ZA871987B - 5h-1,3,4-thiadiazole(3,2-a)pyrimidin-5-one derivatives and fungicidal compositions containing the same - Google Patents

5h-1,3,4-thiadiazole(3,2-a)pyrimidin-5-one derivatives and fungicidal compositions containing the same

Info

Publication number: ZA871987B
Authority: ZA; South Africa
Prior art keywords: pyrimidin; derivatives; thiadiazole; same; compositions containing
Prior art date: 1986-03-19

Application number

ZA871987A

Other languages

English (en)

Inventor

Yukio Tokunaga

Tokunaga Yukio

Yoshiyuki Kojima

Kojima Yoshiyuki

Shinichiro Maeno

Maeno Shinichiro

Nobumitsu Sawai

Sawai Nobumitsu

Yasuo Saso

Saso Yasuo

Original Assignee

Kumiai Chemical Industry Co

Ihara Chemical Ind Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-03-19

Filing date

1987-03-18

Publication date

1988-05-25

1987-03-18 Application filed by Kumiai Chemical Industry Co, Ihara Chemical Ind Co filed Critical Kumiai Chemical Industry Co

1988-05-25 Publication of ZA871987B publication Critical patent/ZA871987B/xx

Links

230000000855 fungicidal effect Effects 0.000 title abstract 2
BDTRIDKONHOQQN-UHFFFAOYSA-N 4h-pyrimidin-5-one Chemical class O=C1CN=CN=C1 BDTRIDKONHOQQN-UHFFFAOYSA-N 0.000 title 1
239000000203 mixture Substances 0.000 title 1
240000008067 Cucumis sativus Species 0.000 abstract 2
235000010799 Cucumis sativus var sativus Nutrition 0.000 abstract 2
241000223600 Alternaria Species 0.000 abstract 1
244000178993 Brassica juncea Species 0.000 abstract 1
235000011332 Brassica juncea Nutrition 0.000 abstract 1
235000010149 Brassica rapa subsp chinensis Nutrition 0.000 abstract 1
235000007688 Lycopersicon esculentum Nutrition 0.000 abstract 1
206010027146 Melanoderma Diseases 0.000 abstract 1
240000007594 Oryza sativa Species 0.000 abstract 1
235000007164 Oryza sativa Nutrition 0.000 abstract 1
241000233679 Peronosporaceae Species 0.000 abstract 1
235000014443 Pyrus communis Nutrition 0.000 abstract 1
240000003768 Solanum lycopersicum Species 0.000 abstract 1
NBWUDDLJZAKVFL-UHFFFAOYSA-N [1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one Chemical class O=C1C=CN=C2SC=NN12 NBWUDDLJZAKVFL-UHFFFAOYSA-N 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
244000053095 fungal pathogen Species 0.000 abstract 1
235000009566 rice Nutrition 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Health & Medical Sciences (AREA)
Pest Control & Pesticides (AREA)
Plant Pathology (AREA)
Agronomy & Crop Science (AREA)
Engineering & Computer Science (AREA)
Dentistry (AREA)
General Health & Medical Sciences (AREA)
Wood Science & Technology (AREA)
Zoology (AREA)
Environmental Sciences (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

ZA871987A 1986-03-19 1987-03-18 5h-1,3,4-thiadiazole(3,2-a)pyrimidin-5-one derivatives and fungicidal compositions containing the same ZA871987B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
JP6174786		1986-03-19

Publications (1)

Publication Number	Publication Date
ZA871987B true ZA871987B (en)	1988-05-25

Family

ID=13180068

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA871987A ZA871987B (en)	1986-03-19	1987-03-18	5h-1,3,4-thiadiazole(3,2-a)pyrimidin-5-one derivatives and fungicidal compositions containing the same

Country Status (7)

