WO2007132134A3 - Compositions comprenant au moins un dérivé de l'acide naphtoïque et du péroxyde de benzoyle, leurs procédés de préparation, et leurs utilisations - Google Patents
Compositions comprenant au moins un dérivé de l'acide naphtoïque et du péroxyde de benzoyle, leurs procédés de préparation, et leurs utilisations Download PDFInfo
- Publication number
- WO2007132134A3 WO2007132134A3 PCT/FR2007/051296 FR2007051296W WO2007132134A3 WO 2007132134 A3 WO2007132134 A3 WO 2007132134A3 FR 2007051296 W FR2007051296 W FR 2007051296W WO 2007132134 A3 WO2007132134 A3 WO 2007132134A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- acid derivative
- benzoyl peroxide
- naphthoic acid
- compositions
- methods
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/20—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Cosmetics (AREA)
Abstract
L'invention concerne une composition pour application topique 5 comprenant, dans un milieu physiologiquement acceptable, au moins un dérivé de l'acide naphtoïque et du peroxyde de benzoyle sous forme encapsulée. L'invention s'applique en particulier en pharmacie humaine ou en cosmétique.
Priority Applications (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07766070A EP2019663A2 (fr) | 2006-05-17 | 2007-05-16 | Compositions comprenant au moins un dérivé de l'acide naphtoïque et du péroxyde de benzoyle, leurs procédés de préparation, et leurs utilisations |
| CA002649124A CA2649124A1 (fr) | 2006-05-17 | 2007-05-16 | Compositions comprenant au moins un derive de l'acide naphtoique et du peroxyde de benzoyle, leurs procedes de preparation, et leurs utilisations |
| US12/272,061 US20090191245A1 (en) | 2006-05-17 | 2008-11-17 | Reduced-irritant dermatological compositions comprising at least one naphthoic acid compound and benzoyl peroxide and treatment of keratinization disorders therewith |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0604407A FR2901139B1 (fr) | 2006-05-17 | 2006-05-17 | Compositions comprenant au moins un derive de l'acide naphtoique et du peroxyde de benzoyle, leurs procedes de preparation, et leurs utilisations |
| FR0604407 | 2006-05-17 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| US12/272,061 Continuation US20090191245A1 (en) | 2006-05-17 | 2008-11-17 | Reduced-irritant dermatological compositions comprising at least one naphthoic acid compound and benzoyl peroxide and treatment of keratinization disorders therewith |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| WO2007132134A2 WO2007132134A2 (fr) | 2007-11-22 |
| WO2007132134A3 true WO2007132134A3 (fr) | 2008-01-10 |
Family
ID=37561252
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PCT/FR2007/051296 Ceased WO2007132134A2 (fr) | 2006-05-17 | 2007-05-16 | Compositions comprenant au moins un dérivé de l'acide naphtoïque et du péroxyde de benzoyle, leurs procédés de préparation, et leurs utilisations |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20090191245A1 (fr) |
| EP (1) | EP2019663A2 (fr) |
| CA (1) | CA2649124A1 (fr) |
| FR (1) | FR2901139B1 (fr) |
| WO (1) | WO2007132134A2 (fr) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8936800B2 (en) | 2001-12-21 | 2015-01-20 | Galderma Research & Development | Gel composition for treatment of common acne comprising a combination of benzoyl peroxide and adapalene and/or adapalene salt |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2903603B1 (fr) * | 2006-07-13 | 2009-03-20 | Galderma Res & Dev S N C Snc | Combinaison d'adapalene et de peroxyde de benzole dans le traitement de l'acne |
| US8080537B2 (en) | 2006-07-13 | 2011-12-20 | Galderma Research & Development | Combinations of adapalene and benzoyl peroxide for treating acne lesions |
| FR2910320B1 (fr) | 2006-12-21 | 2009-02-13 | Galderma Res & Dev S N C Snc | Emulsion comprenant au moins un retinoide et du peroxyde de benzole |
| FR2910321B1 (fr) | 2006-12-21 | 2009-07-10 | Galderma Res & Dev S N C Snc | Gel creme comprenant au moins un retinoide et du peroxyde de benzole |
