US12581252B2 - Substituted pyrrolo[3,4-b]pyridines as PI3K-α inhibitors - Google Patents

Substituted pyrrolo[3,4-b]pyridines as PI3K-α inhibitors

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Publication number
US12581252B2
US12581252B2 US17/921,580 US202117921580A US12581252B2 US 12581252 B2 US12581252 B2 US 12581252B2 US 202117921580 A US202117921580 A US 202117921580A US 12581252 B2 US12581252 B2 US 12581252B2
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Prior art keywords
independently selected
substituted
partially unsaturated
nitrogen
oxygen
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US17/921,580
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US20240287058A1 (en
Inventor
Alessandro Boezio
Lucian V. DiPietro
Hakan Gunaydin
Thomas H. McLean
Levi Charles Thomas Pierce
Fabrizio Giordanetto
Yakov PECHERSKY
Megan BERTRAND-LAPERLE
Alexandre LARIVEE
Kashif Tanveer
Michael Paul Deninno
Tarek MOHAMED
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DE Shaw Research LLC
Relay Therapeutics Inc
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DE Shaw Research LLC
Relay Therapeutics Inc
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Priority to US17/921,580 priority Critical patent/US12581252B2/en
Priority to US18/208,023 priority patent/US12219327B2/en
Publication of US20240287058A1 publication Critical patent/US20240287058A1/en
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Publication of US12581252B2 publication Critical patent/US12581252B2/en
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