Country	Link
US (2)	US4866064A (de)
EP (1)	EP0238059B1 (de)
JP (1)	JPH07110865B2 (de)
AT (1)	ATE90683T1 (de)
DE (1)	DE3786185T2 (de)
ES (1)	ES2058068T3 (de)
ZA (1)	ZA871987B (de)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
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EP0238059B1 (de) *	1986-03-19	1993-06-16	Kumiai Chemical Industry Co., Ltd.	5H-1,3,4-Thiazol[3,2-a]pyrimidin-5-on-Derivate und diese enthaltende fungizide Zubereitungen
DE3763282D1 (de) *	1986-03-19	1990-07-26	Kumiai Chemical Industry Co	Fungizide zur verwendung in der landwirtschaft und im gartenbau.
DE3786365T2 (de) *	1986-04-07	1993-10-21	Ihara Chemical Ind Co	5H-1,3,4-Thiadiazolo[3,2-a]pyrimidin-5-on-Derivate und diese enthaltende Gartenbau- und landwirtschaftliche Fungizidmittel.
EP0282635A3 (de) *	1987-03-18	1989-11-08	Kumiai Chemical Industry Co., Ltd.	5H-1,3,4-Thiadiazolo[3,2-a]pyrimidin-5-onderivate und diese enthaltende fungizide Zubereitungen
IT1255219B (it) *	1992-07-14	1995-10-20	Ct Lab Farm Srl	Derivati del tiadiazolo per la cura degli stati depressivi
KR102107954B1 (ko) *	2007-03-12	2020-05-07	인트라-셀룰라 써래피스, 인코퍼레이티드.	치환된 헤테로환 융합 감마-카르볼린 합성
KR20140146192A (ko)	2012-04-14	2014-12-24	인트라-셀룰라 써래피스, 인코퍼레이티드.	유기 화합물
US9708322B2 (en)	2013-03-15	2017-07-18	Intra-Cellular Therapies, Inc.	Substituted pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalines for inhibiting serotonin reuptake transporter activity
KR102373288B1 (ko)	2013-12-03	2022-03-10	인트라-셀룰라 써래피스, 인코퍼레이티드.	신규한 방법
US10077267B2 (en)	2014-04-04	2018-09-18	Intra-Cellular Therapies, Inc.	Organic compounds
CA2944755A1 (en)	2014-04-04	2015-10-08	Intra-Cellular Therapies, Inc.	Organic compounds
PL3838274T3 (pl)	2016-01-26	2024-04-02	Intra-Cellular Therapies, Inc.	Pochodna pirydo[3',4':4,5]pirolo[1,2,3-DE]chinoksaliny do zastosowania w leczeniu zaburzeń OUN
DK3407889T3 (da)	2016-03-25	2021-08-09	Intra Cellular Therapies Inc	Organiske forbindelser og deres anvendelse til behandling og forebyggelse af lidelser i centralnervesystemet
EP3436455A4 (de)	2016-03-28	2019-09-04	Intra-Cellular Therapies, Inc.	Neuartige salze und kristalle
US10682354B2 (en)	2016-03-28	2020-06-16	Intra-Cellular Therapies, Inc.	Compositions and methods
US11014925B2 (en)	2016-03-28	2021-05-25	Intra-Cellular Therapies, Inc.	Co-crystals of 1-(4-fluoro-phenyl)-4-((6bR,1OaS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H- pyrido[3′,4′:4,51_pyrrolo [1,2,3-delqcuinoxalin-8-yl)-butan-1-one with nicotinamide or isonicotinamide
EP3525763B1 (de)	2016-10-12	2025-03-05	Intra-Cellular Therapies, Inc.	Amorphe feste dispersionen
WO2018126140A1 (en)	2016-12-29	2018-07-05	Intra-Cellular Therapies, Inc.	Organic compounds
EP3562484B1 (de)	2016-12-29	2021-08-25	Intra-Cellular Therapies, Inc.	Pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalinderivate zur behandlung von erkrankungen des zns
RU2767410C2 (ru)	2017-03-24	2022-03-17	Интра-Селлулар Терапиз, Инк.	Новые композиции и способы
WO2019023062A1 (en)	2017-07-26	2019-01-31	Intra-Cellular Therapies, Inc.	ORGANIC COMPOUNDS
EP3658144B1 (de)	2017-07-26	2022-01-26	Intra-Cellular Therapies, Inc.	Pyridopyrroloquinoxalinverbindungen, deren zusammensetzungen und verwendungen in therapie
CN112040940A (zh)	2018-03-23	2020-12-04	细胞内治疗公司	有机化合物
AU2019280850C1 (en)	2018-06-06	2025-02-13	Intra-Cellular Therapies, Inc.	Novel salts and crystals
EP3801527B1 (de)	2018-06-08	2025-02-19	Intra-Cellular Therapies, Inc.	Anellierte gamma-carboline zur akutbehandlung von angst oder depression
CA3240552A1 (en)	2018-06-11	2019-12-19	Intra-Cellular Therapies, Inc.	Substituted heterocycle fused gamma-carbolines synthesis
US12144808B2 (en)	2018-08-29	2024-11-19	Intra-Cellular Therapies, Inc.	Compositions and methods
WO2020047408A1 (en)	2018-08-31	2020-03-05	Intra-Cellular Therapies, Inc.	Novel methods
BR112021003655A2 (pt)	2018-08-31	2021-05-18	Intra-Cellular Therapies, Inc.	métodos novos
WO2021007245A1 (en)	2019-07-07	2021-01-14	Intra-Cellular Therapies, Inc.	Novel methods
US12414948B2 (en)	2022-05-18	2025-09-16	Intra-Cellular Therapies, Inc.	Methods
CN116925104A (zh) *	2023-07-24	2023-10-24	南开大学	一类噻二唑并嘧啶酮类衍生物及其制备方法和用途

