ZA915193B - Antiandrogenic(3,2-c)pyrazole and(3,2-d)triazole steroids - Google Patents

Antiandrogenic(3,2-c)pyrazole and(3,2-d)triazole steroids

Info

Publication number: ZA915193B
Authority: ZA; South Africa
Prior art keywords: antiandrogenic; steroids; pyrazole; triazole; triazole steroids
Prior art date: 1990-07-04

Application number

ZA915193A

Other languages

English (en)

Inventor

Helmut Hofmeister

Hofmeister Helmut

Dieter Bittler

Bittler Dieter

Horst Michna

Michna Horst

Ursula Habenicht

Habenicht Ursula

Karl-Heinrich Fritzemeier

Fritzemeier Karl-Heinrich

Yukishige Nishino

Nishino Yukishige

Original Assignee

Schering Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-07-04

Filing date

1991-07-04

Publication date

1992-04-29

1991-07-04 Application filed by Schering Ag filed Critical Schering Ag

1992-04-29 Publication of ZA915193B publication Critical patent/ZA915193B/xx

Links

WTKZEGDFNFYCGP-UHFFFAOYSA-N Pyrazole Chemical compound C=1C=NNC=1 WTKZEGDFNFYCGP-UHFFFAOYSA-N 0.000 title 1
230000002280 anti-androgenic effect Effects 0.000 title 1
-1 triazole steroids Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0036—Nitrogen-containing hetero ring
- C07J71/0042—Nitrogen only
- C07J71/0047—Nitrogen only at position 2(3)

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

ZA915193A 1990-07-04 1991-07-04 Antiandrogenic(3,2-c)pyrazole and(3,2-d)triazole steroids ZA915193B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE4021433A DE4021433A1 (de)	1990-07-04	1990-07-04	Antiandrogene mit steroid(3,2-c)pyrazol-struktur

Publications (1)

Publication Number	Publication Date
ZA915193B true ZA915193B (en)	1992-04-29

Family

ID=6409714

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA915193A ZA915193B (en)	1990-07-04	1991-07-04	Antiandrogenic(3,2-c)pyrazole and(3,2-d)triazole steroids

Country Status (14)

Country	Link
US (2)	US5236912A (de)
EP (1)	EP0538312A1 (de)
JP (1)	JPH05508637A (de)
CN (1)	CN1059529A (de)
AU (1)	AU644201B2 (de)
CA (1)	CA2086678A1 (de)
DE (1)	DE4021433A1 (de)
FI (1)	FI925977A0 (de)
HU (1)	HUT64364A (de)
IE (1)	IE912333A1 (de)
IL (1)	IL98724A0 (de)
PT (1)	PT98199A (de)
WO (1)	WO1992000992A1 (de)
ZA (1)	ZA915193B (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5879711A (en) *	1997-11-07	1999-03-09	Sequeira; Joel A.	Stable antiandrogenic gel composition
ES2347027T3 (es)	1998-05-22	2010-10-22	The Board Of Trustees Of The Leland Stanford Junior University	Moleculas bifuncionales y terapias basadas en las mismas.
EP2671507A3 (de)	2005-04-28	2014-02-19	Proteus Digital Health, Inc.	Pharma-Informatiksystem
US9062126B2 (en)	2005-09-16	2015-06-23	Raptor Pharmaceuticals Inc.	Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
US20080051380A1 (en)	2006-08-25	2008-02-28	Auerbach Alan H	Methods and compositions for treating cancer
CA2752373C (en)	2009-02-20	2017-10-10	To-Bbb Holding B.V.	Glutathione-based drug delivery system
IL255113B (en)	2009-05-06	2022-09-01	Laboratory Skin Care Inc	Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same
BR112019001398A2 (pt)	2016-07-29	2019-05-07	Janssen Pharmaceutica Nv	métodos para tratamento de câncer de próstata
CN113024513A (zh) *	2021-03-22	2021-06-25	中国药科大学	新型雄激素受体降解剂、制备方法和医药用途
CN117024499A (zh) *	2023-07-17	2023-11-10	陕西汉江药业集团股份有限公司	在2位引入亚甲基羟基的甾体化合物制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL100550C (de) *	1959-02-16
US3290293A (en) *	1961-12-01	1966-12-06	Merck & Co Inc	4-androsteno-[3, 2-c] pyrazoles
US3280112A (en) *	1963-01-28	1966-10-18	Sterling Drug Inc	Steroido [2, 3-d] triazoles
US4297350A (en) *	1978-10-10	1981-10-27	The Upjohn Company	Male contraceptive steroids and methods of use
US4684636A (en) *	1985-06-24	1987-08-04	Sterling Drug Inc.	Antiandrogenic sulfonylsteroidopyrazoles and processes for preparation method of use and compositions thereof

1990
- 1990-07-04 DE DE4021433A patent/DE4021433A1/de not_active Withdrawn
1991
- 1991-07-03 PT PT98199A patent/PT98199A/pt not_active Application Discontinuation
- 1991-07-04 ZA ZA915193A patent/ZA915193B/xx unknown
- 1991-07-04 HU HU9204180A patent/HUT64364A/hu unknown
- 1991-07-04 CA CA002086678A patent/CA2086678A1/en not_active Abandoned
- 1991-07-04 JP JP91511630A patent/JPH05508637A/ja active Pending
- 1991-07-04 WO PCT/EP1991/001253 patent/WO1992000992A1/de not_active Ceased
- 1991-07-04 EP EP91912518A patent/EP0538312A1/de not_active Withdrawn
- 1991-07-04 CN CN91104041A patent/CN1059529A/zh active Pending
- 1991-07-04 AU AU81880/91A patent/AU644201B2/en not_active Ceased
- 1991-07-04 IL IL98724A patent/IL98724A0/xx unknown
- 1991-07-04 IE IE233391A patent/IE912333A1/en unknown
- 1991-07-05 US US07/725,330 patent/US5236912A/en not_active Expired - Fee Related
1992
- 1992-12-31 FI FI925977A patent/FI925977A0/fi not_active Application Discontinuation
1993
- 1993-04-27 US US08/052,976 patent/US5389624A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
FI925977A7 (fi)	1992-12-31
IL98724A0 (en)	1992-07-15
AU644201B2 (en)	1993-12-02
FI925977A0 (fi)	1992-12-31
US5236912A (en)	1993-08-17
HU9204180D0 (en)	1993-09-28
HUT64364A (en)	1993-12-28
CA2086678A1 (en)	1992-01-05
WO1992000992A1 (de)	1992-01-23
CN1059529A (zh)	1992-03-18
PT98199A (pt)	1992-05-29
AU8188091A (en)	1992-02-04
IE912333A1 (en)	1992-01-15
DE4021433A1 (de)	1992-01-09
US5389624A (en)	1995-02-14
JPH05508637A (ja)	1993-12-02
EP0538312A1 (de)	1993-04-28

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