YU15500A - Process for preparation cyclic thioamides - Google Patents

Process for preparation cyclic thioamides

Info

Publication number
YU15500A
YU15500A YU15500A YUP15500A YU15500A YU 15500 A YU15500 A YU 15500A YU 15500 A YU15500 A YU 15500A YU P15500 A YUP15500 A YU P15500A YU 15500 A YU15500 A YU 15500A
Authority
YU
Yugoslavia
Prior art keywords
cyclic thioamides
preparation cyclic
preparation
preparing
thioamides
Prior art date
Application number
YU15500A
Other languages
Serbo-Croatian (sh)
Inventor
George Joseph Quallich
Jeffrey William Raggon
Paul David Hill
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of YU15500A publication Critical patent/YU15500A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C323/24—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/25—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/52—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)

Abstract

The present invention relates to a process for preparing a compound of the formula (I) wherewin b, Y and R3 are defined as above, useful for preparing novel aralkyl and aralkylidene heterocyclic lactams and imides which are selective agonists and antagonists of serotonin 1 (5 - HT1) receptors.
YU15500A 1999-03-30 2000-03-15 Process for preparation cyclic thioamides YU15500A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12683199P 1999-03-30 1999-03-30

Publications (1)

Publication Number Publication Date
YU15500A true YU15500A (en) 2002-03-18

Family

ID=22426907

Family Applications (1)

Application Number Title Priority Date Filing Date
YU15500A YU15500A (en) 1999-03-30 2000-03-15 Process for preparation cyclic thioamides

Country Status (25)

Country Link
US (1) US6388127B1 (en)
EP (1) EP1041070B1 (en)
JP (1) JP3566175B2 (en)
KR (1) KR100386524B1 (en)
CN (2) CN1163490C (en)
AR (1) AR029744A1 (en)
AT (1) ATE277025T1 (en)
AU (1) AU777097B2 (en)
BR (1) BR0001492A (en)
CA (1) CA2302727C (en)
CZ (1) CZ298140B6 (en)
DE (1) DE60013942T2 (en)
DK (1) DK1041070T3 (en)
ES (1) ES2226715T3 (en)
HU (1) HUP0001327A3 (en)
ID (1) ID25428A (en)
IL (1) IL135243A (en)
IN (1) IN188844B (en)
PL (1) PL196446B1 (en)
PT (1) PT1041070E (en)
RU (1) RU2219173C2 (en)
TR (1) TR200000834A2 (en)
TW (1) TW460472B (en)
YU (1) YU15500A (en)
ZA (1) ZA200001536B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE277025T1 (en) * 1999-03-30 2004-10-15 Pfizer Prod Inc METHOD FOR PRODUCING CYCLIC THIOAMIDS
US9557336B2 (en) 2012-09-07 2017-01-31 University Of Rochester Methods and compositions for site-specific labeling of peptides and proteins
US9999921B2 (en) 2015-06-15 2018-06-19 Gm Global Technology Operatioins Llc Method of making aluminum or magnesium based composite engine blocks or other parts with in-situ formed reinforced phases through squeeze casting or semi-solid metal forming and post heat treatment

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2755278A (en) * 1956-07-17 Thiamori
GB8412862D0 (en) * 1984-05-19 1984-06-27 Beecham Group Plc Compounds
EP0233287B1 (en) * 1984-10-04 1991-01-30 Zenyaku Kogyo Kabushikikaisha 1,4-thiazine derivatives, process for their preparation, and cardiotonics containing the same
CA2099233A1 (en) * 1992-06-29 1993-12-30 Conrad P. Dorn Morpholine and thiomorpholine tachykinin receptor antagonists
WO1994003652A1 (en) 1992-07-31 1994-02-17 Yokota Corporation Co., Ltd. Method of making metal of high purity from scrap of worked metal
GB9225377D0 (en) * 1992-12-04 1993-01-27 Ici Plc Herbicides
TW280812B (en) * 1993-07-02 1996-07-11 Bayer Ag
FR2715933B1 (en) * 1994-02-07 1996-04-12 Oreal New alkyl N- (hydroxyalkyl) carbamates and their applications in cosmetics, more particularly in hair compositions.
US5663409A (en) * 1995-06-07 1997-09-02 Novus International, Inc. Process for the preparation of 3-(methylthio) propanal and 2-hydroxy-4-(methylthio) butanenitrile
UA56185C2 (en) * 1996-09-30 2003-05-15 Пфайзер Інк. Aralkyl- and aralkylidene heterocyclic lactams and imids, a pharmaceutical composition and a treatment method
ATE277025T1 (en) * 1999-03-30 2004-10-15 Pfizer Prod Inc METHOD FOR PRODUCING CYCLIC THIOAMIDS

Also Published As

Publication number Publication date
CN1290829C (en) 2006-12-20
AU2263500A (en) 2000-10-05
DE60013942D1 (en) 2004-10-28
HUP0001327A3 (en) 2003-06-30
CA2302727C (en) 2004-02-24
CN1163490C (en) 2004-08-25
TW460472B (en) 2001-10-21
EP1041070B1 (en) 2004-09-22
PL196446B1 (en) 2008-01-31
CA2302727A1 (en) 2000-09-30
HU0001327D0 (en) 2000-06-28
ES2226715T3 (en) 2005-04-01
ZA200001536B (en) 2001-09-27
RU2219173C2 (en) 2003-12-20
ATE277025T1 (en) 2004-10-15
JP3566175B2 (en) 2004-09-15
IL135243A (en) 2005-09-25
AU777097B2 (en) 2004-09-30
HUP0001327A2 (en) 2001-04-28
AR029744A1 (en) 2003-07-16
HK1064364A1 (en) 2005-01-28
PL339287A1 (en) 2000-10-09
DE60013942T2 (en) 2006-02-23
KR20010014647A (en) 2001-02-26
CN1519230A (en) 2004-08-11
HK1032053A1 (en) 2001-07-06
TR200000834A2 (en) 2000-11-21
DK1041070T3 (en) 2005-01-24
IN188844B (en) 2002-11-09
CZ20001142A3 (en) 2000-12-13
PT1041070E (en) 2004-12-31
EP1041070A1 (en) 2000-10-04
JP2000309581A (en) 2000-11-07
KR100386524B1 (en) 2003-06-02
ID25428A (en) 2000-10-05
BR0001492A (en) 2000-10-17
CZ298140B6 (en) 2007-07-04
US6388127B1 (en) 2002-05-14
IL135243A0 (en) 2001-05-20
CN1273244A (en) 2000-11-15

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