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS5129981B2 (de) *	1973-07-17	1976-08-28
JPS52118494A (en) *	1976-03-31	1977-10-04	Kazuyuki Maekawa	Thiadiazolo322a*pyrimidine derivatives
US4537962A (en) *	1982-02-04	1985-08-27	Farmitalia Carlo Erba, S.P.A.	Substituted 1,3,4-thiadiazolo[3,2-A]pyrimidines and compositions containing them
JPS58177997A (ja) *	1982-04-12	1983-10-18	Dai Ichi Seiyaku Co Ltd	チアジアゾロピリミジノン誘導体
GR80916B (en) *	1983-11-14	1985-03-12	Dow Chemical Co	Method of preparing 1,2,4-triazolo (1,5-a)-pyrimidine-2-sulfonyl chlorides
EP0238059B1 (de) *	1986-03-19	1993-06-16	Kumiai Chemical Industry Co., Ltd.	5H-1,3,4-Thiazol[3,2-a]pyrimidin-5-on-Derivate und diese enthaltende fungizide Zubereitungen
DE3763282D1 (de) *	1986-03-19	1990-07-26	Kumiai Chemical Industry Co	Fungizide zur verwendung in der landwirtschaft und im gartenbau.
DE3786365T2 (de) *	1986-04-07	1993-10-21	Ihara Chemical Ind Co	5H-1,3,4-Thiadiazolo[3,2-a]pyrimidin-5-on-Derivate und diese enthaltende Gartenbau- und landwirtschaftliche Fungizidmittel.
US4872907A (en) *	1988-06-30	1989-10-10	Pre-Melt Systems, Inc.	Metal chip furnace charge apparatus and method

