ZA724880B - 6-substituted 4h-imidazo(112-a)(1,4)benzodiazepine and processes for their production - Google Patents

6-substituted 4h-imidazo(112-a)(1,4)benzodiazepine and processes for their production

Info

Publication number: ZA724880B
Authority: ZA; South Africa
Prior art keywords: benzodiazepine; imidazo; substituted; processes; production
Prior art date: 1971-08-04

Application number

ZA724880A

Other languages

English (en)

Inventor

J Hester

A R Hanze

Original Assignee

Upjohn Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1971-08-04

Filing date

1972-07-14

Publication date

1973-06-27

1972-07-14 Application filed by Upjohn Co filed Critical Upjohn Co

1973-06-27 Publication of ZA724880B publication Critical patent/ZA724880B/xx

Links

GUJAGMICFDYKNR-UHFFFAOYSA-N 1,4-benzodiazepine Chemical compound N1C=CN=CC2=CC=CC=C12 GUJAGMICFDYKNR-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/116—Heterocyclic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Neurology (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurosurgery (AREA)
Polymers & Plastics (AREA)
Pain & Pain Management (AREA)
Biomedical Technology (AREA)
Physical Education & Sports Medicine (AREA)
Food Science & Technology (AREA)
Animal Husbandry (AREA)
Orthopedic Medicine & Surgery (AREA)
Anesthesiology (AREA)
Zoology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

ZA724880A 1971-08-04 1972-07-14 6-substituted 4h-imidazo(112-a)(1,4)benzodiazepine and processes for their production ZA724880B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US16909171A	1971-08-04	1971-08-04

Publications (1)

Publication Number	Publication Date
ZA724880B true ZA724880B (en)	1973-06-27

Family

ID=22614230

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA724880A ZA724880B (en)	1971-08-04	1972-07-14	6-substituted 4h-imidazo(112-a)(1,4)benzodiazepine and processes for their production

Country Status (8)

Country	Link
JP (3)	JPS5714351B1 (cs)
AU (1)	AU461139B2 (cs)
BE (1)	BE787251A (cs)
CH (3)	CH574444A5 (cs)
DE (1)	DE2237592C2 (cs)
FR (1)	FR2150732B1 (cs)
GB (4)	GB1389437A (cs)
ZA (1)	ZA724880B (cs)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3917627A (en) *	1971-08-04	1975-11-04	Upjohn Co	6-Substituted 4H-imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines and process for their production
FR2183716A1 (en) *	1972-05-05	1973-12-21	Centre Etd Ind Pharma	Substd-6-phenyl-4h-imidazo (1,2-a)-1,4-benzo diazepines - - tranquillisers anxiolytics,sedatives and muscle-relaxants
ZA755418B (en) *	1974-09-11	1977-06-29	Hoffmann La Roche	Diazepine derivatives
US3910946A (en) *	1974-09-12	1975-10-07	Upjohn Co	4H-Imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines
CA1060892A (en) *	1974-11-06	1979-08-21	Parke, Davis And Company	Diazepine compounds and method for their production
SE422580B (sv) *	1975-08-07	1982-03-15	Hoffmann La Roche	Analogiforfarande for framstellning av imidazo (1,5-a)(1,4)diazepin-foreningar
US4118386A (en) *	1977-04-04	1978-10-03	Hoffmann-La Roche Inc.	Synthesis of imidazo[1,5-a]diazepine-3-carboxylates
WO1994026723A2 (en) *	1993-05-14	1994-11-24	Genentech, Inc.	ras FARNESYL TRANSFERASE INHIBITORS
WO1996023790A1 (de) *	1995-02-02	1996-08-08	F. Hoffmann-La Roche Ag	Acetylimidazobenzodiazepine
EP3160969B1 (en)	2014-06-26	2023-09-13	The Johns Hopkins University	Peripherally restricted gaba positive allosteric modulators for the treatment of irritable bowel syndrome and other ailments of the peripheral nervous system
JP7139323B2 (ja) *	2016-11-01	2022-09-20	エフ．ホフマン－ラロシュアーゲー	Ｃｎｓ関連疾患を処置するための１，３－ジヒドロ－１，４－ベンゾジアゼピン－２－チオン
CN113717176B (zh) *	2021-10-09	2022-07-05	上海再启生物技术有限公司	一种制备瑞马唑仑的方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3987052A (en) *	1969-03-17	1976-10-19	The Upjohn Company	6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines

0
- BE BE787251D patent/BE787251A/xx not_active IP Right Cessation
1972
- 1972-07-13 GB GB3413874A patent/GB1389437A/en not_active Expired
- 1972-07-13 GB GB3288572A patent/GB1389434A/en not_active Expired
- 1972-07-13 GB GB3412474A patent/GB1389435A/en not_active Expired
- 1972-07-13 GB GB3412574A patent/GB1389436A/en not_active Expired
- 1972-07-14 ZA ZA724880A patent/ZA724880B/xx unknown
- 1972-07-18 AU AU44673/72A patent/AU461139B2/en not_active Expired
- 1972-07-28 CH CH1130272A patent/CH574444A5/xx not_active IP Right Cessation
- 1972-07-28 CH CH1435775A patent/CH584206A5/xx not_active IP Right Cessation
- 1972-07-28 CH CH1435675A patent/CH591488A5/xx not_active IP Right Cessation
- 1972-07-31 DE DE2237592A patent/DE2237592C2/de not_active Expired
- 1972-08-03 FR FR7228090A patent/FR2150732B1/fr not_active Expired
- 1972-08-04 JP JP7775772A patent/JPS5714351B1/ja active Pending
1979
- 1979-08-02 JP JP9817279A patent/JPS5547686A/ja active Granted
1980
- 1980-06-16 JP JP8030780A patent/JPS5726667A/ja active Granted

Also Published As

Publication number	Publication date
FR2150732A1 (cs)	1973-04-13
JPS5714351B1 (cs)	1982-03-24
DE2237592C2 (de)	1985-08-14
JPS5734277B2 (cs)	1982-07-22
CH574444A5 (cs)	1976-04-15
CH591488A5 (cs)	1977-09-30
JPS5726667A (en)	1982-02-12
AU461139B2 (en)	1975-05-15
JPS5547686A (en)	1980-04-04
GB1389436A (en)	1975-04-03
JPS5732066B2 (cs)	1982-07-08
GB1389435A (en)	1975-04-03
DE2237592A1 (de)	1973-02-15
AU4467372A (en)	1974-01-24
GB1389437A (en)	1975-04-03
GB1389434A (en)	1975-04-03
CH584206A5 (cs)	1977-01-31
FR2150732B1 (cs)	1976-04-16
BE787251A (fr)	1973-02-05

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