ZA200802194B - Oxazolidinone-quinolone hybrids is antibacterial compounds - Google Patents
Oxazolidinone-quinolone hybrids is antibacterial compoundsInfo
- Publication number
- ZA200802194B ZA200802194B ZA200802194A ZA200802194A ZA200802194B ZA 200802194 B ZA200802194 B ZA 200802194B ZA 200802194 A ZA200802194 A ZA 200802194A ZA 200802194 A ZA200802194 A ZA 200802194A ZA 200802194 B ZA200802194 B ZA 200802194B
- Authority
- ZA
- South Africa
- Prior art keywords
- oxazolidinone
- antibacterial compounds
- quinolone hybrids
- quinolone
- hybrids
- Prior art date
Links
- HGKANZZLRDQFIM-UHFFFAOYSA-N 1,3-oxazolidin-2-one;1h-quinolin-2-one Chemical compound O=C1NCCO1.C1=CC=C2NC(=O)C=CC2=C1 HGKANZZLRDQFIM-UHFFFAOYSA-N 0.000 title 1
- 230000000844 anti-bacterial effect Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP2005008573 | 2005-08-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200802194B true ZA200802194B (en) | 2009-03-25 |
Family
ID=37620798
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200802194A ZA200802194B (en) | 2005-08-08 | 2008-03-07 | Oxazolidinone-quinolone hybrids is antibacterial compounds |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20100222302A1 (fr) |
| EP (2) | EP1931684A2 (fr) |
| JP (1) | JP2009504631A (fr) |
| KR (1) | KR20080038397A (fr) |
| CN (1) | CN101238135B (fr) |
| AR (1) | AR054608A1 (fr) |
| AU (1) | AU2006277662A1 (fr) |
| BR (1) | BRPI0614730A2 (fr) |
| CA (1) | CA2616977A1 (fr) |
| IL (1) | IL189322A0 (fr) |
| MX (1) | MX2008001415A (fr) |
| NO (1) | NO20081180L (fr) |
| RU (1) | RU2008108477A (fr) |
| TW (1) | TW200740829A (fr) |
| WO (1) | WO2007017828A2 (fr) |
| ZA (1) | ZA200802194B (fr) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003031443A1 (fr) | 2001-10-04 | 2003-04-17 | Morphochem Aktiengesellschaft für kombinatorische Chemie | Antibiotiques a action duale renfermant une oxazolidinone et une quinolone ou une fraction de naphthyridinone |
| ES2308171T3 (es) | 2003-04-30 | 2008-12-01 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Uso de antibioticos hibridos de oxazolidinona-quinolina para el tratamiento del antrax y de otras infecciones. |
| DE10340485B4 (de) | 2003-09-03 | 2015-05-13 | Morphochem AG Aktiengesellschaft für kombinatorische Chemie | Verfahren zur Herstellung von Oxazolidinon-Chinolon Hybriden |
| CA2549675C (fr) | 2003-12-18 | 2012-11-20 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Antibiotiques hybrides a base d'oxazolidinone-quinolone |
| US8158797B2 (en) | 2003-12-18 | 2012-04-17 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Oxazolidinone-quinolone hybrid antibiotics |
| AU2006277682A1 (en) * | 2005-04-21 | 2007-02-15 | Targanta Therapeutics Inc. | Phosphonated fluoroquinolones, antibacterial analogs thereof, and methods for the prevention and treatment of bone and joint infections |
| US8124623B2 (en) | 2006-11-10 | 2012-02-28 | Actelion Pharmaceuticals Ltd. | 5-hydroxymethyl-oxazolidin-2-one-derivatives and their uses as antibacterials |
| CL2007003332A1 (es) | 2006-11-24 | 2008-06-20 | Actelion Pharmaceuticals Ltd | Compuestos derivados de heterociclos condensados; compuestos intermediarios; composicion farmaceutica; y uso en la prevencion o tratamiento de infecciones bacterianas. |
| CL2008001002A1 (es) | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
| WO2011031744A1 (fr) * | 2009-09-09 | 2011-03-17 | Achaogen, Inc. | Analogues de fluoroquinolone antibactériens |
| CN105246476B (zh) | 2013-05-28 | 2019-11-15 | 莫弗凯姆联合化学股份公司 | 含噁唑烷酮-喹诺酮的联合疗法在治疗细菌感染中的应用 |
| MX371037B (es) | 2013-05-28 | 2020-01-14 | Morphochem Aktiengesellschaft Fuer Komb Chemie | Antibacterianos híbridos de oxazolidinona-quinolona para el tratamiento parenteral o profilaxis de enfermedades bacterianas. |
| US10087171B2 (en) | 2016-12-19 | 2018-10-02 | Actelion Pharmaceuticals Ltd | Crystalline forms of cadazolid |
