AR045562A1 - Plaguicidas derivados de alquilaminopirazol sustituido en posicion 5 - Google Patents
Plaguicidas derivados de alquilaminopirazol sustituido en posicion 5Info
- Publication number
- AR045562A1 AR045562A1 ARP040103146A ARP040103146A AR045562A1 AR 045562 A1 AR045562 A1 AR 045562A1 AR P040103146 A ARP040103146 A AR P040103146A AR P040103146 A ARP040103146 A AR P040103146A AR 045562 A1 AR045562 A1 AR 045562A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- halogen
- substituted
- group
- haloalkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Epidemiology (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente se refiere a compuestos, procesos para su preparación, composiciones, su uso para el control de plagas (incluyendo artrópodos y helmintos), y su uso para la preparación de un medicamento veterinario. Reivindicación 1: Un compuesto de fórmula (1) en la cual R1 es CSNH2; W es C-halógeno o N; R2 es H o Cl; R3 es CF3, OCF3 o SF5; Q es alquilo C1-6 o -CH2R7; Z es H, alquilo C1-6, haloalquilo C1-6, alquenilo C3-6, alquinilo C3-6, -(CH2)q-R7, COR8, CO2-alquilo C1-6, S(O)pR8, -CO2- (CH2)R7, CO2-alquenilo C3-6, o CO2-alquinilo C3-6; R4 es H, alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6m, haloalquinilo C2-6, cicloalquilo C3-7, cicloalquilo C3-7-alquilo C1-6-CO2-alquenilo C3-6, CO2-alquinilo C3-6, -CO2-(CH2)q-R7, -CH2R7, - CH2R9, OR7, OR8, COCO2R10 o COCONR10R11; o CO2-alquilo C1-3 no sustituido o sustituido con uno o más radicales seleccionados del grupo integrado por halógeno, alcoxi C1-3 y alquiltio C1-3; o alquilo C1-6 no sustituido o sustituido con uno o más radicales seleccionados del grupo integrado por halógeno, alcoxi C1-6, haloalcoxi C1-6, cicloalquilo C3-7, S(O)pR8 y CO2-alquilo C1-6; A es alquileno C1-6 o haloalquileno C1-6; R5 es alquenilo C2-6, haloalquenilo C2-6, alquinilo C2-6, cicloalquilo C3-6 o -(CH2)qR7; o alquilo C1-6 no sustituido o sustituido con uno o más radicales seleccionados del grupo integrado por halógeno, alcoxi C1-6, haloalcoxi c1-6, cicloalquilo C3-7, S(O)pR8 y CO2-alquilo C1-6; X es F o Cl; R6 es F, Cl, o Br; R7 es fenilo no sustituido o sustituido con uno o más radicales seleccionados del grupo integrado por halógeno, alquilo C1-6-haloalquilo c1-6, alcoxi C1-6, haloalcoxi C1-6, CN, NO2, S(O)pR8, CO2-alquilo C1-6COR8, NR12R13 y OH; R8 es alquilo C1-6 o haloalquilo C1-6; R9 es un radical heteroaromático que tiene 5 o 6 átomos de anillo y 1, 2 o 3 heteroátomos en el anillo seleccionados del grupo integrado por N, O y S, no sustituido o sustituido con uno o más radicales seleccionados del grupo integrado por halógeno, alquilo C1-4, haloalquilo C1-4, alcoxi C1-4, haloalcoxi C1-4, NO2, CN, CO2-alquilo C1-6-S(O)pR8 y OH; R10 y R11 son cada uno independientemente entre sí H o R5; o el radical NR10R11 forma un anillo de 5 a 7 miembros saturado el cual contiene opcionalmente un heteroátomo adicional en el anillo el cual se selecciona de O, S y N, el anillo está no sustituido o sustituido con uno o más radicales seleccionados del grupo integrado por halógeno, alquilo C1-6, haloalquilo C1-6, y CO2-alquilo C1-6;: R12 y R13 son cada uno independientemente entre sí H o alquilo C1-6; m, n, y p son cada uno independientemente entre sí, 0, 1 o 2; y q es 0 o 1; o su sal aceptable para uso plaguicida.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP03019619 | 2003-09-04 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR045562A1 true AR045562A1 (es) | 2005-11-02 |
Family
ID=34259146
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP040103146A AR045562A1 (es) | 2003-09-04 | 2004-09-02 | Plaguicidas derivados de alquilaminopirazol sustituido en posicion 5 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20070072850A1 (es) |
| EP (1) | EP1663985B1 (es) |
| JP (1) | JP4982764B2 (es) |
| KR (1) | KR20060096991A (es) |
| CN (1) | CN100537545C (es) |
| AR (1) | AR045562A1 (es) |
| AT (1) | ATE444955T1 (es) |
| AU (1) | AU2004270341B9 (es) |
| BR (1) | BRPI0414081A (es) |
| CA (1) | CA2536637C (es) |
| DE (1) | DE602004023525D1 (es) |
| ES (1) | ES2332274T3 (es) |
| MX (1) | MXPA06002380A (es) |
| NZ (1) | NZ545657A (es) |
| WO (1) | WO2005023775A1 (es) |
| ZA (1) | ZA200601795B (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7517877B2 (en) * | 2002-03-05 | 2009-04-14 | Merial Limited | 5-substituted-alkylaminopyrazole derivatives as pesticides |
| DK1879869T3 (da) * | 2005-05-07 | 2009-03-02 | Merial Ltd | Fremgangsmåde til fremstiling af precursorer for 5-akylthioalkylamino-1-phenylpyrazoler |
| CN104204057B (zh) * | 2012-03-28 | 2016-10-05 | 朗盛德国有限责任公司 | 噻苯咪唑和含碘杀真菌剂的稳定组合物 |
| TWI579274B (zh) * | 2012-04-20 | 2017-04-21 | 龍馬躍公司 | 製備１－芳基－５－烷基吡唑化合物的改良方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4005213A (en) * | 1968-12-21 | 1977-01-25 | Schering Aktiengesellschaft | 2,5-Substituted-1,3,4-thiadiazoles as fungicides |
| US5629335A (en) * | 1995-04-07 | 1997-05-13 | Rhone-Poulenc Inc. | Pesticidal 1-arylpyrazole-3-carboximidothioic acid esters |
| DE19650197A1 (de) * | 1996-12-04 | 1998-06-10 | Bayer Ag | 3-Thiocarbamoylpyrazol-Derivate |
| US6350771B1 (en) * | 1996-12-24 | 2002-02-26 | Rhone-Poulenc, Inc. | Pesticidal 1-arylpyrazoles |
| DE19824487A1 (de) * | 1998-06-02 | 1999-12-09 | Bayer Ag | Substituierte 3-Thiocarbamoylpyrazole |
| DE19853560A1 (de) * | 1998-11-20 | 2000-05-25 | Bayer Ag | Verfahren zur Herstellung von 5-Amino-3-(thio)carbamoylpyrazolen |
| AR021608A1 (es) * | 1998-12-11 | 2002-07-31 | Merial Ltd | Represion de artropodos en animales |
| AU2001275898A1 (en) * | 2000-07-12 | 2002-01-21 | Ocapco, Llc | Avermectin pesticide with an organosilicone surfactant |
-
2004
- 2004-08-21 BR BRPI0414081-8A patent/BRPI0414081A/pt not_active Application Discontinuation
- 2004-08-21 US US10/570,136 patent/US20070072850A1/en not_active Abandoned
- 2004-08-21 EP EP04764358A patent/EP1663985B1/en not_active Expired - Lifetime
- 2004-08-21 DE DE602004023525T patent/DE602004023525D1/de not_active Expired - Lifetime
- 2004-08-21 AT AT04764358T patent/ATE444955T1/de not_active IP Right Cessation
- 2004-08-21 MX MXPA06002380A patent/MXPA06002380A/es active IP Right Grant
- 2004-08-21 CN CNB2004800255503A patent/CN100537545C/zh not_active Expired - Fee Related
- 2004-08-21 ES ES04764358T patent/ES2332274T3/es not_active Expired - Lifetime
- 2004-08-21 CA CA2536637A patent/CA2536637C/en not_active Expired - Fee Related
- 2004-08-21 AU AU2004270341A patent/AU2004270341B9/en not_active Ceased
- 2004-08-21 NZ NZ545657A patent/NZ545657A/en not_active IP Right Cessation
- 2004-08-21 JP JP2006525066A patent/JP4982764B2/ja not_active Expired - Fee Related
- 2004-08-21 KR KR1020067004574A patent/KR20060096991A/ko not_active Ceased
- 2004-08-21 WO PCT/EP2004/009376 patent/WO2005023775A1/en not_active Ceased
- 2004-09-02 AR ARP040103146A patent/AR045562A1/es active IP Right Grant
-
2006
- 2006-03-02 ZA ZA200601795A patent/ZA200601795B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP1663985B1 (en) | 2009-10-07 |
| JP2007504184A (ja) | 2007-03-01 |
| BRPI0414081A (pt) | 2006-10-24 |
| KR20060096991A (ko) | 2006-09-13 |
| EP1663985A1 (en) | 2006-06-07 |
| AU2004270341A1 (en) | 2005-03-17 |
| CN100537545C (zh) | 2009-09-09 |
| US20070072850A1 (en) | 2007-03-29 |
| ATE444955T1 (de) | 2009-10-15 |
| AU2004270341B9 (en) | 2011-06-30 |
| WO2005023775A1 (en) | 2005-03-17 |
| JP4982764B2 (ja) | 2012-07-25 |
| NZ545657A (en) | 2010-01-29 |
| MXPA06002380A (es) | 2006-06-20 |
| CA2536637C (en) | 2011-12-06 |
| ZA200601795B (en) | 2007-05-30 |
| CN1845903A (zh) | 2006-10-11 |
| ES2332274T3 (es) | 2010-02-01 |
| DE602004023525D1 (de) | 2009-11-19 |
| HK1099746A1 (zh) | 2007-08-24 |
| AU2004270341B2 (en) | 2011-04-28 |
| CA2536637A1 (en) | 2005-03-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant, registration |