ZA785691B - Analogs of somatostatin and process for the manufacture thereof - Google Patents

Analogs of somatostatin and process for the manufacture thereof

Info

Publication number: ZA785691B
Authority: ZA; South Africa
Prior art keywords: somatostatin; analogs; manufacture
Prior art date: 1977-10-11

Application number

ZA00785691A

Other languages

English (en)

Inventor

J Meienhofer

A Felix

Torres H Gallo

E Heimer

W Dairman

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-10-11

Filing date

1978-10-09

Publication date

1979-09-26

1978-10-09 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

1979-09-26 Publication of ZA785691B publication Critical patent/ZA785691B/xx

Links

102000005157 Somatostatin Human genes 0.000 title 1
108010056088 Somatostatin Proteins 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
238000000034 method Methods 0.000 title 1
NHXLMOGPVYXJNR-ATOGVRKGSA-N somatostatin Chemical compound C([C@H]1C(=O)N[C@H](C(N[C@@H](CO)C(=O)N[C@@H](CSSC[C@@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC=2C=CC=CC=2)C(=O)N[C@@H](CC=2C=CC=CC=2)C(=O)N[C@@H](CC=2C3=CC=CC=C3NC=2)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N1)[C@@H](C)O)NC(=O)CNC(=O)[C@H](C)N)C(O)=O)=O)[C@H](O)C)C1=CC=CC=C1 NHXLMOGPVYXJNR-ATOGVRKGSA-N 0.000 title 1
229960000553 somatostatin Drugs 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/655—Somatostatins
- C07K14/6555—Somatostatins at least 1 amino acid in D-form
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S930/00—Peptide or protein sequence
- Y10S930/01—Peptide or protein sequence
- Y10S930/16—Somatostatin; related peptides

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Gastroenterology & Hepatology (AREA)
Genetics & Genomics (AREA)
Zoology (AREA)
Toxicology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Endocrinology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

ZA00785691A 1977-10-11 1978-10-09 Analogs of somatostatin and process for the manufacture thereof ZA785691B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US05/840,922 US4145337A (en)	1977-10-11	1977-10-11	Aminoethylglycine containing polypeptides

Publications (1)

Publication Number	Publication Date
ZA785691B true ZA785691B (en)	1979-09-26

Family

ID=25283583

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA00785691A ZA785691B (en)	1977-10-11	1978-10-09	Analogs of somatostatin and process for the manufacture thereof

Country Status (14)

Country	Link
US (1)	US4145337A (it)
EP (1)	EP0001449B1 (it)
JP (1)	JPS5461171A (it)
AT (1)	ATA726778A (it)
AU (1)	AU508559B1 (it)
CA (1)	CA1113457A (it)
DE (1)	DE2860623D1 (it)
DK (1)	DK451578A (it)
IE (1)	IE47448B1 (it)
IL (1)	IL55706A (it)
IT (1)	IT1099359B (it)
NZ (1)	NZ188611A (it)
PH (1)	PH13740A (it)
ZA (1)	ZA785691B (it)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0144290A3 (de) *	1983-12-01	1987-05-27	Ciba-Geigy Ag	Substituierte Aethylendiaminderivate
AU5410786A (en) *	1985-03-04	1986-09-11	Fujisawa Pharmaceutical Co., Ltd.	Amino acid derivatives and processes for preparation thereof
US5824772A (en) *	1995-04-04	1998-10-20	Advanced Bioconcept, Inc.	Fluorescent somatostatin
US5693679A (en) *	1995-04-04	1997-12-02	Advanced Bioconcept, Inc.	Fluorescent somatostatin
AU6382999A (en) *	1998-08-24	2000-03-14	Jeffrey D. White	Somatostatin analogs
YU68102A (sh) *	2000-03-16	2006-01-16	F. Hoffmann-La Roche Ag.	Derivati karboksilne kiseline kao ip antagonisti
CN113501771B (zh) *	2021-07-08	2023-07-28	成都泰和伟业生物科技有限公司	一种n-(2-氨乙基)甘氨酸衍生物的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3862925A (en) *	1973-07-05	1975-01-28	American Home Prod	Preparation of somatotropin release inhibiting factor and intermediates therefor

1977
- 1977-10-11 US US05/840,922 patent/US4145337A/en not_active Expired - Lifetime
1978
- 1978-10-05 DE DE7878101073T patent/DE2860623D1/de not_active Expired
- 1978-10-05 EP EP78101073A patent/EP0001449B1/de not_active Expired
- 1978-10-09 PH PH21690A patent/PH13740A/en unknown
- 1978-10-09 NZ NZ188611A patent/NZ188611A/xx unknown
- 1978-10-09 JP JP12369378A patent/JPS5461171A/ja active Pending
- 1978-10-09 ZA ZA00785691A patent/ZA785691B/xx unknown
- 1978-10-10 AU AU40561/78A patent/AU508559B1/en not_active Expired
- 1978-10-10 DK DK451578A patent/DK451578A/da not_active Application Discontinuation
- 1978-10-10 CA CA312,934A patent/CA1113457A/en not_active Expired
- 1978-10-10 IE IE2017/78A patent/IE47448B1/en unknown
- 1978-10-10 IL IL55706A patent/IL55706A/xx unknown
- 1978-10-10 AT AT0726778A patent/ATA726778A/de not_active Application Discontinuation
- 1978-10-11 IT IT28638/78A patent/IT1099359B/it active

Also Published As

Publication number	Publication date
IL55706A (en)	1981-10-30
US4145337A (en)	1979-03-20
AU508559B1 (en)	1980-03-27
JPS5461171A (en)	1979-05-17
NZ188611A (en)	1981-11-19
EP0001449B1 (de)	1981-04-15
DE2860623D1 (en)	1981-05-07
IT7828638A0 (it)	1978-10-11
ATA726778A (de)	1982-07-15
EP0001449A3 (en)	1979-06-27
PH13740A (en)	1980-09-10
DK451578A (da)	1979-04-12
IE47448B1 (en)	1984-03-21
CA1113457A (en)	1981-12-01
IE782017L (en)	1979-04-11
EP0001449A2 (de)	1979-04-18
IT1099359B (it)	1985-09-18
IL55706A0 (en)	1978-12-17

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