YU213078A - Process for obtaining sulfonylamidine compounds - Google Patents

Process for obtaining sulfonylamidine compounds

Info

Publication number: YU213078A
Authority: YU; Yugoslavia
Prior art keywords: sulfonylamidine; compounds; obtaining; sulfonylamidine compounds; obtaining sulfonylamidine
Prior art date: 1977-09-08

Application number

YU02130/78A

Other languages

English (en)

Inventor

Z Tashma

G J Durant

Joung R Ch

R Ch Joung

Original Assignee

Smith Kline French Lab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-09-08

Filing date

1978-09-08

Publication date

1983-01-21

1978-09-08 Application filed by Smith Kline French Lab filed Critical Smith Kline French Lab

1983-01-21 Publication of YU213078A publication Critical patent/YU213078A/xx

Links

DFEXVBOMMIJOAW-UHFFFAOYSA-N carbamimidoylsulfonylmethanimidamide Chemical class NC(=N)S(=O)(=O)C(N)=N DFEXVBOMMIJOAW-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/32—Sulfur atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/65—One oxygen atom attached in position 3 or 5
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/08—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
- C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D277/26—Radicals substituted by sulfur atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
- C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
- C07D285/135—Nitrogen atoms

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pulmonology (AREA)
Life Sciences & Earth Sciences (AREA)
Immunology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyridine Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

YU02130/78A 1977-09-08 1978-09-08 Process for obtaining sulfonylamidine compounds YU213078A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB3746877		1977-09-08

Publications (1)

Publication Number	Publication Date
YU213078A true YU213078A (en)	1983-01-21

Family

ID=10396713

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
YU02130/78A YU213078A (en)	1977-09-08	1978-09-08	Process for obtaining sulfonylamidine compounds

Country Status (14)

Country	Link
US (3)	US4210658A (de)
EP (1)	EP0009061A1 (de)
JP (1)	JPS5452081A (de)
AT (1)	AT366666B (de)
AU (1)	AU518821B2 (de)
CA (1)	CA1111040A (de)
DK (1)	DK398078A (de)
FI (1)	FI62530C (de)
HU (1)	HU180294B (de)
IL (1)	IL55539A (de)
IT (1)	IT1099492B (de)
NO (1)	NO783053L (de)
YU (1)	YU213078A (de)
ZA (1)	ZA785113B (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4210658A (en) *	1977-09-08	1980-07-01	Smith Kline & French Laboratories Limited	Amidinosulphonic acid derivatives
US4375547A (en) *	1980-10-02	1983-03-01	Eli Lilly And Company	N-Methyl-N'-2-([(2-dimethylaminomethyl)-4-thiazolyl]methylthio)ethyl 2-nitro-1,1-ethenediamine
IE53068B1 (en) *	1981-06-15	1988-05-25	Merck & Co Inc	Diamino isothiazole-1-oxides and -1,1-dioxides as gastic secretion inhibitors
AU2222083A (en) *	1982-12-14	1984-06-21	Smith Kline & French Laboratories Limited	Pyridine derivatives
US4693850A (en) *	1985-03-15	1987-09-15	Mcneilab, Inc.	Methane sulfonic acid derivatives
US4656291A (en) *	1985-03-15	1987-04-07	Mcneilab, Inc.	Process for producing amidine sulfonic acids
US4781866A (en) *	1985-03-15	1988-11-01	Mcneilab, Inc.	Process for producing amidine sulfonic acid intermediates for guanidines
US4656270A (en) *	1985-03-15	1987-04-07	Mcneilab, Inc.	Process for producing guanidines such as linogliride
US4962114A (en) *	1986-01-21	1990-10-09	Yale University	1-alkyl-1-sulfonyl-2-alkoxycarbonylsulfenylhydrazines having antineoplastic activity
US4952573A (en) *	1988-03-23	1990-08-28	Laboratoirs Alcon S.A.	Compounds having GABA like activity, and use of same in tissue irrigating solutions
US5237072A (en) *	1990-02-06	1993-08-17	Allergan, Inc.	Method for producing amino-2-imidazoline derivatives
US5130441A (en) *	1990-02-06	1992-07-14	Allergan, Inc.	Method for producing amino-2-imidazoline derivatives
WO2022034121A1 (en)	2020-08-11	2022-02-17	Université De Strasbourg	H2 blockers targeting liver macrophages for the prevention and treatment of liver disease and cancer

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE758146A (fr) *	1969-10-29	1971-04-28	Smith Kline French Lab	Derives de l'amidine
US3734924A (en) *	1970-10-14	1973-05-22	Smith Kline French Lab	Carboxamidines
US4109003A (en) *	1974-03-12	1978-08-22	Smith Kline & French Laboratories Limited	Pharmacologically active compounds
US4090026A (en) *	1974-09-02	1978-05-16	Smith Kline & French Laboratories Limited	Certain nitrogen heterocyclic isothiocyanate esters
US4156727A (en) *	1975-07-31	1979-05-29	Smith Kline & French Laboratories Limited	Alkoxy pyridine compounds
GB1574214A (en) *	1976-03-11	1980-09-03	Smith Kline French Lab	Amidines
US4210658A (en) *	1977-09-08	1980-07-01	Smith Kline & French Laboratories Limited	Amidinosulphonic acid derivatives

