ZA200501267B - The use of N-(3-methoxy-5-methylpyrazin-2-yl)-2-(4-[1,3,4-oxadiazol-2-yl]phenyl)pyridene-3-sulphonamide as an anti-cancer agent - Google Patents

The use of N-(3-methoxy-5-methylpyrazin-2-yl)-2-(4-[1,3,4-oxadiazol-2-yl]phenyl)pyridene-3-sulphonamide as an anti-cancer agent Download PDF

Info

Publication number: ZA200501267B
Authority: ZA; South Africa
Prior art keywords: cancer; substance; composition; man; pharmaceutically acceptable
Prior art date: 2002-08-23

Application number

ZA200501267A

Other languages

English (en)

Inventor

Tonge David William

Boyle Francis Thomas

Johnstone Donna

Barrass Nigel Charles

Taylor Sian Tomiko

Hughes Andrew Mark

Ashford Marianne Bernice

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-08-23

Filing date

2005-02-11

Publication date

2006-10-25

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9942847&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200501267(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2005-02-11 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2006-10-25 Publication of ZA200501267B publication Critical patent/ZA200501267B/en

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Classifications

- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Organic Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Epidemiology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Oncology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Hematology (AREA)
Rheumatology (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

ZA200501267A 2002-08-23 2005-02-11 The use of N-(3-methoxy-5-methylpyrazin-2-yl)-2-(4-[1,3,4-oxadiazol-2-yl]phenyl)pyridene-3-sulphonamide as an anti-cancer agent ZA200501267B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GBGB0219660.8A GB0219660D0 (en)	2002-08-23	2002-08-23	Therapeutic use

Publications (1)

Publication Number	Publication Date
ZA200501267B true ZA200501267B (en)	2006-10-25

Family

ID=9942847

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200501267A ZA200501267B (en)	2002-08-23	2005-02-11	The use of N-(3-methoxy-5-methylpyrazin-2-yl)-2-(4-[1,3,4-oxadiazol-2-yl]phenyl)pyridene-3-sulphonamide as an anti-cancer agent

Country Status (31)

Country	Link
US (2)	US7820679B2 (de)
EP (2)	EP1545710B1 (de)
JP (2)	JP3663202B2 (de)
KR (1)	KR20050035280A (de)
CN (1)	CN100467023C (de)
AR (1)	AR041037A1 (de)
AT (1)	ATE427773T1 (de)
AU (1)	AU2003255835B8 (de)
BR (1)	BR0313655A (de)
CA (1)	CA2496476C (de)
CL (1)	CL2003001692A1 (de)
CY (1)	CY1110712T1 (de)
DE (1)	DE60327084D1 (de)
DK (1)	DK1545710T3 (de)
ES (1)	ES2323309T3 (de)
GB (1)	GB0219660D0 (de)
IL (1)	IL166730A0 (de)
IS (1)	IS2704B (de)
MX (1)	MXPA05001862A (de)
MY (2)	MY136449A (de)
NO (1)	NO330756B1 (de)
NZ (1)	NZ538114A (de)
PL (1)	PL375561A1 (de)
PT (1)	PT1545710E (de)
RU (1)	RU2340343C2 (de)
SA (1)	SA03240363B1 (de)
SI (1)	SI1545710T1 (de)
TW (1)	TWI302912B (de)
UA (1)	UA82071C2 (de)
WO (1)	WO2004018044A2 (de)
ZA (1)	ZA200501267B (de)

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KR101855382B1 (ko) *	2015-12-31	2018-05-04	경북대학교 산학협력단	설폰아마이드계 화합물을 유효성분으로 포함하는 암의 예방, 치료 및 전이 억제용 약학적 조성물
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GB0514743D0 (en)	2005-07-19	2005-08-24	Astrazeneca Ab	Salt

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- 2005-02-09 NO NO20050689A patent/NO330756B1/no not_active IP Right Cessation
- 2005-02-11 ZA ZA200501267A patent/ZA200501267B/en unknown
- 2005-03-22 IS IS7766A patent/IS2704B/is unknown
2009
- 2009-06-11 CY CY20091100620T patent/CY1110712T1/el unknown
2010
- 2010-09-13 US US12/880,347 patent/US20110003831A1/en not_active Abandoned

Also Published As

Publication number	Publication date
CA2496476A1 (en)	2004-03-04
IL166730A0 (en)	2006-01-15
US20110003831A1 (en)	2011-01-06
EP1545710B1 (de)	2009-04-08
GB0219660D0 (en)	2002-10-02
HK1077534A1 (en)	2006-02-17
AU2003255835B2 (en)	2007-04-05
RU2340343C2 (ru)	2008-12-10
TW200409768A (en)	2004-06-16
DE60327084D1 (de)	2009-05-20
DK1545710T3 (da)	2009-06-29
PL375561A1 (en)	2005-11-28
NO330756B1 (no)	2011-07-04
SI1545710T1 (sl)	2009-08-31
JP3663202B2 (ja)	2005-06-22
MY137595A (en)	2009-02-27
US7820679B2 (en)	2010-10-26
ES2323309T3 (es)	2009-07-13
IS7766A (is)	2005-03-22
PT1545710E (pt)	2009-05-26
AR041037A1 (es)	2005-04-27
EP1545710A2 (de)	2005-06-29
KR20050035280A (ko)	2005-04-15
AU2003255835A1 (en)	2004-03-11
WO2004018044A2 (en)	2004-03-04
EP2072082A2 (de)	2009-06-24
JP2004083590A (ja)	2004-03-18
RU2005108349A (ru)	2005-08-27
MY136449A (en)	2008-10-31
US20060094729A1 (en)	2006-05-04
JP2005097312A (ja)	2005-04-14
CY1110712T1 (el)	2015-06-10
CN100467023C (zh)	2009-03-11
CA2496476C (en)	2009-08-04
MXPA05001862A (es)	2005-06-03
NZ538114A (en)	2008-02-29
UA82071C2 (en)	2008-03-11
EP2072082A3 (de)	2009-12-23
SA03240363B1 (ar)	2009-04-11
AU2003255835B8 (en)	2007-05-17
CL2003001692A1 (es)	2005-01-21
WO2004018044A3 (en)	2004-05-06
BR0313655A (pt)	2005-06-21
WO2004018044A8 (en)	2004-06-24
CN1688365A (zh)	2005-10-26
IS2704B (is)	2010-12-15
ATE427773T1 (de)	2009-04-15
TWI302912B (en)	2008-11-11
NO20050689L (no)	2005-03-21

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