ZA200802194B - Oxazolidinone-quinolone hybrids is antibacterial compounds - Google Patents
Oxazolidinone-quinolone hybrids is antibacterial compoundsInfo
- Publication number
- ZA200802194B ZA200802194B ZA200802194A ZA200802194A ZA200802194B ZA 200802194 B ZA200802194 B ZA 200802194B ZA 200802194 A ZA200802194 A ZA 200802194A ZA 200802194 A ZA200802194 A ZA 200802194A ZA 200802194 B ZA200802194 B ZA 200802194B
- Authority
- ZA
- South Africa
- Prior art keywords
- oxazolidinone
- antibacterial compounds
- quinolone hybrids
- quinolone
- hybrids
- Prior art date
Links
- HGKANZZLRDQFIM-UHFFFAOYSA-N 1,3-oxazolidin-2-one;1h-quinolin-2-one Chemical compound O=C1NCCO1.C1=CC=C2NC(=O)C=CC2=C1 HGKANZZLRDQFIM-UHFFFAOYSA-N 0.000 title 1
- 230000000844 anti-bacterial effect Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP2005008573 | 2005-08-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200802194B true ZA200802194B (en) | 2009-03-25 |
Family
ID=37620798
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200802194A ZA200802194B (en) | 2005-08-08 | 2008-03-07 | Oxazolidinone-quinolone hybrids is antibacterial compounds |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20100222302A1 (fr) |
| EP (2) | EP1931684A2 (fr) |
| JP (1) | JP2009504631A (fr) |
| KR (1) | KR20080038397A (fr) |
| CN (1) | CN101238135B (fr) |
| AR (1) | AR054608A1 (fr) |
| AU (1) | AU2006277662A1 (fr) |
| BR (1) | BRPI0614730A2 (fr) |
| CA (1) | CA2616977A1 (fr) |
| IL (1) | IL189322A0 (fr) |
| MX (1) | MX2008001415A (fr) |
| NO (1) | NO20081180L (fr) |
| RU (1) | RU2008108477A (fr) |
| TW (1) | TW200740829A (fr) |
| WO (1) | WO2007017828A2 (fr) |
| ZA (1) | ZA200802194B (fr) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003031443A1 (fr) | 2001-10-04 | 2003-04-17 | Morphochem Aktiengesellschaft für kombinatorische Chemie | Antibiotiques a action duale renfermant une oxazolidinone et une quinolone ou une fraction de naphthyridinone |
| MXPA05011654A (es) | 2003-04-30 | 2005-12-15 | Morphochem Ag Komb Chemie | Uso de antibioticos hibridos de oxazolidinona-quinolina para el tratamiento del antrax y de otras infecciones. |
| DE10340485B4 (de) | 2003-09-03 | 2015-05-13 | Morphochem AG Aktiengesellschaft für kombinatorische Chemie | Verfahren zur Herstellung von Oxazolidinon-Chinolon Hybriden |
| ES2310299T5 (es) | 2003-12-18 | 2014-02-10 | Morphochem Aktiengesellschaft für kombinatorische Chemie | Antibióticos híbridos a base de oxazolidinona-quinolona |
| US8158797B2 (en) | 2003-12-18 | 2012-04-17 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Oxazolidinone-quinolone hybrid antibiotics |
| CN101300248A (zh) * | 2005-04-21 | 2008-11-05 | 塔甘塔治疗公司 | 膦酸酯化的氟喹诺酮、其抗菌类似物以及预防和治疗骨和关节感染的方法 |
| US8124623B2 (en) | 2006-11-10 | 2012-02-28 | Actelion Pharmaceuticals Ltd. | 5-hydroxymethyl-oxazolidin-2-one-derivatives and their uses as antibacterials |
| CL2007003332A1 (es) | 2006-11-24 | 2008-06-20 | Actelion Pharmaceuticals Ltd | Compuestos derivados de heterociclos condensados; compuestos intermediarios; composicion farmaceutica; y uso en la prevencion o tratamiento de infecciones bacterianas. |
| CL2008001002A1 (es) | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
| WO2011031744A1 (fr) * | 2009-09-09 | 2011-03-17 | Achaogen, Inc. | Analogues de fluoroquinolone antibactériens |
| EP3003289B1 (fr) | 2013-05-28 | 2019-02-20 | Morphochem Aktiengesellschaft für kombinatorische Chemie | L'administration d'antibactériens hybrides de oxazolidinone-quinolone |
| RU2675847C2 (ru) | 2013-05-28 | 2018-12-25 | Морфохем Акциенгезельшафт Фюр Комбинаторише Хеми | Комбинированные терапевтические средства, содержащие оксазолидинон-хинолоны, предназначенные для лечения бактериальных инфекций |
| US10087171B2 (en) | 2016-12-19 | 2018-10-02 | Actelion Pharmaceuticals Ltd | Crystalline forms of cadazolid |
