1/pt active IP Right Grant
- 2006-11-23 AT AT06831163T patent/ATE548030T1/de active
- 2006-11-23 AU AU2006319077A patent/AU2006319077B2/en active Active
- 2006-11-23 WO PCT/FR2006/002577 patent/WO2007063200A1/fr not_active Ceased
- 2006-11-30 TW TW095144284A patent/TWI374035B/zh active
- 2006-12-01 AR ARP060105306A patent/AR057212A1/es not_active Application Discontinuation
-
2008
- 2008-02-28 ZA ZA200801896A patent/ZA200801896B/xx unknown
- 2008-03-07 MA MA30732A patent/MA29770B1/fr unknown
- 2008-04-02 TN TNP2008000152A patent/TNSN08152A1/fr unknown
- 2008-04-29 NO NO20082047A patent/NO339720B1/no unknown
- 2008-05-27 IL IL191758A patent/IL191758A/en active IP Right Grant
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| WO2007006353A3 (de) | Verwendung eines teilneutralisierten, anionischen (meth) acrylat-copolymers als uberzug fur die herstellung einer arzneiform mit einer wirkstofffreisetzung bei erniedrigten ph-werten | |
| IL195407A0 (en) | Pharmaceutical composition with controlled active ingredient delivery for active ingredients with good solubility in water | |
| NO20080202L (no) | Nanopartikulaere clopidogrel og aspirin kombinasjonsformuleringer | |
| DE50107641D1 (de) | Überzugs- und bindemittel für arzneimittelformulierungen mit verbesserter lagerstabilität | |
| WO2006017852A3 (en) | Pharmaceutical compositions for controlled release delivery of biologically active compounds | |
| UA106877C2 (ru) | Фармацевтическая композиция энтакапона или его солей с пролонгированным высвобождением | |
| WO2000019984A3 (de) | Überzogene arzneiformen mit kontrollierter wirkstoffabgabe | |
| MX356579B (es) | Composicion farmaceutica o nutraceutica de resistencia gastrica con resistencia contra la influenza de etanol. | |
| UA93530C2 (ru) | Композиция c пролонгированным высвобождением активного вещества, способ ee получения и применения | |
| NZ595061A (en) | Formulation comprising avermectin particles coated with a photo - protecting agent | |
| WO2010065289A3 (en) | Medical adhesive compositions | |
| NZ589017A (en) | Solid pharmaceutical formulation with delayed release | |
| WO2012085043A3 (en) | Rapidly disintegrating, solid coated dosage form | |
| BRPI0620185B8 (pt) | formulação farmacêutica, comprimidos, e, processo para a preparação de uma formulação farmacêutica | |
| WO2011056785A3 (en) | Microcrystalline cellulose and calcium phosphate compositions useful as pharmaceutical excipients | |
| MX2015010449A (es) | Composicion farmaceutica multiparticulada que comprende una multitud de dos clases de granulos. | |
| MX2010007579A (es) | Preparacion nutriceutica o farmaceutica revestida con una liberacion de sustancia activa de impulsion mejorada. | |
| IL174830A0 (en) | Pellets containing venlafaxine hydrochloride, pharmaceutical compositions comprising them and processes for their preparation | |
| TW200635963A (en) | Partially neutralized anionic (meth)acrylate copolymer | |
| MX2010007578A (es) | Preparacion nutriceutica o farmaceutica revestida con una liberacion acelerada controlada de sustancia activa. | |
| NO20044926L (no) | Kopolymer, fremgangsmate for fremstilling og anvendelse som film ved belegging av farmasoytiske formuleringer. | |
| WO2007145993A3 (en) | Modified compositions and methods for enhancing brain function | |
| PT1815850E (pt) | Formulação de libertação controlada de ácido divalpróico e seus derivados | |
| MX2024000522A (es) | Composicion que comprende un copolimero de (met)acrilato, una sal alcalina o de amonio de un acido monocarboxilico alifatico saturado y deslizantes especificos. | |
| WO2006064321A3 (en) | Controlled release compositions of divalproex sodium |