1987
- 1987-03-18 EP EP87103966A patent/EP0238059B1/de not_active Expired - Lifetime
- 1987-03-18 DE DE87103966T patent/DE3786185T2/de not_active Expired - Fee Related
- 1987-03-18 ES ES87103966T patent/ES2058068T3/es not_active Expired - Lifetime
- 1987-03-18 JP JP62062878A patent/JPH07110865B2/ja not_active Expired - Fee Related
- 1987-03-18 ZA ZA871987A patent/ZA871987B/xx unknown
- 1987-03-18 AT AT87103966T patent/ATE90683T1/de not_active IP Right Cessation
- 1987-09-14 US US07/095,672 patent/US4866064A/en not_active Expired - Fee Related
1989
- 1989-08-28 US US07/399,331 patent/US4971971A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
DE3786185T2 (de)	1993-10-21
EP0238059B1 (de)	1993-06-16
JPS6310794A (ja)	1988-01-18
AU581563B2 (en)	1989-02-23
AU7012087A (en)	1987-09-24
JPH07110865B2 (ja)	1995-11-29
ES2058068T3 (es)	1994-11-01
DE3786185D1 (de)	1993-07-22
US4971971A (en)	1990-11-20
EP0238059A2 (de)	1987-09-23
US4866064A (en)	1989-09-12
ATE90683T1 (de)	1993-07-15
EP0238059A3 (en)	1989-01-11

Publication	Publication Date	Title
ZA871987B (en)	1988-05-25	5h-1,3,4-thiadiazole(3,2-a)pyrimidin-5-one derivatives and fungicidal compositions containing the same
GB2087880B (en)	1985-05-01	7-oxo-4-thia-1-azabicyclo(3,2,0)-heptane and 7-oxo-4-thia-1-azabicyclo(3,2,0)hept-2-ene derivatives
EP0192060B1 (de)	1991-09-18	Heterocyclische Verbindungen
MX9702682A (es)	1998-02-28	Pirrolocarbazoles fusionados.
GEP19960641B (en)	1996-11-15	Process for production of [3h]-imidazo[5,1-d]-1,2,3,5-tetrazin-4-one derivatives
MY105344A (en)	1994-09-30	New sulphonyl compounds
MY103241A (en)	1993-05-29	Imidazole and 1,2,4 triazole derivatives
AU5715190A (en)	1990-10-04	Intermediates for the production of podophyllotoxin and related compounds and processes for the preparation and use thereof
EP0641770A4 (de)	1995-06-28	Neue verbindungen mit blutblättchenaggregations hemmender aktivität.
MY105128A (en)	1994-08-30	Bu-3608 derivatives.
MY132057A (en)	2007-09-28	Quinoxalinones, a process for their preparation and their use
ES2013035A6 (es)	1990-04-16	Un metodo para preparar derivados de acilfenol.
HUT49557A (en)	1989-10-30	Process for production of derivatives of cycloprophane
IL111966A0 (en)	1995-03-15	4-Benzoylisoxazole derivatives, their preparation and herbicidal compositions containing them
ES487585A1 (es)	1980-07-01	Procedimiento para la obtencion de n-fenilureas, de efecto herbicida
AU557559B2 (en)	1986-12-24	7 - acylthio-15,16-methylene-3-oxo-17 - pregna-1,4-diene- 21,17-carbolactones
ZA881430B (de)	1988-10-28
EP0282635A3 (de)	1989-11-08	5H-1,3,4-Thiadiazolo[3,2-a]pyrimidin-5-onderivate und diese enthaltende fungizide Zubereitungen
GB2191191A (en)	1987-12-09	Herbicidal 5-amino-3-oxo-4-(substituted--phenyl)-2,3-dihydrothiophene and derivatives thereof
AU6653190A (en)	1991-07-18	Fungicides
GR3001543T3 (en)	1992-11-23	New 2'-substituted-4-deoxythiazolo(5,4-c)rifamycin sv derivatives
AU578335B2 (en)	1988-10-20	N-substituted aziridine-2-carboxylic acid derivatives
IL86665A0 (en)	1988-11-30	Mitomycin analogs
EP0198190A3 (en)	1986-11-26	Compounds having antiplatelet aggregation activity, a process for the preparation thereof and pharmaceutical compositions containing them
PH25608A (en)	1991-08-08	3-amino-tetrahydro-isoquinoline