ZA200100607B - Methods of treating diabetic cardiomyopathy using glycogen phosphorylase inhibitors. - Google Patents

Methods of treating diabetic cardiomyopathy using glycogen phosphorylase inhibitors.

Info

Publication number
ZA200100607B
ZA200100607B ZA200100607A ZA200100607A ZA200100607B ZA 200100607 B ZA200100607 B ZA 200100607B ZA 200100607 A ZA200100607 A ZA 200100607A ZA 200100607 A ZA200100607 A ZA 200100607A ZA 200100607 B ZA200100607 B ZA 200100607B
Authority
ZA
South Africa
Prior art keywords
methods
glycogen phosphorylase
treating diabetic
phosphorylase inhibitors
diabetic cardiomyopathy
Prior art date
Application number
ZA200100607A
Other languages
English (en)
Inventor
Judith Lee Treadway
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of ZA200100607B publication Critical patent/ZA200100607B/xx

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • A61K31/4045Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
    • AHUMAN NECESSITIES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
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    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
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    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
ZA200100607A 2000-01-24 2001-01-22 Methods of treating diabetic cardiomyopathy using glycogen phosphorylase inhibitors. ZA200100607B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17777000P 2000-01-24 2000-01-24

Publications (1)

Publication Number Publication Date
ZA200100607B true ZA200100607B (en) 2002-07-22

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ID=22649922

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200100607A ZA200100607B (en) 2000-01-24 2001-01-22 Methods of treating diabetic cardiomyopathy using glycogen phosphorylase inhibitors.

Country Status (12)

Country Link
US (1) US6867184B2 (fr)
EP (1) EP1125580A3 (fr)
JP (1) JP2001206856A (fr)
KR (1) KR20010083148A (fr)
AU (1) AU1639901A (fr)
CA (1) CA2331847A1 (fr)
CO (1) CO5271699A1 (fr)
HU (1) HUP0100321A3 (fr)
IL (1) IL140904A0 (fr)
NZ (1) NZ509481A (fr)
PE (1) PE20011053A1 (fr)
ZA (1) ZA200100607B (fr)

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GB0205176D0 (en) 2002-03-06 2002-04-17 Astrazeneca Ab Chemical compounds
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WO2006041922A2 (fr) * 2004-10-08 2006-04-20 Dara Biosciences, Inc. Agents, et procedes d'administration au systeme nerveux central
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WO2006055462A1 (fr) 2004-11-15 2006-05-26 Bristol-Myers Squibb Company Derives 2-amino-4- tetraline fonctionnalisee et inhibiteurs de la glycogene phosphorylase associes
WO2006053274A2 (fr) * 2004-11-15 2006-05-18 Bristol-Myers Squibb Company Derives de tetraline 2-amino-1-fonctionnalises et inhibiteurs correspondants de glycogene phosphorylase
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US20070026079A1 (en) * 2005-02-14 2007-02-01 Louis Herlands Intranasal administration of modulators of hypothalamic ATP-sensitive potassium channels
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
CN101516834B (zh) * 2006-09-13 2013-04-03 塞诺菲-安万特股份有限公司 用作凝血因子IXa抑制剂的异丝氨酸衍生物
KR101481041B1 (ko) * 2007-11-30 2015-01-12 (주)아모레퍼시픽 글루코오스-6-인산 탈수소효소의 활성 억제제 및 이를포함하는 지방세포 분화 억제용 조성물
CA2880432C (fr) 2012-08-21 2023-03-14 Ardelyx, Inc. Composes et procedes destines a inhiber un antiport medie par nhe dans le traitement des troubles associes a une retention de fluide ou a une surcharge de sel et des troubles du t ractus gastro-intestinal
KR102687458B1 (ko) * 2016-06-16 2024-07-24 호유 가부시키가이샤 생선 알레르기의 항원
HUE058867T2 (hu) 2017-12-15 2022-09-28 Medizinische Hochschule Hannover Javított vegyület szívelégtelenség kezelésére
CN113304149A (zh) * 2021-06-23 2021-08-27 广州医科大学 一种化合物在制备治疗2型糖尿病心肌病的药物中的应用

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US6867184B2 (en) 2005-03-15
HU0100321D0 (en) 2001-03-28
EP1125580A3 (fr) 2002-11-27
NZ509481A (en) 2005-02-25
PE20011053A1 (es) 2001-10-17
CA2331847A1 (fr) 2001-07-24
HUP0100321A3 (en) 2004-03-01
US20010046958A1 (en) 2001-11-29
KR20010083148A (ko) 2001-08-31
EP1125580A2 (fr) 2001-08-22
HUP0100321A2 (en) 2002-10-28
AU1639901A (en) 2001-07-26
CO5271699A1 (es) 2003-04-30

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