UA95239C2 - Макроциклические ингибиторы вируса гепатита с - Google Patents

Макроциклические ингибиторы вируса гепатита с

Info

Publication number: UA95239C2
Authority: UA; Ukraine
Prior art keywords: inhibitors; hepatitis; virus; hcv; formula
Prior art date: 2005-07-29

Application number

UAA200714714A

Other languages

English (en)

Ukrainian (uk)

Inventor

Кок Герман Августинус Де

Пьер Жан-Мари Бернар Рабуассон

Кеннет Алан Симмен

Матс Стефан Линдстром

Пиа Сесилия Канберг

Дмитрий Антонов

Карл Магнус Нилссон

Бенгт Бертил Самуэльссон

Эса Анника Кристина Розенквист

Original Assignee

Тиботек Фармасьютикелз Лтд.

Медивир Аб

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-07-29

Filing date

2006-07-28

Publication date

2011-07-25

2006-07-28 Application filed by Тиботек Фармасьютикелз Лтд., Медивир Аб filed Critical Тиботек Фармасьютикелз Лтд.

2011-07-25 Publication of UA95239C2 publication Critical patent/UA95239C2/ru

Links

239000003112 inhibitor Substances 0.000 title abstract 3
241000711549 Hepacivirus C Species 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
NCDNCNXCDXHOMX-UHFFFAOYSA-N Ritonavir Natural products C=1C=CC=CC=1CC(NC(=O)OCC=1SC=NC=1)C(O)CC(CC=1C=CC=CC=1)NC(=O)C(C(C)C)NC(=O)N(C)CC1=CSC(C(C)C)=N1 NCDNCNXCDXHOMX-UHFFFAOYSA-N 0.000 abstract 1
125000004429 atom Chemical group 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
NCDNCNXCDXHOMX-XGKFQTDJSA-N ritonavir Chemical compound N([C@@H](C(C)C)C(=O)N[C@H](C[C@H](O)[C@H](CC=1C=CC=CC=1)NC(=O)OCC=1SC=NC=1)CC=1C=CC=CC=1)C(=O)N(C)CC1=CSC(C(C)C)=N1 NCDNCNXCDXHOMX-XGKFQTDJSA-N 0.000 abstract 1
229960000311 ritonavir Drugs 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Medicinal Chemistry (AREA)
Molecular Biology (AREA)
Virology (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

UAA200714714A 2005-07-29 2006-07-28 Макроциклические ингибиторы вируса гепатита с UA95239C2 (ru)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP05107066		2005-07-29

Publications (1)

Publication Number	Publication Date
UA95239C2 true UA95239C2 (ru)	2011-07-25

Family

ID=35601774

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
UAA200714714A UA95239C2 (ru)	2005-07-29	2006-07-28	Макроциклические ингибиторы вируса гепатита с

Country Status (4)

Country	Link
AP (1)	AP2387A (ru)
ES (1)	ES2360417T3 (ru)
UA (1)	UA95239C2 (ru)
ZA (1)	ZA200800856B (ru)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
UA74546C2 (en) *	1999-04-06	2006-01-16	Boehringer Ingelheim Ca Ltd	Macrocyclic peptides having activity relative to hepatitis c virus, a pharmaceutical composition and use of the pharmaceutical composition
ES2336009T3 (es) *	2004-01-30	2010-04-07	Medivir Ab	Inhibidores de la ns-3 serina proteasa del vhc.

2006
- 2006-07-28 UA UAA200714714A patent/UA95239C2/ru unknown
- 2006-07-28 ES ES06764263T patent/ES2360417T3/es not_active Expired - Lifetime
- 2006-07-28 AP AP2008004304A patent/AP2387A/xx active
2008
- 2008-01-28 ZA ZA200800856A patent/ZA200800856B/xx unknown

Also Published As

Publication number	Publication date
ZA200800856B (en)	2009-06-24
AP2387A (en)	2012-03-26
ES2360417T3 (es)	2011-06-03

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