1978
- 1978-09-06 US US05/940,063 patent/US4210658A/en not_active Expired - Lifetime
- 1978-09-07 NO NO783053A patent/NO783053L/no unknown
- 1978-09-07 HU HU78SI1647A patent/HU180294B/hu unknown
- 1978-09-07 CA CA310,844A patent/CA1111040A/en not_active Expired
- 1978-09-08 FI FI782760A patent/FI62530C/fi not_active IP Right Cessation
- 1978-09-08 YU YU02130/78A patent/YU213078A/xx unknown
- 1978-09-08 EP EP78300359A patent/EP0009061A1/de not_active Withdrawn
- 1978-09-08 AT AT0652178A patent/AT366666B/de not_active IP Right Cessation
- 1978-09-08 IL IL55539A patent/IL55539A/xx unknown
- 1978-09-08 DK DK398078A patent/DK398078A/da not_active Application Discontinuation
- 1978-09-08 AU AU39704/78A patent/AU518821B2/en not_active Expired
- 1978-09-08 JP JP11121478A patent/JPS5452081A/ja active Pending
- 1978-09-08 IT IT27493/78A patent/IT1099492B/it active
- 1978-09-08 ZA ZA00785113A patent/ZA785113B/xx unknown
1979
- 1979-11-05 US US06/090,949 patent/US4265896A/en not_active Expired - Lifetime
1980
- 1980-11-24 US US06/209,449 patent/US4375472A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
US4265896A (en)	1981-05-05
HU180294B (en)	1983-02-28
IT1099492B (it)	1985-09-18
AT366666B (de)	1982-04-26
FI62530B (fi)	1982-09-30
US4375472A (en)	1983-03-01
EP0009061A1 (de)	1980-04-02
ZA785113B (en)	1979-08-29
FI62530C (fi)	1983-01-10
AU518821B2 (en)	1981-10-22
US4210658A (en)	1980-07-01
FI782760A7 (fi)	1979-03-09
CA1111040A (en)	1981-10-20
NO783053L (no)	1979-03-09
IT7827493A0 (it)	1978-09-08
JPS5452081A (en)	1979-04-24
IL55539A (en)	1982-01-31
AU3970478A (en)	1980-03-13
ATA652178A (de)	1981-09-15
DK398078A (da)	1979-03-09
IL55539A0 (en)	1978-12-17

Publication	Publication Date	Title
YU33278A (en)	1982-10-31	Process for obtaining new pyrrolidinederivatives
YU63678A (en)	1983-01-21	Process for obtaining new pyridinyl-aminoalkylethers
YU42073B (en)	1988-04-30	Process for obtaining 1-oxadethiaceptham compounds
YU91378A (en)	1982-10-31	Process for obtaining 2-hydroxymethyl-3-hydroxy-6-(1-hydroxy-2-tert.-butylamino-ethyl)
YU250378A (en)	1983-04-30	Process for obtaining n-cyano-and n-alkinyl-2-(substitutedphenoxy)-butyramids
YU91478A (en)	1983-01-21	Process for obtaining hexahydro-gamma-carboline compounds
YU143678A (en)	1983-02-28	Process for obtaining substituted cyclopropylmethoxyanilides
YU137578A (en)	1983-01-21	Process for obtaining mercaptoacyl-aminobenzoylglycine
YU300377A (en)	1982-10-31	Process for obtaining 4-amino-epimeric oleandomycins
YU47478A (en)	1983-01-21	Process for obtaining new benzylpyrimidines
YU39417B (en)	1984-12-31	Process for obtaining auranophine
YU147978A (en)	1982-10-31	New process for obtaining auranophine
YU144078A (en)	1982-10-31	New process for obtaining benzoylcarbamide
YU184278A (en)	1983-01-21	Process for obtaining substituted 2-cyclopropyl-chromones
GB2003475B (en)	1982-03-17	Process for 2-chlorosulphinylazetidin-4-ones
YU42072B (en)	1988-04-30	Process for obtaining 1-oxadethiacepham compounds
YU71178A (en)	1983-01-21	Process for obtaining 2-hydroxybenzothiazole compounds
YU160978A (en)	1982-08-31	Process for obtaining tetrahydro-s-triazine-thione
YU40674B (en)	1986-04-30	Process for obtaining di-n-propylacetonitrile
YU137378A (en)	1983-01-21	New process for obtaining auranophin
YU40675B (en)	1986-04-30	Process for obtaining di-n-propyl-acetamide
YU42477B (en)	1988-10-31	Process for obtaining haloarylmalone amido-1-dethio-1-oxa-cephalosporins
YU42074B (en)	1988-04-30	Process for obtaining 1-oxadethiacepham compounds
YU7278A (en)	1983-01-21	Process for obtaining 1-formyl-dime-ring-indole-dihydroindole
IL54182A0 (en)	1978-06-15	Process for 3-beta-aminoazetiden-2-ones