| KR102476708B1 (ko) | 2017-11-01 | 2022-12-09 | 삼성전자주식회사 | 광학 필터, 및 이를 포함하는 카메라 모듈 및 전자 장치 |
| KR102673362B1 (ko) * | 2018-03-27 | 2024-06-05 | 삼성전자주식회사 | 근적외선 흡수 필름, 광학 필터 및 전자 장치 |
| CN115772176A (zh) * | 2022-12-02 | 2023-03-10 | 常州兰陵制药有限公司 | 左氧氟沙星关键药物中间体的合成方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU196411B (en) * | 1985-09-24 | 1988-11-28 | Hoffmann La Roche | Process for producing quinoline derivatives and pharmaceutical compositions containing them |
| DK164287A (da) | 1986-03-31 | 1987-10-01 | Sankyo Co | Quinolin-3-carboxylsyrederivater og fremgangsmaade til fremstilling deraf og deres anvendelse |
| JPH04128288A (ja) * | 1990-09-18 | 1992-04-28 | Teikoku Chem Ind Corp Ltd | キノロンカルボン酸誘導体及びその製造方法 |
| EP1349853B1 (fr) * | 2000-12-21 | 2006-03-08 | Pharmacia & Upjohn Company LLC | Derives antimicrobiens de la quinolone et leur utilisation pour le traitement d'infections bacteriennes |
| WO2003031443A1 (fr) | 2001-10-04 | 2003-04-17 | Morphochem Aktiengesellschaft für kombinatorische Chemie | Antibiotiques a action duale renfermant une oxazolidinone et une quinolone ou une fraction de naphthyridinone |
| EP2292615A1 (fr) | 2002-02-01 | 2011-03-09 | AstraZeneca AB | Dérivés de quinazoline |
| US6803469B2 (en) | 2002-08-05 | 2004-10-12 | The Procter & Gamble Company | Process for preparing quinolone antibiotic intermediates |
| MXPA05011654A (es) | 2003-04-30 | 2005-12-15 | Morphochem Ag Komb Chemie | Uso de antibioticos hibridos de oxazolidinona-quinolina para el tratamiento del antrax y de otras infecciones. |
| MXPA06000228A (es) * | 2003-07-02 | 2006-06-27 | Merck & Co Inc | Antibioticos de oxazolidinona sustituidos con un grupo ciclopropilo y derivados de los mismos. |
| ES2310299T5 (es) | 2003-12-18 | 2014-02-10 | Morphochem Aktiengesellschaft für kombinatorische Chemie | Antibióticos híbridos a base de oxazolidinona-quinolona |
-
2006
- 2006-08-03 AR ARP060103389A patent/AR054608A1/es unknown
- 2006-08-07 BR BRPI0614730A patent/BRPI0614730A2/pt not_active IP Right Cessation
- 2006-08-07 WO PCT/IB2006/052714 patent/WO2007017828A2/fr not_active Ceased
- 2006-08-07 EP EP06795600A patent/EP1931684A2/fr not_active Withdrawn
- 2006-08-07 US US12/063,305 patent/US20100222302A1/en not_active Abandoned
- 2006-08-07 MX MX2008001415A patent/MX2008001415A/es not_active Application Discontinuation
- 2006-08-07 TW TW095128893A patent/TW200740829A/zh unknown
- 2006-08-07 KR KR1020087005799A patent/KR20080038397A/ko not_active Ceased
- 2006-08-07 RU RU2008108477/04A patent/RU2008108477A/ru not_active Application Discontinuation
- 2006-08-07 JP JP2008525696A patent/JP2009504631A/ja active Pending
- 2006-08-07 AU AU2006277662A patent/AU2006277662A1/en not_active Abandoned
- 2006-08-07 CA CA002616977A patent/CA2616977A1/fr not_active Abandoned
- 2006-08-07 CN CN2006800290493A patent/CN101238135B/zh not_active Expired - Fee Related
- 2006-08-07 EP EP10004213A patent/EP2256120A1/fr not_active Withdrawn
-
2008
- 2008-02-06 IL IL189322A patent/IL189322A0/en unknown
- 2008-03-06 NO NO20081180A patent/NO20081180L/no not_active Application Discontinuation
- 2008-03-07 ZA ZA200802194A patent/ZA200802194B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AR054608A1 (es) | 2007-06-27 |
| MX2008001415A (es) | 2008-04-04 |
| EP1931684A2 (fr) | 2008-06-18 |
| US20100222302A1 (en) | 2010-09-02 |
| AU2006277662A1 (en) | 2007-02-15 |
| WO2007017828A2 (fr) | 2007-02-15 |
| NO20081180L (no) | 2008-04-15 |
| RU2008108477A (ru) | 2009-09-20 |
| KR20080038397A (ko) | 2008-05-06 |
| BRPI0614730A2 (pt) | 2016-11-01 |
| CA2616977A1 (fr) | 2007-02-15 |
| JP2009504631A (ja) | 2009-02-05 |
| TW200740829A (en) | 2007-11-01 |
| WO2007017828A3 (fr) | 2007-07-19 |
| IL189322A0 (en) | 2008-06-05 |
| CN101238135A (zh) | 2008-08-06 |
| EP2256120A1 (fr) | 2010-12-01 |
| CN101238135B (zh) | 2011-05-11 |
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