| FR2916966B1 (fr) * | 2007-06-11 | 2011-01-14 | Galderma Res & Dev | Compositions comprenant au moins un compose retinoide, un compose anti-irritant et du peroxyde de benzoyle, et leurs utilisations |
| FR2916975B1 (fr) * | 2007-06-11 | 2009-09-04 | Galderma Res & Dev | Compositions comprenant au moins un compose retinoide, un compose anti-irritant et du peroxyde de benzoyle, et leurs utilisations |
| CN102686208A (zh) * | 2009-10-07 | 2012-09-19 | 塔格拉生物科技有限公司 | 包含过氧化苯甲酰的微胶囊和包含所述微胶囊的局部用组合物 |
| JP5784619B2 (ja) * | 2009-10-21 | 2015-09-24 | ドウ ファーマシューティカル サイエンシーズ、インク. | 過酸化ベンゾイルを含む粉末を湿潤させるための方法 |
| US9744150B2 (en) * | 2009-10-21 | 2017-08-29 | Dow Pharmaceutical Sciences Inc. | Suspension containing micronized benzoyl peroxide |
| BR112016022743A2 (pt) * | 2014-04-01 | 2017-08-15 | Galderma Res & Dev | Método para tratar e/ou evitar pelo menos uma cicatriz de acne, uso de uma combinação fixa de adapaleno e peróxido de benzoíla e composição |
| WO2017068673A1 (fr) * | 2015-10-21 | 2017-04-27 | マルホ株式会社 | Composition pharmaceutique pour la peau |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0375520A1 (fr) * | 1988-12-20 | 1990-06-27 | Centre International De Recherches Dermatologiques Galderma - Cird Galderma | Composition cosmétique ou pharmaceutique contenant des microsphères de polymères ou de corps gras chargées d'au moins un produit actif |
| US5879716A (en) * | 1985-12-18 | 1999-03-09 | Advanced Polymer Systems, Inc. | Methods and compositions for topical delivery of benzoyl peroxide |
| WO2003055472A1 (fr) * | 2001-12-21 | 2003-07-10 | Galderma Research & Development, Snc | Gel comprenant au moins un retinoide et du peroxyde de benzoyle |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7820186B2 (en) * | 2001-12-21 | 2010-10-26 | Galderma Research & Development | Gel composition for once-daily treatment of common acne comprising a combination of benzoyl peroxide and adapalene and/or adapalene salt |
-
2006
- 2006-05-17 FR FR0604407A patent/FR2901139B1/fr not_active Expired - Fee Related
-
2007
- 2007-05-16 CA CA002649124A patent/CA2649124A1/fr not_active Abandoned
- 2007-05-16 EP EP07766070A patent/EP2019663A2/fr not_active Withdrawn
- 2007-05-16 WO PCT/FR2007/051296 patent/WO2007132134A2/fr not_active Ceased
-
2008
- 2008-11-17 US US12/272,061 patent/US20090191245A1/en not_active Abandoned
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5879716A (en) * | 1985-12-18 | 1999-03-09 | Advanced Polymer Systems, Inc. | Methods and compositions for topical delivery of benzoyl peroxide |
| EP0375520A1 (fr) * | 1988-12-20 | 1990-06-27 | Centre International De Recherches Dermatologiques Galderma - Cird Galderma | Composition cosmétique ou pharmaceutique contenant des microsphères de polymères ou de corps gras chargées d'au moins un produit actif |
| WO2003055472A1 (fr) * | 2001-12-21 | 2003-07-10 | Galderma Research & Development, Snc | Gel comprenant au moins un retinoide et du peroxyde de benzoyle |
Non-Patent Citations (1)
| Title |
|---|
| EMBIL K ET AL: "THE MICROSPONGE DELIVERY SYSTEM (MDS): A TOPICAL DELIVERY SYSTEM WITH REDUCED IRRITANCY INCORPORATING MULTIPLE TRIGGERING MECHANISMS FOR THE RELEASE OF ACTIVES", JOURNAL OF MICROENCAPSULATION, TAYLOR AND FRANCIS, BASINGSTOKE, GB, vol. 13, no. 5, 1 September 1996 (1996-09-01), pages 575 - 588, XP000599288, ISSN: 0265-2048 * |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8936800B2 (en) | 2001-12-21 | 2015-01-20 | Galderma Research & Development | Gel composition for treatment of common acne comprising a combination of benzoyl peroxide and adapalene and/or adapalene salt |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007132134A2 (fr) | 2007-11-22 |
| CA2649124A1 (fr) | 2007-11-22 |
| FR2901139A1 (fr) | 2007-11-23 |
| US20090191245A1 (en) | 2009-07-30 |
| EP2019663A2 (fr) | 2009-02-04 |
| FR2901139B1 (fr) | 2009-03-20 |
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