WO2019203746A3 - Combinaison pharmaceutique comprenant du raloxifène et de l'aripiprazole - Google Patents

Combinaison pharmaceutique comprenant du raloxifène et de l'aripiprazole Download PDF

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Publication number
WO2019203746A3
WO2019203746A3 PCT/TR2018/050772 TR2018050772W WO2019203746A3 WO 2019203746 A3 WO2019203746 A3 WO 2019203746A3 TR 2018050772 W TR2018050772 W TR 2018050772W WO 2019203746 A3 WO2019203746 A3 WO 2019203746A3
Authority
WO
WIPO (PCT)
Prior art keywords
aripiprazole
raloxifene
pharmaceutical combination
pharmaceutically acceptable
acceptable salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/TR2018/050772
Other languages
English (en)
Other versions
WO2019203746A2 (fr
Inventor
Ali TÜRKYILMAZ
Nur PEHLIVAN AKALIN
Merve ERGUN DÖNMEZ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanovel Ilac Sanayi ve Ticaret AS
Original Assignee
Sanovel Ilac Sanayi ve Ticaret AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanovel Ilac Sanayi ve Ticaret AS filed Critical Sanovel Ilac Sanayi ve Ticaret AS
Publication of WO2019203746A2 publication Critical patent/WO2019203746A2/fr
Publication of WO2019203746A3 publication Critical patent/WO2019203746A3/fr
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4535Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom, e.g. pizotifen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Zoology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

La présente invention concerne une combinaison qui comprend du raloxifène ou un sel pharmaceutiquement acceptable de celui-ci et de l'aripiprazole ou un sel pharmaceutiquement acceptable de celui-ci et éventuellement au moins un excipient pharmaceutiquement acceptable pour une utilisation simultanée, séparée ou séquentielle.
PCT/TR2018/050772 2017-12-08 2018-12-06 Combinaison pharmaceutique comprenant du raloxifène et de l'aripiprazole Ceased WO2019203746A2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
TR2017/19919A TR201719919A2 (tr) 2017-12-08 2017-12-08 The pharmaceutical combination comprising raloxifene and aripiprazole
TR2017/19919 2017-12-08

Publications (2)

Publication Number Publication Date
WO2019203746A2 WO2019203746A2 (fr) 2019-10-24
WO2019203746A3 true WO2019203746A3 (fr) 2020-01-16

Family

ID=67952525

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/TR2018/050772 Ceased WO2019203746A2 (fr) 2017-12-08 2018-12-06 Combinaison pharmaceutique comprenant du raloxifène et de l'aripiprazole

Country Status (2)

Country Link
TR (1) TR201719919A2 (fr)
WO (1) WO2019203746A2 (fr)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070014864A1 (en) * 2005-07-15 2007-01-18 Teva Pharmaceutical Industries, Ltd. Novel pharmaceutical granulate
WO2015082562A1 (fr) * 2013-12-05 2015-06-11 Alrise Biosystems Gmbh Procédé de production de formulations médicamenteuses pour une administration par voie orale
WO2017149392A1 (fr) * 2016-03-04 2017-09-08 Sharon Anavi-Goffer Compositions auto-émulsifiantes de modulateurs du récepteur cb2

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070014864A1 (en) * 2005-07-15 2007-01-18 Teva Pharmaceutical Industries, Ltd. Novel pharmaceutical granulate
WO2015082562A1 (fr) * 2013-12-05 2015-06-11 Alrise Biosystems Gmbh Procédé de production de formulations médicamenteuses pour une administration par voie orale
WO2017149392A1 (fr) * 2016-03-04 2017-09-08 Sharon Anavi-Goffer Compositions auto-émulsifiantes de modulateurs du récepteur cb2

Also Published As

Publication number Publication date
TR201719919A2 (tr) 2019-06-21
WO2019203746A2 (fr) 2019-10-24

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