AR102995A1 - USE OF SIGMA RECEIVER LIGANDS IN OSTEOARTRITIS - Google Patents
USE OF SIGMA RECEIVER LIGANDS IN OSTEOARTRITISInfo
- Publication number
- AR102995A1 AR102995A1 ARP150104064A ARP150104064A AR102995A1 AR 102995 A1 AR102995 A1 AR 102995A1 AR P150104064 A ARP150104064 A AR P150104064A AR P150104064 A ARP150104064 A AR P150104064A AR 102995 A1 AR102995 A1 AR 102995A1
- Authority
- AR
- Argentina
- Prior art keywords
- osteoartritis
- sigma receiver
- ligands
- sigma
- receiver ligands
- Prior art date
Links
- 239000003446 ligand Substances 0.000 title 1
- 201000008482 osteoarthritis Diseases 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000000144 pharmacologic effect Effects 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 108010085082 sigma receptors Proteins 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente se refiere a compuestos de fórmula (1) o fórmula (2) con actividad farmacológica contra el receptor sigma, para su uso en el tratamiento o la prevención de la osteoartritis y el dolor debido a la osteoartritis.This refers to compounds of formula (1) or formula (2) with pharmacological activity against the sigma receptor, for use in the treatment or prevention of osteoarthritis and pain due to osteoarthritis.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14382519 | 2014-12-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR102995A1 true AR102995A1 (en) | 2017-04-05 |
Family
ID=52146389
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP150104064A AR102995A1 (en) | 2014-12-15 | 2015-12-14 | USE OF SIGMA RECEIVER LIGANDS IN OSTEOARTRITIS |
Country Status (1)
| Country | Link |
|---|---|
| AR (1) | AR102995A1 (en) |
-
2015
- 2015-12-14 AR ARP150104064A patent/AR102995A1/en unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |