AR061967A1 - Ester isopropilico del acido 4-[6-(6-metanosulfonil-2-metil-piridin-3-il-amino)-5-metil-pirimidin-4-iloxi]-piperidin-i-carboxilico, composicion farmaceutica que lo comprende y un metodo de preparacion de la misma y el uso de este compuesto para el tratamiento de trastornos metabolicos - Google Patents

Ester isopropilico del acido 4-[6-(6-metanosulfonil-2-metil-piridin-3-il-amino)-5-metil-pirimidin-4-iloxi]-piperidin-i-carboxilico, composicion farmaceutica que lo comprende y un metodo de preparacion de la misma y el uso de este compuesto para el tratamiento de trastornos metabolicos

Info

Publication number: AR061967A1
Authority: AR; Argentina
Prior art keywords: methyl; treatment; metabolic disorders; pyrimidin; pharmaceutical composition
Prior art date: 2006-07-06

Application number

ARP070103026A

Other languages

English (en)

Spanish (es)

Original Assignee

Arena Pharm Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-07-06

Filing date

2007-07-06

Publication date

2008-08-10

2007-07-06 Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc

2008-08-10 Publication of AR061967A1 publication Critical patent/AR061967A1/es

Links

208000030159 metabolic disease Diseases 0.000 title abstract 3
238000000034 method Methods 0.000 title abstract 2
239000008194 pharmaceutical composition Substances 0.000 title abstract 2
239000002253 acid Substances 0.000 title 1
239000002131 composite material Substances 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 2
208000008589 Obesity Diseases 0.000 abstract 1
206010012601 diabetes mellitus Diseases 0.000 abstract 1
239000003814 drug Substances 0.000 abstract 1
230000004153 glucose metabolism Effects 0.000 abstract 1
150000004677 hydrates Chemical class 0.000 abstract 1
238000004519 manufacturing process Methods 0.000 abstract 1
235000020824 obesity Nutrition 0.000 abstract 1
BTVNNMSDLVBWRW-UHFFFAOYSA-N propan-2-yl 4-[5-methyl-6-[(2-methyl-6-methylsulfonylpyridin-3-yl)amino]pyrimidin-4-yl]oxypiperidine-1-carboxylate Chemical compound C1CN(C(=O)OC(C)C)CCC1OC1=NC=NC(NC=2C(=NC(=CC=2)S(C)(=O)=O)C)=C1C BTVNNMSDLVBWRW-UHFFFAOYSA-N 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
239000012453 solvate Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/12—Ophthalmic agents for cataracts
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Diabetes (AREA)
Obesity (AREA)
Cardiology (AREA)
Hematology (AREA)
Endocrinology (AREA)
Heart & Thoracic Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Rheumatology (AREA)
Ophthalmology & Optometry (AREA)
Orthopedic Medicine & Surgery (AREA)
Reproductive Health (AREA)
Urology & Nephrology (AREA)
Emergency Medicine (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Gynecology & Obstetrics (AREA)
Neurology (AREA)
Child & Adolescent Psychology (AREA)
Vascular Medicine (AREA)
Hospice & Palliative Care (AREA)
Dermatology (AREA)
Immunology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

ARP070103026A 2006-07-06 2007-07-06 Ester isopropilico del acido 4-[6-(6-metanosulfonil-2-metil-piridin-3-il-amino)-5-metil-pirimidin-4-iloxi]-piperidin-i-carboxilico, composicion farmaceutica que lo comprende y un metodo de preparacion de la misma y el uso de este compuesto para el tratamiento de trastornos metabolicos AR061967A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US81950006P	2006-07-06	2006-07-06

Publications (1)

Publication Number	Publication Date
AR061967A1 true AR061967A1 (es)	2008-08-10

Family

ID=38707392

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ARP070103026A AR061967A1 (es)	2006-07-06	2007-07-06	Ester isopropilico del acido 4-[6-(6-metanosulfonil-2-metil-piridin-3-il-amino)-5-metil-pirimidin-4-iloxi]-piperidin-i-carboxilico, composicion farmaceutica que lo comprende y un metodo de preparacion de la misma y el uso de este compuesto para el tratamiento de trastornos metabolicos

Country Status (26)

Country	Link
US (1)	US20100004272A1 (2)
EP (1)	EP2049523A1 (2)
JP (1)	JP2009542702A (2)
KR (1)	KR20090024779A (2)
CN (1)	CN101484440A (2)
AR (1)	AR061967A1 (2)
AU (1)	AU2007269577A1 (2)
BR (1)	BRPI0714006A2 (2)
CA (1)	CA2656520A1 (2)
CL (1)	CL2007001972A1 (2)
CO (1)	CO6160320A2 (2)
CR (1)	CR10538A (2)
EA (1)	EA015343B1 (2)
EC (1)	ECSP099036A (2)
GT (1)	GT200800305A (2)
IL (1)	IL195819A0 (2)
MA (1)	MA30601B1 (2)
MX (1)	MX2008016251A (2)
NI (1)	NI200800328A (2)
NO (1)	NO20090590L (2)
PE (1)	PE20080737A1 (2)
TN (1)	TNSN08534A1 (2)
TW (1)	TW200811140A (2)
UY (1)	UY30466A1 (2)
WO (1)	WO2008005576A1 (2)
ZA (1)	ZA200900051B (2)

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2007
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- 2007-07-04 PE PE2007000858A patent/PE20080737A1/es not_active Application Discontinuation
- 2007-07-05 MX MX2008016251A patent/MX2008016251A/es not_active Application Discontinuation
- 2007-07-05 EP EP07810288A patent/EP2049523A1/en not_active Withdrawn
- 2007-07-05 AU AU2007269577A patent/AU2007269577A1/en not_active Withdrawn
- 2007-07-05 JP JP2009518404A patent/JP2009542702A/ja not_active Withdrawn
- 2007-07-05 CN CNA2007800249135A patent/CN101484440A/zh not_active Withdrawn
- 2007-07-05 CA CA002656520A patent/CA2656520A1/en not_active Abandoned
- 2007-07-05 WO PCT/US2007/015681 patent/WO2008005576A1/en not_active Ceased
- 2007-07-05 CL CL200701972A patent/CL2007001972A1/es unknown
- 2007-07-05 BR BRPI0714006-1A patent/BRPI0714006A2/pt not_active IP Right Cessation
- 2007-07-05 KR KR1020097000109A patent/KR20090024779A/ko not_active Withdrawn
- 2007-07-05 US US12/307,545 patent/US20100004272A1/en not_active Abandoned
- 2007-07-05 EA EA200970090A patent/EA015343B1/ru not_active IP Right Cessation
- 2007-07-06 AR ARP070103026A patent/AR061967A1/es unknown
- 2007-07-06 UY UY30466A patent/UY30466A1/es unknown
2008
- 2008-12-09 IL IL195819A patent/IL195819A0/en unknown
- 2008-12-15 NI NI200800328A patent/NI200800328A/es unknown
- 2008-12-19 CR CR10538A patent/CR10538A/es not_active Application Discontinuation
- 2008-12-24 CO CO08136751A patent/CO6160320A2/es unknown
- 2008-12-25 TN TNP2008000534A patent/TNSN08534A1/en unknown
- 2008-12-29 GT GT200800305A patent/GT200800305A/es unknown
2009
- 2009-01-05 ZA ZA200900051A patent/ZA200900051B/xx unknown
- 2009-01-06 EC EC2009009036A patent/ECSP099036A/es unknown
- 2009-01-27 MA MA31590A patent/MA30601B1/fr unknown
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AU2007269577A1 (en)	2008-01-10
CR10538A (es)	2009-01-27
EP2049523A1 (en)	2009-04-22
NO20090590L (no)	2009-02-06
ZA200900051B (en)	2010-01-27
CN101484440A (zh)	2009-07-15
TW200811140A (en)	2008-03-01
UY30466A1 (es)	2008-02-29
BRPI0714006A2 (pt)	2012-12-18
KR20090024779A (ko)	2009-03-09
MX2008016251A (es)	2009-02-25
GT200800305A (es)	2009-04-25
CA2656520A1 (en)	2008-01-10
WO2008005576A1 (en)	2008-01-10
EA200970090A1 (ru)	2009-06-30
IL195819A0 (en)	2009-09-22
EA015343B1 (ru)	2011-06-30
ECSP099036A (es)	2009-02-27
CL2007001972A1 (es)	2008-04-04
JP2009542702A (ja)	2009-12-03
NI200800328A (es)	2010-01-07
MA30601B1 (fr)	2009-07-01
TNSN08534A1 (en)	2010-04-14
US20100004272A1 (en)	2010-01-07
CO6160320A2 (es)	2010-05-20
PE20080737A1 (es)	2008-06-13

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Publication	Publication Date	Title
AR061967A1 (es)	2008-08-10	Ester isopropilico del acido 4-[6-(6-metanosulfonil-2-metil-piridin-3-il-amino)-5-metil-pirimidin-4-iloxi]-piperidin-i-carboxilico, composicion farmaceutica que lo comprende y un metodo de preparacion de la misma y el uso de este compuesto para el tratamiento de trastornos metabolicos
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