UY33100A - Derivados de 9h-beta-carbolina (o 9h-piridino (3,4-b) indol) trisustituidos, su preparacion y su utilizacion terapeutica - Google Patents

Derivados de 9h-beta-carbolina (o 9h-piridino (3,4-b) indol) trisustituidos, su preparacion y su utilizacion terapeutica

Info

Publication number
UY33100A
UY33100A UY33100A UY33100A UY33100A UY 33100 A UY33100 A UY 33100A UY 33100 A UY33100 A UY 33100A UY 33100 A UY33100 A UY 33100A UY 33100 A UY33100 A UY 33100A
Authority
UY
Uruguay
Prior art keywords
trisustituidos
carbolina
indol
pyridine
beta
Prior art date
Application number
UY33100A
Other languages
English (en)
Inventor
Didier Babin
Olivier Bedel
Thierry Gouyon
Serge Mignani
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of UY33100A publication Critical patent/UY33100A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
UY33100A 2009-12-10 2010-12-10 Derivados de 9h-beta-carbolina (o 9h-piridino (3,4-b) indol) trisustituidos, su preparacion y su utilizacion terapeutica UY33100A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0958831A FR2953838B1 (fr) 2009-12-10 2009-12-10 Derives de 9h-beta-carboline (ou 9h-pyridino[3,4-b]indole) trisubstitues, leur preparation et leur utilisation therapeutique

Publications (1)

Publication Number Publication Date
UY33100A true UY33100A (es) 2011-07-29

Family

ID=42062314

Family Applications (1)

Application Number Title Priority Date Filing Date
UY33100A UY33100A (es) 2009-12-10 2010-12-10 Derivados de 9h-beta-carbolina (o 9h-piridino (3,4-b) indol) trisustituidos, su preparacion y su utilizacion terapeutica

Country Status (5)

Country Link
AR (1) AR079613A1 (es)
FR (1) FR2953838B1 (es)
TW (1) TW201124414A (es)
UY (1) UY33100A (es)
WO (1) WO2011070299A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105330665B (zh) * 2015-11-04 2017-10-03 衡阳师范学院 一种抑制激肽释放酶klk7的化合物、制备方法和用途
US11485734B2 (en) 2018-10-02 2022-11-01 Northwestern University Beta-carbolines as positive allosteric modulators of the human serotonin receptor 2C (5-HT2C)
US12129265B2 (en) 2020-07-21 2024-10-29 Ankh Life Sciences Limited Therapeutic agents and uses thereof

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57123180A (en) * 1980-12-17 1982-07-31 Schering Ag 3-substituted beta-carboline, manufacture and psychotropic drug containing same
DK240084D0 (da) * 1984-05-15 1984-05-15 Ferrosan As New beta-carboline-3-oxadiazolyl derivatives
DE3540653A1 (de) * 1985-11-13 1987-05-14 Schering Ag Neue 3-oxadiazol- und 3-carbonsaeure-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel
DE3608089A1 (de) * 1986-03-08 1987-09-10 Schering Ag Heteroaryl-oxy-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel
AU619203B2 (en) * 1987-08-28 1992-01-23 Schering Aktiengesellschaft Isoxazole-beta-carboline derivatives
WO1996034865A1 (en) * 1995-05-05 1996-11-07 Novo Nordisk A/S Novel heterocyclic chemistry
JP2002542246A (ja) * 1999-04-20 2002-12-10 ノボ ノルディスク アクティーゼルスカブ 新規な化合物、それらの製造及び使用
US6492406B1 (en) * 1999-05-21 2002-12-10 Astrazeneca Ab Pharmaceutically active compounds
EP1209158A1 (en) * 2000-11-18 2002-05-29 Aventis Pharma Deutschland GmbH Substituted beta-carbolines
DE60217532T8 (de) * 2001-11-07 2008-02-07 Millennium Pharmaceuticals, Inc., Cambridge Carboline derivate als ikb-inhibitoren zur behandlung des m ultiplen myelomas
FR2869540B1 (fr) * 2004-04-30 2008-05-16 Centre Nat Rech Scient Cnrse Compositions pharmaceutiques contenant des derives de b-carboline, et leur utilisation pour le traitement des cancers
US8119655B2 (en) * 2005-10-07 2012-02-21 Takeda Pharmaceutical Company Limited Kinase inhibitors
EP2137184B1 (en) * 2007-04-03 2013-05-08 Array Biopharma, Inc. Imidazo[1,2-a]pyridine compounds as receptor tyrosine kinase inhibitors
GB0723815D0 (en) * 2007-12-05 2008-01-16 Glaxo Group Ltd Compounds
AR072084A1 (es) * 2008-06-12 2010-08-04 Sanofi Aventis Derivados de azacarbolinas, su preparacion y su utilizacion terapeutica como inhibidores de las quinasas pim

Also Published As

Publication number Publication date
TW201124414A (en) 2011-07-16
FR2953838B1 (fr) 2012-02-24
WO2011070299A1 (fr) 2011-06-16
FR2953838A1 (fr) 2011-06-17
AR079613A1 (es) 2012-02-08

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20181127