| KR102476708B1 (ko) | 2017-11-01 | 2022-12-09 | 삼성전자주식회사 | 광학 필터, 및 이를 포함하는 카메라 모듈 및 전자 장치 |
| KR102673362B1 (ko) * | 2018-03-27 | 2024-06-05 | 삼성전자주식회사 | 근적외선 흡수 필름, 광학 필터 및 전자 장치 |
| CN115772176A (zh) * | 2022-12-02 | 2023-03-10 | 常州兰陵制药有限公司 | 左氧氟沙星关键药物中间体的合成方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE72668T1 (de) * | 1985-09-24 | 1992-03-15 | Hoffmann La Roche | Chinolinderivate. |
| FI871419L (fi) | 1986-03-31 | 1987-10-01 | Sankyo Co | Kinolin-3-karboxylsyraderivat, deras framstaellning och anvaendning. |
| JPH04128288A (ja) * | 1990-09-18 | 1992-04-28 | Teikoku Chem Ind Corp Ltd | キノロンカルボン酸誘導体及びその製造方法 |
| ATE319710T1 (de) * | 2000-12-21 | 2006-03-15 | Pharmacia & Upjohn Co Llc | Antimikrobielle chinolonderivate und ihre verwendung zur behandlung bakterieller infektionen |
| WO2003031443A1 (fr) | 2001-10-04 | 2003-04-17 | Morphochem Aktiengesellschaft für kombinatorische Chemie | Antibiotiques a action duale renfermant une oxazolidinone et une quinolone ou une fraction de naphthyridinone |
| CN1625555A (zh) | 2002-02-01 | 2005-06-08 | 阿斯特拉曾尼卡有限公司 | 喹唑啉化合物 |
| US6803469B2 (en) | 2002-08-05 | 2004-10-12 | The Procter & Gamble Company | Process for preparing quinolone antibiotic intermediates |
| ES2308171T3 (es) | 2003-04-30 | 2008-12-01 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Uso de antibioticos hibridos de oxazolidinona-quinolina para el tratamiento del antrax y de otras infecciones. |
| EP1646629B1 (fr) * | 2003-07-02 | 2010-06-23 | Merck Sharp & Dohme Corp. | Antibiotiques a base d'oxazolidinone substituee par un groupe cyclipropyl et derives |
| CA2549675C (fr) * | 2003-12-18 | 2012-11-20 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Antibiotiques hybrides a base d'oxazolidinone-quinolone |
-
2006
- 2006-08-03 AR ARP060103389A patent/AR054608A1/es unknown
- 2006-08-07 CN CN2006800290493A patent/CN101238135B/zh not_active Expired - Fee Related
- 2006-08-07 TW TW095128893A patent/TW200740829A/zh unknown
- 2006-08-07 KR KR1020087005799A patent/KR20080038397A/ko not_active Ceased
- 2006-08-07 EP EP06795600A patent/EP1931684A2/fr not_active Withdrawn
- 2006-08-07 EP EP10004213A patent/EP2256120A1/fr not_active Withdrawn
- 2006-08-07 JP JP2008525696A patent/JP2009504631A/ja active Pending
- 2006-08-07 BR BRPI0614730A patent/BRPI0614730A2/pt not_active IP Right Cessation
- 2006-08-07 WO PCT/IB2006/052714 patent/WO2007017828A2/fr not_active Ceased
- 2006-08-07 AU AU2006277662A patent/AU2006277662A1/en not_active Abandoned
- 2006-08-07 RU RU2008108477/04A patent/RU2008108477A/ru not_active Application Discontinuation
- 2006-08-07 US US12/063,305 patent/US20100222302A1/en not_active Abandoned
- 2006-08-07 CA CA002616977A patent/CA2616977A1/fr not_active Abandoned
- 2006-08-07 MX MX2008001415A patent/MX2008001415A/es not_active Application Discontinuation
-
2008
- 2008-02-06 IL IL189322A patent/IL189322A0/en unknown
- 2008-03-06 NO NO20081180A patent/NO20081180L/no not_active Application Discontinuation
- 2008-03-07 ZA ZA200802194A patent/ZA200802194B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2616977A1 (fr) | 2007-02-15 |
| CN101238135A (zh) | 2008-08-06 |
| EP1931684A2 (fr) | 2008-06-18 |
| MX2008001415A (es) | 2008-04-04 |
| EP2256120A1 (fr) | 2010-12-01 |
| CN101238135B (zh) | 2011-05-11 |
| WO2007017828A2 (fr) | 2007-02-15 |
| BRPI0614730A2 (pt) | 2016-11-01 |
| TW200740829A (en) | 2007-11-01 |
| US20100222302A1 (en) | 2010-09-02 |
| RU2008108477A (ru) | 2009-09-20 |
| JP2009504631A (ja) | 2009-02-05 |
| KR20080038397A (ko) | 2008-05-06 |
| AR054608A1 (es) | 2007-06-27 |
| AU2006277662A1 (en) | 2007-02-15 |
| WO2007017828A3 (fr) | 2007-07-19 |
| NO20081180L (no) | 2008-04-15 |
| IL189322A0 (en) | 2008-06-05 |
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